IT1276171B1 - Derivati chinolinici - Google Patents

Derivati chinolinici

Info

Publication number
IT1276171B1
IT1276171B1 ITMI952462A IT1276171B1 IT 1276171 B1 IT1276171 B1 IT 1276171B1 IT MI952462 A ITMI952462 A IT MI952462A IT 1276171 B1 IT1276171 B1 IT 1276171B1
Authority
IT
Italy
Prior art keywords
neurokinin
treating
useful
carboxamide derivatives
receptor antagonists
Prior art date
Application number
Other languages
English (en)
Inventor
Giuseppe Arnaldo Mari Giardina
Mario Grugni
Luca Francesco Raveglia
Original Assignee
Smithkline Beecham Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Spa filed Critical Smithkline Beecham Spa
Publication of ITMI952462A0 publication Critical patent/ITMI952462A0/it
Priority to IT95MI002462 priority Critical patent/IT1276171B1/it
Priority to ARP960105282A priority patent/AR004735A1/es
Priority to HU9901016A priority patent/HUP9901016A3/hu
Priority to PL96326928A priority patent/PL326928A1/xx
Priority to TR1998/00883T priority patent/TR199800883T2/xx
Priority to IL12441896A priority patent/IL124418A0/xx
Priority to JP09520158A priority patent/JP2000513325A/ja
Priority to SK668-98A priority patent/SK66898A3/sk
Priority to CA002238328A priority patent/CA2238328A1/en
Priority to BR9611757A priority patent/BR9611757A/pt
Priority to ZA9609811A priority patent/ZA969811B/xx
Priority to PCT/EP1996/005207 priority patent/WO1997019926A1/en
Priority to EP96941025A priority patent/EP1019377A1/en
Priority to UY24375A priority patent/UY24375A1/es
Priority to CN96199747A priority patent/CN1207729A/zh
Priority to CZ981580A priority patent/CZ158098A3/cs
Priority to EA199800538A priority patent/EA001771B1/ru
Priority to KR1019980703874A priority patent/KR19990071598A/ko
Priority to APAP/P/1998/001238A priority patent/AP9801238A0/en
Priority to AU10318/97A priority patent/AU1031897A/en
Priority to MA24399A priority patent/MA24011A1/fr
Priority to DZ960173A priority patent/DZ2128A1/fr
Priority to TW085114501A priority patent/TW409123B/zh
Priority to UY24555A priority patent/UY24555A1/es
Publication of ITMI952462A1 publication Critical patent/ITMI952462A1/it
Application granted granted Critical
Publication of IT1276171B1 publication Critical patent/IT1276171B1/it
Priority to OA9800062A priority patent/OA11011A/en
Priority to NO19982333A priority patent/NO311213B1/no
Priority to MX9804108A priority patent/MX9804108A/es
Priority to BG102557A priority patent/BG102557A/bg
Priority to US09/994,402 priority patent/US20020068827A1/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IT95MI002462 1995-11-24 1995-11-24 Derivati chinolinici IT1276171B1 (it)

Priority Applications (29)

Application Number Priority Date Filing Date Title
IT95MI002462 IT1276171B1 (it) 1995-11-24 1995-11-24 Derivati chinolinici
ARP960105282A AR004735A1 (es) 1995-11-24 1996-11-21 Quinoleina 4-amido sustituida, un procedimiento para su preparacion, una composicion farmaceutica que los contiene y el uso de los mismos para lapreparacion de un medicamento.
CN96199747A CN1207729A (zh) 1995-11-24 1996-11-22 喹啉-4-酰胺衍生物,它们的制备以及它们作为神经激肽3(nk-3)和神经激肽2(nk-2)受体拮抗剂的应用
KR1019980703874A KR19990071598A (ko) 1995-11-24 1996-11-22 퀴놀린-4-카르복사미드 유도체, 그의 제조 방법 및 뉴로키닌3 (nk-3) 및 뉴로키닌 2 (nk-2) 수용체 길항제로서의 그 용도
TR1998/00883T TR199800883T2 (xx) 1995-11-24 1996-11-22 Kuinolin-4-Karboksamid t�revleri, haz�rlanmalar� ve n�rokinin 3 (NK-3)- ve n�rokinin 2 (NK-2) resept�r antagonistleri olarak kullan�mlar�.
IL12441896A IL124418A0 (en) 1995-11-24 1996-11-22 Quinoline-4-carboxamide derivatives their preparation and their use as neurokinin 3 (NK-3)- and neurokinin 2 (NK-2) receptor antagonists
JP09520158A JP2000513325A (ja) 1995-11-24 1996-11-22 キノリン―4―カルボキシアミド誘導体、その製法およびそのニューロキニン3(nk―3)およびニューロキニン2(nk―2)レセプター・アンタゴニストとしての使用
SK668-98A SK66898A3 (en) 1995-11-24 1996-11-22 Quinoline-4-carboxamide derivatives, their preparation and their use
CA002238328A CA2238328A1 (en) 1995-11-24 1996-11-22 Quinoline-4-carboxamide derivatives, their preparation and their use as neurokinin 3 (nk-3)- and neurokinin 2 (nk-2) receptor antagonists.
BR9611757A BR9611757A (pt) 1995-11-24 1996-11-22 Derivados quinolino-4-carboxamida sua preparação e seu uso como antagonitas de receptor neuroquinina 3 (nk-3)-e neuroquinina 2 (nk-2)
ZA9609811A ZA969811B (en) 1995-11-24 1996-11-22 Novel quinoline derivatives.
PCT/EP1996/005207 WO1997019926A1 (en) 1995-11-24 1996-11-22 Quinoline-4-carboxamide derivatives, their preparation and their use as neurokinin 3 (nk-3)- and neurokinin 2 (nk-2) receptor antagonists.
EP96941025A EP1019377A1 (en) 1995-11-24 1996-11-22 Quinoline-4-carboxamide derivatives, their preparation and their use as neurokinin 3 (nk-3)- and neurokinin 2 (nk-2) receptor antagonists.
UY24375A UY24375A1 (es) 1995-11-24 1996-11-22 Procedimiento para la preparacion de derivados de quinolin-4 -carboxamida
HU9901016A HUP9901016A3 (en) 1995-11-24 1996-11-22 Quinoline-4-carboxamide derivatives, their preparation and their use as neurokinin 3(nk-3)-and neurokinin 2(nk-2) receptor antagonists
CZ981580A CZ158098A3 (cs) 1995-11-24 1996-11-22 Chinolin-4-karboxamidové deriváty, způsob jejich přípravy, farmaceutický prostředek a použití jako antagonistů receptorů neurokininu 3(NK-3) a 2(NK-2)
EA199800538A EA001771B1 (ru) 1995-11-24 1996-11-22 Производные хинолин-4-карбоксамида, их получение и их применение в качестве антагонистов рецептора нейрокинина-3 (-к-3) и нейрокинина-2 (-к-2)
PL96326928A PL326928A1 (en) 1995-11-24 1996-11-22 Quinolin-4-carboxyamidic derivatives, their production and their application as antagonists ofneurokinin-3 (nk-3) and neurokinin-2 (nk-2)
APAP/P/1998/001238A AP9801238A0 (en) 1995-11-24 1996-11-22 Quinoline-4-carboxamide derivatives, their preparation and their use as neurokinin 3 (NK-3)- and neurokinin 2 (NK-2) receptor antagonists.
AU10318/97A AU1031897A (en) 1995-11-24 1996-11-22 Quinoline-4-carboxamide derivatives, their preparation and their use as neurokinin 3 (nk-3)- and neurokinin 2 (nk-2) receptor antagonists.
MA24399A MA24011A1 (fr) 1995-11-24 1996-11-22 Procede pour la preparation de nouveaux composes
DZ960173A DZ2128A1 (fr) 1995-11-24 1996-11-23 Composés nouveaux, procédé pour leur préparation et compositions pharmaceutiques les contenant.
TW085114501A TW409123B (en) 1995-11-24 1996-11-23 Quinoline derivatives and pharmaceutical composition containing the same
UY24555A UY24555A1 (es) 1995-11-24 1997-05-16 Nuevos compuestos
OA9800062A OA11011A (en) 1995-11-24 1998-05-22 Quinoline-4-carboxamide derivatives their preparation and their use as neurokin 3 (nk-3)-and neurokin 2 (nk-2)receptor antagonists
NO19982333A NO311213B1 (no) 1995-11-24 1998-05-22 Kinolinkarboksamid-derivater, deres fremstilling og deres anvendelse som Neurokinin 3 (NK-3)- og Neurokinin 2 (NK-2)reseptorantagonister, samt farmasöytiske preparater inneholdendedem
MX9804108A MX9804108A (es) 1995-11-24 1998-05-22 Derivados de quinolina-4-carboxamida, su preparacion y uso como antagonistas receptores de neuroquinina 3 (nk-3)- y neuroquinina 2 (kn-2).
BG102557A BG102557A (bg) 1995-11-24 1998-06-18 Производни на хинолин-4-карбоксамиди, метод за получаването им и използването им като антагонисти на неврокинин 3 / nк-/ и неврокинин 2 / nк-/ рецепторите
US09/994,402 US20020068827A1 (en) 1995-11-24 2001-11-26 Quinoline-4-carboxamide derivatives, their preparation and their use as neurokinin 3 ( NK-3 ) - and neurokinin 2 ( NK-3 ) receptor antagonists

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT95MI002462 IT1276171B1 (it) 1995-11-24 1995-11-24 Derivati chinolinici

Publications (3)

Publication Number Publication Date
ITMI952462A0 ITMI952462A0 (it) 1995-11-24
ITMI952462A1 ITMI952462A1 (it) 1997-05-24
IT1276171B1 true IT1276171B1 (it) 1997-10-27

Family

ID=11372597

Family Applications (1)

Application Number Title Priority Date Filing Date
IT95MI002462 IT1276171B1 (it) 1995-11-24 1995-11-24 Derivati chinolinici

Country Status (2)

Country Link
IT (1) IT1276171B1 (it)
ZA (1) ZA969811B (it)

Also Published As

Publication number Publication date
ITMI952462A0 (it) 1995-11-24
ZA969811B (en) 1998-05-22
ITMI952462A1 (it) 1997-05-24

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Legal Events

Date Code Title Description
0001 Granted