NL8302353A - Fosforyleringsmiddel; werkwijze voor het bereiden daarvan; werkwijze voor het fosforyleren van een organische hydroxyl- of amineverbinding. - Google Patents

Fosforyleringsmiddel; werkwijze voor het bereiden daarvan; werkwijze voor het fosforyleren van een organische hydroxyl- of amineverbinding. Download PDF

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Publication number
NL8302353A
NL8302353A NL8302353A NL8302353A NL8302353A NL 8302353 A NL8302353 A NL 8302353A NL 8302353 A NL8302353 A NL 8302353A NL 8302353 A NL8302353 A NL 8302353A NL 8302353 A NL8302353 A NL 8302353A
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NL
Netherlands
Prior art keywords
mse
group
phosphorylating agent
formula
phosphorylating
Prior art date
Application number
NL8302353A
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English (en)
Dutch (nl)
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Stichting Katholieke Univ
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Stichting Katholieke Univ filed Critical Stichting Katholieke Univ
Priority to NL8302353A priority Critical patent/NL8302353A/nl
Priority to CA000456949A priority patent/CA1224165A/en
Priority to US06/622,571 priority patent/US4692542A/en
Priority to AU29787/84A priority patent/AU572158B2/en
Priority to DK312784A priority patent/DK312784A/da
Priority to NO842662A priority patent/NO842662L/no
Priority to JP59135055A priority patent/JPS6069087A/ja
Priority to AT84200951T priority patent/ATE34577T1/de
Priority to DE8484200951T priority patent/DE3471484D1/de
Priority to EP84200951A priority patent/EP0131993B1/de
Publication of NL8302353A publication Critical patent/NL8302353A/nl

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H11/00Compounds containing saccharide radicals esterified by inorganic acids; Metal salts thereof
    • C07H11/04Phosphates; Phosphites; Polyphosphates
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/06Phosphorus compounds without P—C bonds
    • C07F9/08Esters of oxyacids of phosphorus
    • C07F9/09Esters of phosphoric acids
    • C07F9/091Esters of phosphoric acids with hydroxyalkyl compounds with further substituents on alkyl
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/06Phosphorus compounds without P—C bonds
    • C07F9/08Esters of oxyacids of phosphorus
    • C07F9/09Esters of phosphoric acids
    • C07F9/094Esters of phosphoric acids with arylalkanols
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/06Phosphorus compounds without P—C bonds
    • C07F9/08Esters of oxyacids of phosphorus
    • C07F9/09Esters of phosphoric acids
    • C07F9/12Esters of phosphoric acids with hydroxyaryl compounds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/06Phosphorus compounds without P—C bonds
    • C07F9/08Esters of oxyacids of phosphorus
    • C07F9/09Esters of phosphoric acids
    • C07F9/14Esters of phosphoric acids containing P(=O)-halide groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/06Phosphorus compounds without P—C bonds
    • C07F9/08Esters of oxyacids of phosphorus
    • C07F9/141Esters of phosphorous acids
    • C07F9/146Esters of phosphorous acids containing P-halide groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6527Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07F9/6533Six-membered rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6564Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms
    • C07F9/6571Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms having phosphorus and oxygen atoms as the only ring hetero atoms
    • C07F9/6574Esters of oxyacids of phosphorus
    • C07F9/65744Esters of oxyacids of phosphorus condensed with carbocyclic or heterocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16Purine radicals
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Saccharide Compounds (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
NL8302353A 1983-07-01 1983-07-01 Fosforyleringsmiddel; werkwijze voor het bereiden daarvan; werkwijze voor het fosforyleren van een organische hydroxyl- of amineverbinding. NL8302353A (nl)

Priority Applications (10)

