AR036317A1 - Nuevo cristal de compuesto lipopeptido ciclico - Google Patents
Nuevo cristal de compuesto lipopeptido ciclicoInfo
- Publication number
- AR036317A1 AR036317A1 ARP020103266A ARP020103266A AR036317A1 AR 036317 A1 AR036317 A1 AR 036317A1 AR P020103266 A ARP020103266 A AR P020103266A AR P020103266 A ARP020103266 A AR P020103266A AR 036317 A1 AR036317 A1 AR 036317A1
- Authority
- AR
- Argentina
- Prior art keywords
- lipopeptide
- composite crystal
- crystal
- new
- new cycling
- Prior art date
Links
- 108010028921 Lipopeptides Proteins 0.000 title abstract 3
- 239000013078 crystal Substances 0.000 title abstract 3
- 239000002131 composite material Substances 0.000 title 1
- 230000001351 cycling effect Effects 0.000 title 1
- CSCPPACGZOOCGX-UHFFFAOYSA-N Acetone Chemical compound CC(C)=O CSCPPACGZOOCGX-UHFFFAOYSA-N 0.000 abstract 3
- WEVYAHXRMPXWCK-UHFFFAOYSA-N Acetonitrile Chemical compound CC#N WEVYAHXRMPXWCK-UHFFFAOYSA-N 0.000 abstract 3
- YMWUJEATGCHHMB-UHFFFAOYSA-N Dichloromethane Chemical compound ClCCl YMWUJEATGCHHMB-UHFFFAOYSA-N 0.000 abstract 3
- XEKOWRVHYACXOJ-UHFFFAOYSA-N Ethyl acetate Chemical compound CCOC(C)=O XEKOWRVHYACXOJ-UHFFFAOYSA-N 0.000 abstract 3
- LFQSCWFLJHTTHZ-UHFFFAOYSA-N Ethanol Chemical compound CCO LFQSCWFLJHTTHZ-UHFFFAOYSA-N 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 125000004122 cyclic group Chemical group 0.000 abstract 2
- 230000000843 anti-fungal effect Effects 0.000 abstract 1
- 229940121375 antifungal agent Drugs 0.000 abstract 1
- 239000004599 antimicrobial Substances 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 239000000126 substance Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/50—Cyclic peptides containing at least one abnormal peptide link
- C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
- C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Pulmonology (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2001263320A JP2005053782A (ja) | 2001-08-31 | 2001-08-31 | 環状リポペプチド化合物の新規結晶 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR036317A1 true AR036317A1 (es) | 2004-08-25 |
Family
ID=19090093
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP020103266A AR036317A1 (es) | 2001-08-31 | 2002-08-29 | Nuevo cristal de compuesto lipopeptido ciclico |
Country Status (3)
| Country | Link |
|---|---|
| JP (1) | JP2005053782A (fr) |
| AR (1) | AR036317A1 (fr) |
| WO (1) | WO2003018615A1 (fr) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW200826957A (en) | 2006-10-16 | 2008-07-01 | Teva Gyogyszergyar Zartkoruen Mukodo Reszvenytarsasag | Purification processes for echinocandin-type compounds |
| BR112013026420A2 (pt) * | 2011-04-20 | 2020-11-03 | Xellia Pharmaceuticals Aps | método de produção de um sal de micafungina farmaceuticamente aceitável |
| CN102627689B (zh) | 2012-03-30 | 2014-08-06 | 上海天伟生物制药有限公司 | 一种环肽类化合物的水合物及其制备方法和用途 |
| CN102627688B (zh) | 2012-03-30 | 2014-12-31 | 上海天伟生物制药有限公司 | 一种高纯度环肽化合物及其制备方法和用途 |
| CN102659930B (zh) * | 2012-03-30 | 2014-04-23 | 上海天伟生物制药有限公司 | 一种高纯度环肽类物质的晶体及其制备方法和用途 |
| JP6491325B2 (ja) * | 2014-05-29 | 2019-03-27 | シャンハイ テックウェル バイオファーマシューティカル カンパニー リミテッドShanghai Techwell Biopharmaceutical Co.,Ltd | シクロペプチド系化合物の溶媒和物およびその製造方法と使用 |
| WO2015180678A1 (fr) * | 2014-05-29 | 2015-12-03 | 上海天伟生物制药有限公司 | Cristal de composé peptidique cyclique, son procédé de préparation et ses utilisations |
| JP7109189B2 (ja) * | 2014-05-29 | 2022-07-29 | シャンハイ テックウェル バイオファーマシューティカル カンパニー リミテッド | シクロペプチド系化合物の組成物およびその製造方法と使用 |
| CN104788545B (zh) | 2014-05-29 | 2019-03-01 | 上海天伟生物制药有限公司 | 一种环肽类化合物的结晶粉末及其制备方法和用途 |
| CN108752430B (zh) * | 2018-05-31 | 2022-02-18 | 杭州中美华东制药有限公司 | 米卡芬净钠新晶型及其制备方法 |
| TW202430537A (zh) * | 2022-10-20 | 2024-08-01 | 日商中外製藥股份有限公司 | 環狀胜肽的結晶的製造方法 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5336756A (en) * | 1991-05-01 | 1994-08-09 | Merck & Co., Inc. | Process for crystalline cyclic lipopeptides |
| WO1996011210A1 (fr) * | 1994-10-07 | 1996-04-18 | Fujisawa Pharmaceutical Co., Ltd. | Hexapeptides cycliques a activite antibiotique |
| KR20020003864A (ko) * | 1999-03-03 | 2002-01-15 | 피터 지. 스트링거 | 에키노칸딘/탄수화물 착물 |
-
2001
- 2001-08-31 JP JP2001263320A patent/JP2005053782A/ja not_active Withdrawn
-
2002
- 2002-08-28 WO PCT/JP2002/008694 patent/WO2003018615A1/fr not_active Ceased
- 2002-08-29 AR ARP020103266A patent/AR036317A1/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| JP2005053782A (ja) | 2005-03-03 |
| WO2003018615A1 (fr) | 2003-03-06 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |