EP0712493A4 - METHOD FOR THE PREPARATION AND SELECTION OF NON-PEPTIDE COMPOUNDS FOR PHARMACOLOGICAL USE FROM A UNIVERSAL LIBRARY OF ELEMENTS WITH VARIOUS STRUCTURES - Google Patents
METHOD FOR THE PREPARATION AND SELECTION OF NON-PEPTIDE COMPOUNDS FOR PHARMACOLOGICAL USE FROM A UNIVERSAL LIBRARY OF ELEMENTS WITH VARIOUS STRUCTURESInfo
- Publication number
- EP0712493A4 EP0712493A4 EP94923427A EP94923427A EP0712493A4 EP 0712493 A4 EP0712493 A4 EP 0712493A4 EP 94923427 A EP94923427 A EP 94923427A EP 94923427 A EP94923427 A EP 94923427A EP 0712493 A4 EP0712493 A4 EP 0712493A4
- Authority
- EP
- European Patent Office
- Prior art keywords
- selection
- preparation
- elements
- various structures
- peptide compounds
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C279/00—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
- C07C279/04—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to acyclic carbon atoms of a carbon skeleton
- C07C279/08—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to acyclic carbon atoms of a carbon skeleton being further substituted by singly-bound oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C65/00—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
- C07C65/21—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing ether groups, groups, groups, or groups
- C07C65/24—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing ether groups, groups, groups, or groups polycyclic
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US10107493A | 1993-08-03 | 1993-08-03 | |
| US101074 | 1993-08-03 | ||
| US23954294A | 1994-05-08 | 1994-05-08 | |
| US239542 | 1994-05-08 | ||
| PCT/US1994/007780 WO1995004277A1 (en) | 1993-08-03 | 1994-07-07 | A method for preparing and selecting pharmaceutically useful non-peptide compounds from a structurally diverse universal library |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| EP0712493A1 EP0712493A1 (en) | 1996-05-22 |
| EP0712493A4 true EP0712493A4 (en) | 1997-01-15 |
Family
ID=26797874
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EP94923427A Withdrawn EP0712493A4 (en) | 1993-08-03 | 1994-07-07 | METHOD FOR THE PREPARATION AND SELECTION OF NON-PEPTIDE COMPOUNDS FOR PHARMACOLOGICAL USE FROM A UNIVERSAL LIBRARY OF ELEMENTS WITH VARIOUS STRUCTURES |
Country Status (6)
| Country | Link |
|---|---|
| EP (1) | EP0712493A4 (en) |
| JP (1) | JPH09504511A (en) |
| AU (1) | AU7329394A (en) |
| CA (1) | CA2168886A1 (en) |
| PE (1) | PE14895A1 (en) |
| WO (1) | WO1995004277A1 (en) |
Families Citing this family (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5712171A (en) | 1995-01-20 | 1998-01-27 | Arqule, Inc. | Method of generating a plurality of chemical compounds in a spatially arranged array |
| US5811241A (en) * | 1995-09-13 | 1998-09-22 | Cortech, Inc. | Method for preparing and identifying N-substitued 1,4-piperazines and N-substituted 1,4-piperazinediones |
| US5874443A (en) * | 1995-10-19 | 1999-02-23 | Trega Biosciences, Inc. | Isoquinoline derivatives and isoquinoline combinatorial libraries |
| US5840500A (en) * | 1996-07-11 | 1998-11-24 | Trega Biosciences, Inc. | Quinoline derivatives and quinoline combinatorial libraries |
| GB9616563D0 (en) * | 1996-08-07 | 1996-09-25 | Oxford Asymmetry Ltd | Compounds and methods |
| US5916899A (en) * | 1996-10-18 | 1999-06-29 | Trega Biosciences, Inc. | Isoquinoline derivatives and isoquinoline combinatorial libraries |
| US6893815B1 (en) * | 1997-06-30 | 2005-05-17 | Isis Pharmaceuticals, Inc. | Nucleobase heterocyclic combinatorialization |
| US6080587A (en) * | 1998-01-23 | 2000-06-27 | Eli Lilly And Company | Method for preparing and selecting pharmaceutically useful sulfur-bridged bi- and triaromatic ring compounds from a structurally diverse universal library |
| US6534503B1 (en) | 1998-04-28 | 2003-03-18 | Lion Bioscience Ag | Melanocortin receptor-3 ligands to treat sexual dysfunction |
| US6284735B1 (en) | 1998-04-28 | 2001-09-04 | Lion Bioscience Ag | HP-3228 and related peptides to treat sexual dysfunction |
| US6127381A (en) | 1998-04-28 | 2000-10-03 | Basu; Amaresh | Isoquinoline compound melanocortin receptor ligands and methods of using same |
| EP1085895A1 (en) * | 1998-06-08 | 2001-03-28 | Advanced Medicine, Inc. | Bradykinin antagonists |
| ES2639020T3 (en) | 1998-11-27 | 2017-10-25 | Ucb Pharma S.A. | Compositions and methods to increase bone substance mineralization |
