JP5818791B2 - ５−フルオロ−２−オキソピリミジン−１（２ｈ）−カルボキシレート誘導体 - Google Patents

５−フルオロ−２−オキソピリミジン−１（２ｈ）−カルボキシレート誘導体 Download PDF

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Publication number: JP5818791B2
Authority: JP; Japan
Prior art keywords: membered; optionally substituted; benzyl; phenyl; ring system
Prior art date: 2009-08-07
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Active

Application number

JP2012523954A

Other languages

English (en)

Japanese (ja)

Other versions

JP2013501726A5 (2

JP2013501726A (ja

Inventor

ボベル，ティモシー

ブライアン，クリスティー

ロールスバッハ，ベス

マーティン，ティモシー

オーウェン，ダブリュー．

ポバンズ，マーク

ソーンバーグ，スコット

ウェブスター，ジェフェリー

ヤオ，チェンリン

Original Assignee

ダウアグロサイエンシィズエルエルシー

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2009-08-07

Filing date

2010-08-05

Publication date

2015-11-18

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535293&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=JP5818791(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2010-08-05 Application filed by ダウアグロサイエンシィズエルエルシー, ダウアグロサイエンシィズエルエルシー filed Critical ダウアグロサイエンシィズエルエルシー

2013-01-17 Publication of JP2013501726A publication Critical patent/JP2013501726A/ja

2015-04-16 Publication of JP2013501726A5 publication Critical patent/JP2013501726A5/ja

2015-11-18 Application granted granted Critical

2015-11-18 Publication of JP5818791B2 publication Critical patent/JP5818791B2/ja

Status Active legal-status Critical Current

2030-08-05 Anticipated expiration legal-status Critical

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
- A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
- A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
- A01N47/16—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof the nitrogen atom being part of a heterocyclic ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/20—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D239/22—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to ring carbon atoms

Landscapes

Life Sciences & Earth Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Environmental Sciences (AREA)
Engineering & Computer Science (AREA)
Dentistry (AREA)
General Health & Medical Sciences (AREA)
Wood Science & Technology (AREA)
Zoology (AREA)
Plant Pathology (AREA)
Pest Control & Pesticides (AREA)
Agronomy & Crop Science (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Plural Heterocyclic Compounds (AREA)

JP2012523954A 2009-08-07 2010-08-05 ５−フルオロ−２−オキソピリミジン−１（２ｈ）−カルボキシレート誘導体 Active JP5818791B2 (ja)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US23223209P	2009-08-07	2009-08-07
US61/232,232		2009-08-07
PCT/US2010/044585 WO2011017544A1 (en)	2009-08-07	2010-08-05	5-fluoro-2-oxopyrimidine- 1(2h)-carboxylate derivatives

Publications (3)

Publication Number	Publication Date
JP2013501726A JP2013501726A (ja)	2013-01-17
JP2013501726A5 JP2013501726A5 (2)	2015-04-16
JP5818791B2 true JP5818791B2 (ja)	2015-11-18

Family

ID=43535293

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
JP2012523954A Active JP5818791B2 (ja)	2009-08-07	2010-08-05	５−フルオロ−２−オキソピリミジン−１（２ｈ）−カルボキシレート誘導体

Country Status (28)

