EA014840B1 - Комбинации пиримидинсодержащего nnrti с ингибиторами обратной транскриптазы - Google Patents

Комбинации пиримидинсодержащего nnrti с ингибиторами обратной транскриптазы Download PDF

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Publication number: EA014840B1
Authority: EA; Eurasian Patent Office
Prior art keywords: tms278; reverse transcriptase; combination; hiv; transcriptase inhibitor
Prior art date: 2003-09-03

Application number

EA200600522A

Other languages

English (en)

Russian (ru)

Other versions

EA200600522A1 (ru

Inventor

Пол Стоффелс

Original Assignee

Тиботек Фармасьютикалз Лтд.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-09-03

Filing date

2004-09-03

Publication date

2011-02-28

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43778148&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA014840(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2004-09-03 Application filed by Тиботек Фармасьютикалз Лтд. filed Critical Тиботек Фармасьютикалз Лтд.

2004-09-03 Priority claimed from PCT/EP2004/052028 external-priority patent/WO2005021001A1/en

2006-08-25 Publication of EA200600522A1 publication Critical patent/EA200600522A1/ru

2011-02-28 Publication of EA014840B1 publication Critical patent/EA014840B1/ru

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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine

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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

EA200600522A 2003-09-03 2004-09-03 Комбинации пиримидинсодержащего nnrti с ингибиторами обратной транскриптазы EA014840B1 (ru)

Applications Claiming Priority (7)

Application Number	Priority Date	Filing Date	Title
US49977103P	2003-09-03	2003-09-03
EP03103275		2003-09-03
EP03103319		2003-09-08
EP03103335		2003-09-10
EP03103668		2003-10-02
US50848603P	2003-10-03	2003-10-03
PCT/EP2004/052028 WO2005021001A1 (en)	2003-09-03	2004-09-03	Combinations of a pyrimidine containing nnrti with rt inhibitors

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EA200600522A1 EA200600522A1 (ru)	2006-08-25
EA014840B1 true EA014840B1 (ru)	2011-02-28

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KR (2)	KR101539245B1 (da)
CN (1)	CN102319433A (da)
DK (1)	DK1663240T4 (da)
EA (1)	EA014840B1 (da)
ES (1)	ES2542017T5 (da)
HU (1)	HUE025576T2 (da)
PT (1)	PT1663240E (da)
SI (1)	SI1663240T2 (da)
TW (1)	TWI365744B (da)

Citations (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO2003016306A1 (en) *	2001-08-13	2003-02-27	Janssen Pharmaceutica N.V.	Hiv inhibiting pyrimidines derivatives

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- 2004-09-03 ES ES04787096T patent/ES2542017T5/es not_active Expired - Lifetime
- 2004-09-03 KR KR1020117025799A patent/KR101539245B1/ko not_active Expired - Lifetime
- 2004-09-03 KR KR1020137024817A patent/KR101638999B1/ko not_active Expired - Lifetime
- 2004-09-03 SI SI200432257T patent/SI1663240T2/sl unknown
- 2004-09-03 EA EA200600522A patent/EA014840B1/ru active Protection Beyond IP Right Term
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- 2004-09-03 HU HUE04787096A patent/HUE025576T2/en unknown
- 2004-09-03 CN CN2011102800883A patent/CN102319433A/zh active Pending
- 2004-09-03 DK DK04787096.9T patent/DK1663240T4/da active

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO2003016306A1 (en) *	2001-08-13	2003-02-27	Janssen Pharmaceutica N.V.	Hiv inhibiting pyrimidines derivatives

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GILEAD SCIENCES INC.: "Gilead initiates study 934, a 48-week clinical trial evaluating VireadTM and EmtrivaTM versus CombivirTM" INTERNET ARTICLE, 'Online! 11 August 2003 (2003-08-11), XP002314669 Retrieved from the Internet: URL:http://www.gilead.com/wt/sec/pr_106063 1111> 'retrieved on 2005-01-24! page 1, paragraph 1 *
PAVIA A.T.: "Abacavir/Lamivudine in Combination with Efavirenz, Amprenavir/Ritonavir or Stavudine" INTERNET ARTICLE, 'Online! 9 July 2002 (2002-07-09), XP002274550 Retrieved from the Internet: URL:http://www.thebody.com/confs/aids2002/pavia5.html> 'retrieved on 2004-03-23! page 1, second paragraph, page 2, second and third paragraphs *
SQUIRES K.E.: "An introduction to nucleoside and nucleotide analogues." ANTIVIRAL THERAPY. 2001, vol. 6 Suppl 3, 2001, pages 1-14, XP009042950 ISSN: 1359-6535 pages 4 and 5, table 2 *
YOUNG B.: "Can Abacavir be given Once-a Day?" INTERNET ARTICLE, 'Online! 16 September 2003 (2003-09-16), XP002274551 Retrieved from the Internet: URL:http://www.thebody.com/confs/icaac2003 /young3.html> 'retrieved on 2004-03-23! page 1, last paragraph - page 2, second paragraph *

Also Published As

Publication number	Publication date
KR101539245B1 (ko)	2015-07-27
DK1663240T4 (da)	2023-04-17
TWI365744B (en)	2012-06-11
SI1663240T2 (sl)	2023-05-31
KR20130127515A (ko)	2013-11-22
EA200600522A1 (ru)	2006-08-25
ES2542017T5 (es)	2023-06-15
SI1663240T1 (sl)	2015-10-30
HUE025576T2 (en)	2016-04-28
KR20110132475A (ko)	2011-12-07
PT1663240E (pt)	2015-09-01
DK1663240T3 (da)	2015-07-20
ES2542017T3 (es)	2015-07-29
KR101638999B1 (ko)	2016-07-12
TW200524612A (en)	2005-08-01
CN102319433A (zh)	2012-01-18

Legal Events

Date	Code	Title
2014-08-29	ND4A	Extension of term of a eurasian patent
2015-01-30	TC4A	Change in name of a patent proprietor in a eurasian patent
2016-01-29	PC4A	Registration of transfer of a eurasian patent by assignment
2017-11-30	ND4A	Extension of term of a eurasian patent

Publication	Publication Date	Title
US20220008417A1 (en)	2022-01-13	Combinations of a pyrimidine containing nnrti with rt inhibitors
EP1159005B1 (en)	2003-11-12	Pharmaceutical combination of antiviral agents
EA014840B1 (ru)	2011-02-28	Комбинации пиримидинсодержащего nnrti с ингибиторами обратной транскриптазы
HK1092698B (en)	2015-10-16	Combinations of a pyrimidine containing nnrti with rt inhibitors
HK1165277A (en)	2012-10-05	Combinations of a pyrimidine containing nnrti with rt inhibitors
ZA200601820B (en)	2007-07-25	Combinations of a pyrimidine containing NNRTI with RT inhibitors