FI962880A7 - Menetelmä ja välituotteita naftyridonikarboksyylihapposuolojen valmistusta varten - Google Patents

Menetelmä ja välituotteita naftyridonikarboksyylihapposuolojen valmistusta varten Download PDF

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Publication number
FI962880A7
FI962880A7 FI962880A FI962880A FI962880A7 FI 962880 A7 FI962880 A7 FI 962880A7 FI 962880 A FI962880 A FI 962880A FI 962880 A FI962880 A FI 962880A FI 962880 A7 FI962880 A7 FI 962880A7
Authority
FI
Finland
Prior art keywords
intermediates
preparation
acid salts
naphthyridonecarboxylic acid
naphthyridonecarboxylic
Prior art date
Application number
FI962880A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI962880A0 (fi
Inventor
Tamim F Braish
Darrell E Fox
Timothy Norris
Peter R Rose
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI962880A7 publication Critical patent/FI962880A7/fi
Publication of FI962880A0 publication Critical patent/FI962880A0/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
FI962880A 1994-01-18 1996-07-17 Menetelmä ja välituotteita naftyridonikarboksyylihapposuolojen valmistusta varten FI962880A0 (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US18194294A 1994-01-18 1994-01-18
PCT/IB1994/000410 WO1995019361A1 (fr) 1994-01-18 1994-12-12 Procede et intermediaires destines a la preparation de sels d'acide naphtyridonecarboxylique

Publications (2)

Publication Number Publication Date
FI962880A7 true FI962880A7 (fi) 1996-07-17
FI962880A0 FI962880A0 (fi) 1996-07-17

Family

ID=22666458

Family Applications (1)

Application Number Title Priority Date Filing Date
FI962880A FI962880A0 (fi) 1994-01-18 1996-07-17 Menetelmä ja välituotteita naftyridonikarboksyylihapposuolojen valmistusta varten

Country Status (19)

Country Link
EP (1) EP0740667A1 (fr)
JP (1) JP2891543B2 (fr)
KR (1) KR100221386B1 (fr)
CN (1) CN1141634A (fr)
AU (1) AU694149B2 (fr)
BR (1) BR9408490A (fr)
CA (1) CA2181351C (fr)
CZ (1) CZ286896B6 (fr)
FI (1) FI962880A0 (fr)
HU (1) HUT74883A (fr)
IL (1) IL112323A (fr)
MY (1) MY130510A (fr)
NO (1) NO305838B1 (fr)
NZ (1) NZ276478A (fr)
PL (1) PL179996B1 (fr)
RU (1) RU2147303C1 (fr)
TW (1) TW414791B (fr)
WO (1) WO1995019361A1 (fr)
ZA (1) ZA95340B (fr)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5763454A (en) * 1995-06-06 1998-06-09 Pfizer, Inc. Crystal form of anhydrous 7-( 1α,5α,6α!-6-amino-3-azabicyclo 3.1.0!hex-3-yl)-6-fluoro-1-(2,4-difluorophenyl)-1,4-dihydro-4-oxo-1,8 naphthyridine-3-carboxylic acid, methanessulfonic acid salt
ES2095809B1 (es) * 1995-07-27 1997-12-16 Sint Quimica Sa Procedimiento para la preparacion de acidos naftiridin carboxilicos y sus sales.
GB9524466D0 (en) * 1995-11-30 1996-01-31 Pfizer Ltd Process
JPH1087617A (ja) * 1996-07-09 1998-04-07 Pfizer Inc キノリン系抗生物質の合成に有用な中間体の製法
GB9614422D0 (en) * 1996-07-09 1996-09-04 Pfizer Ltd Novel process
HN1998000106A (es) 1997-08-01 1999-01-08 Pfizer Prod Inc Composiciones parenterales de alatroflaxacino
US6114531A (en) * 1998-07-28 2000-09-05 Pfizer Inc. Process for preparing quinolone and naphthyridone carboxylic acids
HN1999000141A (es) * 1998-09-03 2000-06-19 Pfizer Prod Inc Procedimiento para preparar sales de trovafloxacina de adicion de acidos.

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5164402A (en) * 1989-08-16 1992-11-17 Pfizer Inc Azabicyclo quinolone and naphthyridinone carboxylic acids
US5256791A (en) 1992-03-02 1993-10-26 Pfizer Inc. Preparation of intermediates in the synthesis of quinoline antibiotics

Also Published As

Publication number Publication date
NO305838B1 (no) 1999-08-02
EP0740667A1 (fr) 1996-11-06
CZ286896B6 (en) 2000-07-12
AU694149B2 (en) 1998-07-16
ZA95340B (en) 1996-07-17
AU1075495A (en) 1995-08-01
HU9601957D0 (en) 1996-09-30
BR9408490A (pt) 1997-08-26
IL112323A0 (en) 1995-03-30
RU2147303C1 (ru) 2000-04-10
MY130510A (en) 2007-06-29
IL112323A (en) 2001-03-19
TW414791B (en) 2000-12-11
HUT74883A (en) 1997-02-28
KR100221386B1 (ko) 1999-09-15
CN1141634A (zh) 1997-01-29
PL179996B1 (en) 2000-11-30
WO1995019361A1 (fr) 1995-07-20
JPH09501182A (ja) 1997-02-04
CA2181351A1 (fr) 1995-07-20
NO962990D0 (no) 1996-07-17
CZ211196A3 (en) 1997-01-15
NZ276478A (en) 1998-05-27
NO962990L (no) 1996-07-17
JP2891543B2 (ja) 1999-05-17
CA2181351C (fr) 1999-09-28
PL317043A1 (en) 1997-03-03
FI962880A0 (fi) 1996-07-17

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