Country	Link
US (1)	US8318758B2 (2)
EP (1)	EP2462133B1 (2)
JP (1)	JP5818791B2 (2)
KR (1)	KR101792286B1 (2)
CN (1)	CN102548979B (2)
AU (1)	AU2010279408B2 (2)
BR (1)	BR112012002807B1 (2)
CA (1)	CA2769251C (2)
CL (1)	CL2012000314A1 (2)
CO (1)	CO6491089A2 (2)
CR (1)	CR20120033A (2)
DK (1)	DK2462133T3 (2)
EA (1)	EA022930B1 (2)
EC (1)	ECSP12011651A (2)
ES (1)	ES2506169T3 (2)
HN (1)	HN2012000261A (2)
IL (1)	IL217954A (2)
IN (1)	IN2012DN00695A (2)
MX (1)	MX2012001623A (2)
NI (1)	NI201200019A (2)
NZ (1)	NZ597638A (2)
PE (1)	PE20120689A1 (2)
PL (1)	PL2462133T3 (2)
PT (1)	PT2462133E (2)
RS (1)	RS53658B1 (2)
UA (1)	UA106086C2 (2)
WO (1)	WO2011017544A1 (2)
ZA (1)	ZA201305992B (2)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DK2462134T3 (da) *	2009-08-07	2014-08-11	Dow Agrosciences Llc	N1-sulfonyl-5-fluorpyrimidinonderivater
JP6324994B2 (ja) *	2012-12-28	2018-05-16	アダマ・マクテシム・リミテッド	Ｎ−（置換）−５−フルオロ−４−イミノ−３−メチル−２−オキソ−３，４−ジヒドロピリミジン−１（２ｈ）−カルボキシレート誘導体
KR20150100869A (ko)	2012-12-28	2015-09-02	다우 아그로사이언시즈 엘엘씨	N-(치환된)-5-플루오로-4-이미노-3-메틸-2-옥소-3,4-디히드로피리미딘-1(2h)-카르복스아미드 유도체
RU2018118951A (ru)	2012-12-28	2018-11-02	Адама Мактешим Лтд.	Производные 1-(замещенный бензоил)-5-фтор-4-имино-3-метил-3,4-дигидропиримидин-2(1h)-она
CN105007737A (zh)	2012-12-31	2015-10-28	美国陶氏益农公司	作为杀真菌剂的3-烷基-5-氟-4-取代的-亚氨基-3,4-二氢嘧啶-2(1h)-酮衍生物
CN114794123B (zh)	2013-12-31	2024-11-12	阿达玛马克西姆股份有限公司	用防治谷类中真菌的协同杀真菌混合物
JP6585057B2 (ja)	2013-12-31	2019-10-02	アダマ・マクテシム・リミテッド	５−フルオロ−４−イミノ−３−（アルキル／置換アルキル）−１−（アリールスルホニル）−３，４−ジヒドロピリミジン−２（１ｈ）−オンおよびそれらの調製方法
WO2016040193A1 (en)	2014-09-08	2016-03-17	Samumed, Llc	3-(1h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[3,4-b]pyridine and therapeutic uses thereof
MX380092B (es)	2015-11-06	2025-03-11	Samumed Llc	Tratamiento de la osteoartritis.
MX390577B (es)	2016-06-01	2025-03-20	Samumed Llc	Proceso de preparación de n-(5-(3-(7-(3-fluorofenil)-3h-imidazo[4,5-c]piridin-2-il)-1h-indazol-5-il)piridin-3-il)-3-metilbutanamida.
MA49639A (fr)	2017-07-17	2020-05-27	Adama Makhteshim Ltd	Polymorphes de 5-fluoro-4-imino-3-méthyl-1-tosyl-3,4-dihydropyrimidin-2-one
PE20212103A1 (es)	2018-11-05	2021-11-04	Adama Makhteshim Ltd	Mezclas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2-ona, y metodos de uso de los mismos
PY2057637A (es)	2019-09-23	2021-10-05	Adama Makhteshim Ltd	Proceso para preparar 5-(fluoro-4-imino-3-metil)-1-tosil-3,4-dihidropirimidin-(1h)-ona y derivados del compuesto

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3368938A (en) *	1966-01-13	1968-02-13	Hoffmann La Roche	Controlling fungi with 5-fluorocytosine
PT888359E (pt)	1996-03-11	2002-10-31	Syngenta Participations Ag	Derivados de pirimidin-4-ona como pesticida
WO2004037159A2 (en) *	2002-10-23	2004-05-06	Obetherapy Biotechnology	Compounds, compositions and methods for modulating fat metabolism
US8592435B2 (en) *	2007-04-27	2013-11-26	Daiichi Sankyo Company, Limited	Nitrogen-containing six-membered aromatic ring derivatives and pharmaceutical products containing the same
KR20110042204A (ko) *	2008-08-01	2011-04-25	다우 아그로사이언시즈 엘엘씨	살진균제로서의 5-플루오로시토신의 용도

