SU1103795A3 - Способ получени производных диазепинона - Google Patents

Способ получени производных диазепинона Download PDF

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Publication number
SU1103795A3
SU1103795A3 SU823441915A SU3441915A SU1103795A3 SU 1103795 A3 SU1103795 A3 SU 1103795A3 SU 823441915 A SU823441915 A SU 823441915A SU 3441915 A SU3441915 A SU 3441915A SU 1103795 A3 SU1103795 A3 SU 1103795A3
Authority
SU
USSR - Soviet Union
Prior art keywords
hydrogen
general formula
diazepinone
pyrido
derivatives
Prior art date
Application number
SU823441915A
Other languages
English (en)
Russian (ru)
Inventor
Шмидт Гюнтер
Энгель Вольфхард
Эберлейн Вольфганг
Труммлитц Гюнтер
Энгельхардт Гюнтер
Original Assignee
Др. Карл Томэ Гмбх (Фирма)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Др. Карл Томэ Гмбх (Фирма) filed Critical Др. Карл Томэ Гмбх (Фирма)
Application granted granted Critical
Publication of SU1103795A3 publication Critical patent/SU1103795A3/ru

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/16—Halogen atoms or nitro radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Rheumatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
SU823441915A 1981-06-06 1982-05-25 Способ получени производных диазепинона SU1103795A3 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19813122670 DE3122670A1 (de) 1981-06-06 1981-06-06 "neue 1,4,9,10-tetrahydro-pyrazolo(4,3-e) pyrido(3,2-b)(1,4)diazepin-10-one, verfahren zu ihrer herstellung und ihre verwendung zur herstellung von pharmazeutischen wirkstoffen"

Publications (1)

Publication Number Publication Date
SU1103795A3 true SU1103795A3 (ru) 1984-07-15

Family

ID=6134176

Family Applications (1)

Application Number Title Priority Date Filing Date
SU823441915A SU1103795A3 (ru) 1981-06-06 1982-05-25 Способ получени производных диазепинона

Country Status (27)

Country Link
US (1) US4381303A (2)
EP (1) EP0066774B1 (2)
JP (1) JPS57212182A (2)
KR (1) KR880001719B1 (2)
AR (1) AR229124A1 (2)
AT (1) ATE10744T1 (2)
AU (1) AU552765B2 (2)
CA (1) CA1167440A (2)
CS (1) CS226743B2 (2)
DD (1) DD202574A5 (2)
DE (2) DE3122670A1 (2)
DK (1) DK253382A (2)
ES (1) ES8304571A1 (2)
FI (1) FI71560C (2)
GB (1) GB2117755B (2)
GR (1) GR76438B (2)
HU (1) HU186067B (2)
IE (1) IE53067B1 (2)
IL (1) IL65977A (2)
NO (1) NO158063C (2)
NZ (1) NZ200859A (2)
PH (1) PH17719A (2)
PL (1) PL135845B1 (2)
PT (1) PT75016B (2)
SU (1) SU1103795A3 (2)
YU (1) YU118282A (2)
ZA (1) ZA823919B (2)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2124014C1 (ru) * 1993-12-29 1998-12-27 Пфайзер Инк. Диазабициклические соединения и содержащая их фармацевтическая композиция
RU2142464C1 (ru) * 1994-02-18 1999-12-10 Берингер Ингельгейм Фармасьютикалз, Инк. 2-гетероарил-5,11-дигидро-6н-дипиридо[3,2-b:2',3'-e][1,4] диазепин-6-оны, их фармацевтически приемлемые соли, фармацевтическая композиция, обладающая ингибирующей активностью в отношении обратной транскриптазы вич-1