Application Number Priority Date Filing Date Title
NL8302353A NL8302353A (nl) 1983-07-01 1983-07-01 Fosforyleringsmiddel; werkwijze voor het bereiden daarvan; werkwijze voor het fosforyleren van een organische hydroxyl- of amineverbinding.
CA000456949A CA1224165A (en) 1983-07-01 1984-06-19 Phosphorylating agent; a process for the preparation thereof; a process for phosphorylating an organic hydroxyl or amine compound
US06/622,571 US4692542A (en) 1983-07-01 1984-06-20 Phosphorylating agent
AU29787/84A AU572158B2 (en) 1983-07-01 1984-06-22 Phosphorylating agents and process for phosphorylating an organic hydroxyl or amine compound
DK312784A DK312784A (da) 1983-07-01 1984-06-27 Phosphorylerende middel, fremgangsmaade til fremstilling af et saadant samt en fremgangsmaade til phosphorylering af en organisk hydroxyl- eller amin-forbindelse
NO842662A NO842662L (no) 1983-07-01 1984-06-29 Fosforyleringsreagens, fremgangsmaate ved fremstilling og anvendelse derav
JP59135055A JPS6069087A (ja) 1983-07-01 1984-06-29 リン酸化剤
AT84200951T ATE34577T1 (de) 1983-07-01 1984-06-29 Phosphorylierungsmittel, verfahren zu seiner herstellung, verfahren zur phosphorylierung einer organischen hydroxyl- oder amin-verbindung.
DE8484200951T DE3471484D1 (en) 1983-07-01 1984-06-29 Phosphorylating agent; a process for the preparation thereof; a process for phosphorylating an organic hydroxyl or amine compound
EP84200951A EP0131993B1 (de) 1983-07-01 1984-06-29 Phosphorylierungsmittel, Verfahren zu seiner Herstellung, Verfahren zur Phosphorylierung einer organischen Hydroxyl- oder Amin-Verbindung

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
NL8302353A NL8302353A (nl) 1983-07-01 1983-07-01 Fosforyleringsmiddel; werkwijze voor het bereiden daarvan; werkwijze voor het fosforyleren van een organische hydroxyl- of amineverbinding.
NL8302353 1983-07-01

Publications (1)

Publication Number Publication Date
NL8302353A true NL8302353A (nl) 1985-02-01

Family

ID=19842103

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8302353A NL8302353A (nl) 1983-07-01 1983-07-01 Fosforyleringsmiddel; werkwijze voor het bereiden daarvan; werkwijze voor het fosforyleren van een organische hydroxyl- of amineverbinding.

Country Status (10)

Country Link
US (1) US4692542A (de)
EP (1) EP0131993B1 (de)
JP (1) JPS6069087A (de)
AT (1) ATE34577T1 (de)
AU (1) AU572158B2 (de)
CA (1) CA1224165A (de)
DE (1) DE3471484D1 (de)
DK (1) DK312784A (de)
NL (1) NL8302353A (de)
NO (1) NO842662L (de)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL8302353A (nl) * 1983-07-01 1985-02-01 Stichting Katholieke Univ Fosforyleringsmiddel; werkwijze voor het bereiden daarvan; werkwijze voor het fosforyleren van een organische hydroxyl- of amineverbinding.
USRE34069E (en) * 1983-08-18 1992-09-15 Biosyntech Gmbh Process for the preparation of oligonucleotides
DE3329892A1 (de) * 1983-08-18 1985-03-07 Köster, Hubert, Prof. Dr., 2000 Hamburg Verfahren zur herstellung von oligonucleotiden
DE3507881A1 (de) 1985-03-06 1986-09-11 Hoechst Ag, 6230 Frankfurt Verfahren und mittel zur phosphorylierung
US5332845A (en) * 1985-03-28 1994-07-26 Chiron Corporation Phosphorylating reagents
US5252760A (en) * 1985-03-28 1993-10-12 Chiron Corporation Method of using colored phosphorylating reagents
JPH0291088A (ja) * 1988-09-29 1990-03-30 Central Glass Co Ltd ホスファイトおよびヌクレオシド‐3’‐ホスファイト誘導体およびこれを用いるオリゴヌクレオチドの合成法
ES2019839A6 (es) * 1990-05-10 1991-07-01 Europharma Sa Procedimiento de obtencion de derivados polifosforilados de galactosa con actividad insulinica.
JPWO2015037587A1 (ja) * 2013-09-11 2017-03-02 株式会社PRISM Pharma ピラジノ[2,1−c][1,2,4]トリアジン化合物の製造方法
CN110627830A (zh) * 2019-10-15 2019-12-31 安徽昊帆生物有限公司 对硝基苯磷酸二钠及其制备方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL8302353A (nl) * 1983-07-01 1985-02-01 Stichting Katholieke Univ Fosforyleringsmiddel; werkwijze voor het bereiden daarvan; werkwijze voor het fosforyleren van een organische hydroxyl- of amineverbinding.

Also Published As

Publication number Publication date
DK312784A (da) 1985-01-02
EP0131993A3 (en) 1985-05-15
CA1224165A (en) 1987-07-14
DE3471484D1 (en) 1988-06-30
US4692542A (en) 1987-09-08
JPS6069087A (ja) 1985-04-19
DK312784D0 (da) 1984-06-27
EP0131993B1 (de) 1988-05-25
NO842662L (no) 1985-01-02
AU572158B2 (en) 1988-05-05
EP0131993A2 (de) 1985-01-23
AU2978784A (en) 1985-01-03
ATE34577T1 (de) 1988-06-15

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