MX346193B - Composiciones farmaceuticas. - Google Patents

Composiciones farmaceuticas.

Info

Publication number
MX346193B
MX346193B MX2013003037A MX2013003037A MX346193B MX 346193 B MX346193 B MX 346193B MX 2013003037 A MX2013003037 A MX 2013003037A MX 2013003037 A MX2013003037 A MX 2013003037A MX 346193 B MX346193 B MX 346193B
Authority
MX
Mexico
Prior art keywords
pharmaceutical compositions
methyl
oxazolo
pyrazin
pyrido
Prior art date
Application number
MX2013003037A
Other languages
English (en)
Other versions
MX2013003037A (es
Inventor
B Mundhra Deepak
Pan Rennan
Original Assignee
Viiv Healthcare Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Viiv Healthcare Co filed Critical Viiv Healthcare Co
Publication of MX2013003037A publication Critical patent/MX2013003037A/es
Publication of MX346193B publication Critical patent/MX346193B/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invención se refiere a composiciones farmacéuticas de (3S, 11aR)-N-[(2, 4-difluorofenil)metil]-2, 3, 5, 7,11,11a-hexahidro-6-hidroxi-3-metil-5, 7-dioxo-oxazolo[3, 2-a]pirido[1 ,2-d]pirazin-8-carboxamida, útiles en el tratamiento o prevención de infección por Virus de Inmunodeficiencia Humana (VIH).
MX2013003037A 2010-09-16 2011-09-15 Composiciones farmaceuticas. MX346193B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US38354110P 2010-09-16 2010-09-16
PCT/US2011/051713 WO2012037320A2 (en) 2010-09-16 2011-09-15 Pharmaceutical compositions

Publications (2)

Publication Number Publication Date
MX2013003037A MX2013003037A (es) 2013-09-02
MX346193B true MX346193B (es) 2017-03-10

Family

ID=45832235

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2013003037A MX346193B (es) 2010-09-16 2011-09-15 Composiciones farmaceuticas.

Country Status (28)

Country Link
US (7) US20130171214A1 (es)
EP (1) EP2616076B1 (es)
JP (1) JP6231385B2 (es)
KR (1) KR101938662B1 (es)
CN (1) CN103547266B (es)
AU (1) AU2011302030B2 (es)
BR (1) BR112013005907B1 (es)
CA (1) CA2810524C (es)
CL (1) CL2013000715A1 (es)
CY (1) CY1118279T1 (es)
DK (1) DK2616076T3 (es)
EA (1) EA024924B1 (es)
ES (1) ES2594557T3 (es)
HR (1) HRP20161280T1 (es)
HU (1) HUE031336T2 (es)
IL (1) IL225028A (es)
LT (1) LT2616076T (es)
ME (1) ME02520B (es)
MX (1) MX346193B (es)
PL (1) PL2616076T3 (es)
PT (1) PT2616076T (es)
RS (1) RS55222B1 (es)
SI (1) SI2616076T1 (es)
SM (1) SMT201600350B (es)
TW (1) TWI577377B (es)
UA (1) UA108250C2 (es)
WO (1) WO2012037320A2 (es)
ZA (1) ZA201301766B (es)

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WO2020112931A1 (en) 2018-11-29 2020-06-04 Board Of Regents Of The University Of Nebraska Antiviral prodrugs and nanoformulations thereof
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FI4196479T3 (fi) 2021-01-19 2024-01-17 Gilead Sciences Inc Substituoituja pyridotriatsiiniyhdisteitä ja niiden käyttöjä
TWI856796B (zh) 2022-04-06 2024-09-21 美商基利科學股份有限公司 橋聯三環胺甲醯基吡啶酮化合物及其用途
CN115844838B (zh) * 2022-12-01 2023-10-24 浙江萃泽医药科技有限公司 一种可注射的药物组合物
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Also Published As

Publication number Publication date
CN103547266A (zh) 2014-01-29
SI2616076T1 (sl) 2016-11-30
US20170027933A1 (en) 2017-02-02
US20250268893A1 (en) 2025-08-28
ZA201301766B (en) 2016-11-30
PL2616076T3 (pl) 2017-07-31
ME02520B (me) 2017-02-20
EP2616076B1 (en) 2016-07-13
CA2810524C (en) 2018-06-26
ES2594557T3 (es) 2016-12-21
MX2013003037A (es) 2013-09-02
CA2810524A1 (en) 2012-03-22
CY1118279T1 (el) 2017-06-28
EP2616076A2 (en) 2013-07-24
US20130171214A1 (en) 2013-07-04
EA201390233A1 (ru) 2014-03-31
HUE031336T2 (hu) 2017-07-28
BR112013005907B1 (pt) 2021-04-27
TWI577377B (zh) 2017-04-11
US11224597B2 (en) 2022-01-18
HRP20161280T1 (hr) 2016-11-18
EA024924B1 (ru) 2016-11-30
AU2011302030B2 (en) 2015-01-22
JP6231385B2 (ja) 2017-11-15
US20220096469A1 (en) 2022-03-31
US20240307387A1 (en) 2024-09-19
IL225028A (en) 2017-04-30
KR101938662B1 (ko) 2019-01-15
KR20130116254A (ko) 2013-10-23
AU2011302030A1 (en) 2013-04-04
CL2013000715A1 (es) 2013-07-05
DK2616076T3 (en) 2016-10-24
JP2014500849A (ja) 2014-01-16
RS55222B1 (sr) 2017-02-28
SMT201600350B (it) 2016-11-10
TW201223529A (en) 2012-06-16
WO2012037320A2 (en) 2012-03-22
US20250017923A1 (en) 2025-01-16
UA108250C2 (uk) 2015-04-10
EP2616076A4 (en) 2015-01-21
CN103547266B (zh) 2016-04-06
US12138264B2 (en) 2024-11-12
LT2616076T (lt) 2016-10-10
BR112013005907A2 (pt) 2016-06-07
US20250017924A1 (en) 2025-01-16
PT2616076T (pt) 2016-09-30
WO2012037320A3 (en) 2014-03-27

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