2010
- 2010-08-05 BR BR112012002807-3A patent/BR112012002807B1/pt active IP Right Grant
- 2010-08-05 PT PT108071747T patent/PT2462133E/pt unknown
- 2010-08-05 MX MX2012001623A patent/MX2012001623A/es active IP Right Grant
- 2010-08-05 US US12/851,304 patent/US8318758B2/en active Active
- 2010-08-05 EP EP10807174.7A patent/EP2462133B1/en active Active
- 2010-08-05 AU AU2010279408A patent/AU2010279408B2/en not_active Ceased
- 2010-08-05 EA EA201270255A patent/EA022930B1/ru not_active IP Right Cessation
- 2010-08-05 PL PL10807174T patent/PL2462133T3/pl unknown
- 2010-08-05 ES ES10807174.7T patent/ES2506169T3/es active Active
- 2010-08-05 RS RS20140630A patent/RS53658B1/sr unknown
- 2010-08-05 JP JP2012523954A patent/JP5818791B2/ja active Active
- 2010-08-05 PE PE2012000170A patent/PE20120689A1/es not_active Application Discontinuation
- 2010-08-05 KR KR1020127005932A patent/KR101792286B1/ko not_active Expired - Fee Related
- 2010-08-05 DK DK10807174.7T patent/DK2462133T3/en active
- 2010-08-05 UA UAA201202680A patent/UA106086C2/uk unknown
- 2010-08-05 IN IN695DEN2012 patent/IN2012DN00695A/en unknown
- 2010-08-05 CN CN201080045339.3A patent/CN102548979B/zh active Active
- 2010-08-05 NZ NZ597638A patent/NZ597638A/en unknown
- 2010-08-05 WO PCT/US2010/044585 patent/WO2011017544A1/en not_active Ceased
- 2010-08-05 CA CA2769251A patent/CA2769251C/en not_active Expired - Fee Related
2012
- 2012-01-18 CR CR20120033A patent/CR20120033A/es unknown
- 2012-01-27 CO CO12012413A patent/CO6491089A2/es active IP Right Grant
- 2012-02-02 HN HN2012000261A patent/HN2012000261A/es unknown
- 2012-02-03 NI NI201200019A patent/NI201200019A/es unknown
- 2012-02-05 IL IL217954A patent/IL217954A/en active IP Right Grant
- 2012-02-06 CL CL2012000314A patent/CL2012000314A1/es unknown
- 2012-02-07 EC ECSP12011651 patent/ECSP12011651A/es unknown
2013
- 2013-08-14 ZA ZA2013/05992A patent/ZA201305992B/en unknown

Also Published As

Publication number	Publication date
NI201200019A (es)	2012-05-22
CO6491089A2 (es)	2012-07-31
BR112012002807A2 (pt)	2015-10-13
KR101792286B1 (ko)	2017-10-31
US20110034491A1 (en)	2011-02-10
RS53658B1 (sr)	2015-04-30
CR20120033A (es)	2012-03-22
CA2769251A1 (en)	2011-02-10
US8318758B2 (en)	2012-11-27
PL2462133T3 (pl)	2015-03-31
NZ597638A (en)	2014-06-27
AU2010279408B2 (en)	2015-09-10
HK1172892A1 (en)	2013-05-03
ES2506169T3 (es)	2014-10-13
CL2012000314A1 (es)	2012-10-05
HN2012000261A (es)	2015-01-05
BR112012002807A8 (pt)	2017-07-11
UA106086C2 (uk)	2014-07-25
CN102548979A (zh)	2012-07-04
PT2462133E (pt)	2014-12-26
CN102548979B (zh)	2015-05-13
WO2011017544A1 (en)	2011-02-10
EA201270255A1 (ru)	2012-07-30
ECSP12011651A (es)	2012-03-30
CA2769251C (en)	2018-05-15
IL217954A0 (en)	2012-03-29
EP2462133A4 (en)	2013-01-16
ZA201305992B (en)	2014-10-29
IN2012DN00695A (2)	2015-06-19
BR112012002807B1 (pt)	2018-07-10
DK2462133T3 (en)	2015-01-05
KR20120043069A (ko)	2012-05-03
EA022930B1 (ru)	2016-03-31
EP2462133A1 (en)	2012-06-13
IL217954A (en)	2016-02-29
JP2013501726A (ja)	2013-01-17
AU2010279408A1 (en)	2012-02-09
MX2012001623A (es)	2012-04-11
EP2462133B1 (en)	2014-09-24
PE20120689A1 (es)	2012-06-06