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3643666A1 (de) * 1986-12-20 1988-06-30 Thomae Gmbh Dr K Neue kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
US4749788A (en) * 1987-04-13 1988-06-07 A. H. Robins Company, Incorporated Process for the preparation of aryl-pyrido(1,4) benzodiazepines
US5366972A (en) * 1989-04-20 1994-11-22 Boehringer Ingelheim Pharmaceuticals, Inc. 5,11-dihydro-6H-dipyrido(3,2-B:2',3'-E)(1,4)diazepines and their use in the prevention or treatment of HIV infection
EP0410148B1 (en) * 1989-06-28 1994-04-06 Boehringer Ingelheim Pharmaceuticals Inc. Novel 5,11-dihydro-6H-dipyrido[3,2-b:2',3'-e][1,4]diazepin-6-ones and thiones and their use in the prevention or treatment of AIDS
CA2052946A1 (en) * 1990-10-19 1992-04-20 Karl G. Grozinger Method for the preparation of 5,11-dihydro-6h-dipyrido ¬3,2-b:2', 3'-e| ¬1,4|diazepines
ES2137113B1 (es) 1997-07-29 2000-09-16 Almirall Prodesfarma Sa Nuevos derivados de triazolo-piridazinas heterociclicos.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3450694A (en) * 1966-02-23 1969-06-17 Abbott Lab Substituted benzoxazepines and benzothiazepines
DE2707269A1 (de) * 1977-02-19 1978-08-24 Hoechst Ag Heterocyclische stickstoffverbindungen und verfahren zu ihrer herstellung
EP0023707B1 (de) * 1979-08-03 1986-04-30 Byk Gulden Lomberg Chemische Fabrik GmbH Substituierte Tetraazatricyclen, Verfahren zu ihrer Herstellung, ihre Verwendung und sie enthaltende Arzneimittel

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
Патент US № 3539554, кл. 260-239.3, опублик. 1970. 2. Патент DE № 1620572, кл. 12р 10/10, опублик. 1972. *

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2124014C1 (ru) * 1993-12-29 1998-12-27 Пфайзер Инк. Диазабициклические соединения и содержащая их фармацевтическая композиция
RU2142464C1 (ru) * 1994-02-18 1999-12-10 Берингер Ингельгейм Фармасьютикалз, Инк. 2-гетероарил-5,11-дигидро-6н-дипиридо[3,2-b:2',3'-e][1,4] диазепин-6-оны, их фармацевтически приемлемые соли, фармацевтическая композиция, обладающая ингибирующей активностью в отношении обратной транскриптазы вич-1

Also Published As

Publication number Publication date
YU118282A (en) 1986-04-30
FI821992A0 (fi) 1982-06-04
IE53067B1 (en) 1988-05-25
AR229124A1 (es) 1983-06-15
NZ200859A (en) 1985-08-16
KR840000543A (ko) 1984-02-25
GR76438B (2) 1984-08-10
ZA823919B (en) 1984-02-29
ATE10744T1 (de) 1984-12-15
NO158063B (no) 1988-03-28
PL236742A1 (en) 1984-03-26
ES512846A0 (es) 1983-03-01
ES8304571A1 (es) 1983-03-01
PH17719A (en) 1984-11-21
NO821882L (no) 1982-12-07
EP0066774A1 (de) 1982-12-15
NO158063C (no) 1988-07-06
CS226743B2 (en) 1984-04-16
GB2117755A (en) 1983-10-19
FI71560C (fi) 1987-01-19
FI71560B (fi) 1986-10-10
IE821350L (en) 1982-12-06
KR880001719B1 (ko) 1988-09-08
DD202574A5 (de) 1983-09-21
PT75016A (de) 1982-07-01
AU552765B2 (en) 1986-06-19
AU8460582A (en) 1982-12-16
GB2117755B (en) 1985-01-30
DE3122670A1 (de) 1982-12-23
DE3261530D1 (en) 1985-01-24
IL65977A0 (en) 1982-09-30
IL65977A (en) 1984-12-31
HU186067B (en) 1985-05-28
JPS57212182A (en) 1982-12-27
PL135845B1 (en) 1985-12-31
US4381303A (en) 1983-04-26
DK253382A (da) 1982-12-07
EP0066774B1 (de) 1984-12-12
CA1167440A (en) 1984-05-15
PT75016B (de) 1985-05-17

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