ES373698A1 - Un procedimiento para la preparacion de 5-nr1r2-6-cloro - 1h-imidazo (4,5-b) pirazin-2-onas. - Google Patents

Un procedimiento para la preparacion de 5-nr1r2-6-cloro - 1h-imidazo (4,5-b) pirazin-2-onas.

Info

Publication number
ES373698A1
ES373698A1 ES373698A ES373698A ES373698A1 ES 373698 A1 ES373698 A1 ES 373698A1 ES 373698 A ES373698 A ES 373698A ES 373698 A ES373698 A ES 373698A ES 373698 A1 ES373698 A1 ES 373698A1
Authority
ES
Spain
Prior art keywords
general formula
hydrogen atom
amino
alkyl
diamino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES373698A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Publication of ES373698A1 publication Critical patent/ES373698A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/10Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/14Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D241/24Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D241/26Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with nitrogen atoms directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
ES373698A 1968-11-20 1969-11-19 Un procedimiento para la preparacion de 5-nr1r2-6-cloro - 1h-imidazo (4,5-b) pirazin-2-onas. Expired ES373698A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US77747968A 1968-11-20 1968-11-20

Publications (1)

Publication Number Publication Date
ES373698A1 true ES373698A1 (es) 1972-02-01

Family

ID=25110373

Family Applications (1)

Application Number Title Priority Date Filing Date
ES373698A Expired ES373698A1 (es) 1968-11-20 1969-11-19 Un procedimiento para la preparacion de 5-nr1r2-6-cloro - 1h-imidazo (4,5-b) pirazin-2-onas.

Country Status (8)

Country Link
US (1) US3549633A (es)
AT (1) AT291250B (es)
BR (1) BR6914169D0 (es)
CH (1) CH518957A (es)
ES (1) ES373698A1 (es)
FR (1) FR2070653A1 (es)
GB (1) GB1242625A (es)
NL (1) NL6915958A (es)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4053577A (en) * 1972-02-18 1977-10-11 Tioxide Group Limited Process for the gaseous phase production of metal oxide particles
GR74944B (es) * 1980-07-02 1984-07-12 Merck & Co Inc
BR112013011868A2 (pt) * 2010-11-16 2016-08-23 Acetylon Pharmaceuticals Inc compostos de pirimidina hidróxi amida como inibidores da proteína desacetilase, composição farmacêutica e uso dos referidos compostos
ES2929576T3 (es) 2013-10-08 2022-11-30 Acetylon Pharmaceuticals Inc Combinaciones de inhibidores de histona deacetilasa 6 y el inhibidor de Her2 lapatinib para el uso en el tratamiento del cáncer de mama
WO2015054474A1 (en) 2013-10-10 2015-04-16 Acetylon Pharmaceuticals, Inc. Pyrimidine hydroxy amide compounds as histone deacetylase inhibitors
US10660890B2 (en) 2013-10-24 2020-05-26 National Institutes Of Health (Nih), U.S. Dept. Of Health And Human Services (Dhhs), U.S. Government Nih Division Of Extramural Inventions And Technology Resources (Deitr) Treatment of polycystic diseases with an HDAC6 inhibitor
CR20160308A (es) 2013-12-03 2016-11-08 Acetylon Pharmaceuticals Inc Combinaciones de inhibidores de histona deacetilasa y farmacos inmunomoduladores
US9464073B2 (en) 2014-02-26 2016-10-11 Acetylon Pharmaceuticals, Inc. Pyrimidine hydroxy amide compounds as HDAC6 selective inhibitors
SG11201700094TA (en) 2014-07-07 2017-02-27 Acetylon Pharmaceuticals Inc Treatment of leukemia with histone deacetylase inhibitors
US9937174B2 (en) 2014-12-05 2018-04-10 University of Modena and Reggio Emilia Combinations of histone deacetylase inhibitors and bendamustine
US10272084B2 (en) 2015-06-01 2019-04-30 Regenacy Pharmaceuticals, Llc Histone deacetylase 6 selective inhibitors for the treatment of cisplatin-induced peripheral neuropathy
EP3445364A4 (en) 2016-04-19 2019-11-27 Acetylon Pharmaceuticals, Inc. HDAC INHIBITORS, ONLY OR IN COMBINATION WITH BTK INHIBITORS, FOR THE TREATMENT OF CHRONIC LYMPHOCYTIC LEUKEMIA

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE651729A (es) * 1962-10-30 1965-02-12
US3361748A (en) * 1965-11-22 1968-01-02 Merck & Co Inc Process for the preparation of pteridinones

Also Published As

Publication number Publication date
GB1242625A (en) 1971-08-11
US3549633A (en) 1970-12-22
CH518957A (de) 1972-02-15
NL6915958A (es) 1970-05-22
BR6914169D0 (pt) 1973-02-22
FR2070653A1 (es) 1971-09-17
AT291250B (de) 1971-07-12

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