Legal Events

Date	Code	Title	Description
2013-08-01	A621	Written request for application examination	Free format text: JAPANESE INTERMEDIATE CODE: A621 Effective date: 20130731
2014-08-29	A977	Report on retrieval	Free format text: JAPANESE INTERMEDIATE CODE: A971007 Effective date: 20140828
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2014-12-27	A601	Written request for extension of time	Free format text: JAPANESE INTERMEDIATE CODE: A601 Effective date: 20141226
2015-02-27	A524	Written submission of copy of amendment under article 19 pct	Free format text: JAPANESE INTERMEDIATE CODE: A524 Effective date: 20150227
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2015-09-02	A01	Written decision to grant a patent or to grant a registration (utility model)	Free format text: JAPANESE INTERMEDIATE CODE: A01 Effective date: 20150901
2015-10-08	A61	First payment of annual fees (during grant procedure)	Free format text: JAPANESE INTERMEDIATE CODE: A61 Effective date: 20150929
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Publication	Publication Date	Title
JP5818791B2 (ja)	2015-11-18	５−フルオロ−２−オキソピリミジン−１（２ｈ）−カルボキシレート誘導体
KR102732893B1 (ko)	2024-11-22	살진균제로서의 피콜린아미드
JP5784603B2 (ja)	2015-09-24	Ｎ１−スルホニル−５−フルオロピリミジノン誘導体
JP5759991B2 (ja)	2015-08-05	５−フルオロピリミジノン誘導体
JP6128658B2 (ja)	2017-05-17	５−フルオロ−４−イミノ−３−（置換）−３，４−ジヒドロピリミジン−２−（１ｈ）−オン誘導体
ES2549046T3 (es)	2015-10-22	Derivados de N-ciano-4-amino-5-fluoro-pirimidina como fungicidas
JP5735510B2 (ja)	2015-06-17	Ｎ１−置換−５−フルオロ−２−オキソピリミジノン−１（２ｈ）−カルボキサミド誘導体
JP5748754B2 (ja)	2015-07-15	Ｎ１−アシル−５−フルオロピリミジノン誘導体
BR112012004024B1 (pt)	2018-07-10	Método para distribuir material sinterizado a partir de uma correia de sínter e calha de distribuição para distribuir material sinterizado
KR20120094140A (ko)	2012-08-23	2-알독시미노-5-플루오로피리미딘 유도체
JP2014527530A (ja)	2014-10-16	Ｎ−（５−フルオロ−２（（４−メチルベンジル）オキシ）ピリミジン−４−イル）ベンズアミド誘導体
HK1176005A (en)	2013-07-19	2-aldoximino-5-fluoropyrimidine derivatives
HK1172892B (en)	2016-04-08	5-fluoro-2-oxopyrimidine- 1(2h)-carboxylate derivatives
HK1172894B (en)	2016-04-08	N1-acyl-5-fluoropyrimidinone derivatives
HK1173142B (en)	2015-10-23	N1-sulfonyl-5-fluoropyrimidinone derivatives