| US20040009535A1 (en) | 1998-11-27 | 2004-01-15 | Celltech R&D, Inc. | Compositions and methods for increasing bone mineralization |
| WO2000056724A1 (en) * | 1999-03-22 | 2000-09-28 | The Board Of Governors For Higher Education, State Of Rhode Island And Providence Plantations | Oxazole and thiazole combinatorial libraries |
| US6864235B1 (en) | 1999-04-01 | 2005-03-08 | Eva A. Turley | Compositions and methods for treating cellular response to injury and other proliferating cell disorders regulated by hyaladherin and hyaluronans |
| US6911429B2 (en) | 1999-04-01 | 2005-06-28 | Transition Therapeutics Inc. | Compositions and methods for treating cellular response to injury and other proliferating cell disorders regulated by hyaladherin and hyaluronans |
| US7507542B2 (en) | 2001-05-08 | 2009-03-24 | Ucb Sa | Method for regulating immune function using the FOXP3 protein |
| AU2003252140A1 (en) * | 2002-07-24 | 2004-02-09 | Janssen Pharmaceutica N.V. | Acetylenic compounds useful in treating inflammatory disorders |
| EP1572976B1 (en) | 2002-11-21 | 2010-09-15 | Celltech R & D, Inc. | Modulating immune responses |
| US7022703B2 (en) | 2003-07-24 | 2006-04-04 | Janssen Pharmaceutica, N.V. | Acetylenic compound useful in treating inflammatory disorders |
| EP2257536A4 (en) | 2008-02-14 | 2011-03-23 | Amira Pharmaceuticals Inc | Cyclic diaryl ether as antagonists of prostaglandin d2 receptors |
| US8426449B2 (en) | 2008-04-02 | 2013-04-23 | Panmira Pharmaceuticals, Llc | Aminoalkylphenyl antagonists of prostaglandin D2 receptors |
| US8383654B2 (en) | 2008-11-17 | 2013-02-26 | Panmira Pharmaceuticals, Llc | Heterocyclic antagonists of prostaglandin D2 receptors |
| GB0903482D0 (en) * | 2009-02-27 | 2009-04-08 | Ucl Business Plc | New compounds |
| US20240374761A1 (en) | 2021-05-05 | 2024-11-14 | Radius Pharmaceuticals, Inc. | Animal model having homologous recombination of mouse pth1 receptor |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5218124A (en) * | 1989-10-27 | 1993-06-08 | American Home Products Corporation | Substituted benzoylbenzene-, biphenyl- and 2-oxazole-alkanoic acid derivatives as inhibitors of pla2 and lipoxygenase |
| US5250548A (en) * | 1990-09-10 | 1993-10-05 | Abbott Laboratories | Angiotensin II receptor antagonists |
-
1994
- 1994-07-07 EP EP94923427A patent/EP0712493A4/en not_active Withdrawn
- 1994-07-07 CA CA002168886A patent/CA2168886A1/en not_active Abandoned
- 1994-07-07 WO PCT/US1994/007780 patent/WO1995004277A1/en not_active Ceased
- 1994-07-07 AU AU73293/94A patent/AU7329394A/en not_active Abandoned
- 1994-07-07 JP JP7505836A patent/JPH09504511A/en active Pending
- 1994-08-03 PE PE1994247887A patent/PE14895A1/en not_active Application Discontinuation
Non-Patent Citations (2)
| Title |
|---|
| No further relevant documents disclosed * |
| See also references of WO9504277A1 * |
Also Published As
| Publication number | Publication date |
|---|---|
| WO1995004277A1 (en) | 1995-02-09 |
| PE14895A1 (en) | 1995-06-08 |
| AU7329394A (en) | 1995-02-28 |
| CA2168886A1 (en) | 1995-02-09 |
| JPH09504511A (en) | 1997-05-06 |
| EP0712493A1 (en) | 1996-05-22 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PUAI | Public reference made under article 153(3) epc to a published international application that has entered the european phase |
Free format text: ORIGINAL CODE: 0009012 |
|
| 17P | Request for examination filed |
Effective date: 19960221 |
|
| AK | Designated contracting states |
Kind code of ref document: A1 Designated state(s): AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE |
|
| RIN1 | Information on inventor provided before grant (corrected) |
Inventor name: HEDIGER, MARK, EDWARD Inventor name: HANGAUER, DAVID, GARRY, JR. Inventor name: WHITESIDES, GEORGE, MCCLELLAND Inventor name: PAVIA, MICHAEL, RAYMOND |
|
| A4 | Supplementary search report drawn up and despatched |
Effective date: 19961202 |
|
| AK | Designated contracting states |
Kind code of ref document: A4 Designated state(s): AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE |
|
| 17Q | First examination report despatched |
Effective date: 19991118 |
|
| STAA | Information on the status of an ep patent application or granted ep patent |
Free format text: STATUS: THE APPLICATION IS DEEMED TO BE WITHDRAWN |
|
| 18D | Application deemed to be withdrawn |
Effective date: 20001104 |