AR048197A1 - Metodos para tratar la esquizofrenia y/o anomalias de glucorregulacion - Google Patents

Metodos para tratar la esquizofrenia y/o anomalias de glucorregulacion

Info

Publication number
AR048197A1
AR048197A1 ARP050101275A ARP050101275A AR048197A1 AR 048197 A1 AR048197 A1 AR 048197A1 AR P050101275 A ARP050101275 A AR P050101275A AR P050101275 A ARP050101275 A AR P050101275A AR 048197 A1 AR048197 A1 AR 048197A1
Authority
AR
Argentina
Prior art keywords
alkyl
halogen
hydrogen
glucorregulation
independently hydrogen
Prior art date
Application number
ARP050101275A
Other languages
English (en)
Original Assignee
Aventis Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Inc filed Critical Aventis Pharma Inc
Publication of AR048197A1 publication Critical patent/AR048197A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Psychiatry (AREA)
  • Emergency Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

La presente proporciona composiciones farmacéuticas para tratar la esquizofrenia y/o anomalías de glucorregulacion en un paciente que lo necesite, que comprende una cantidad terapéuticamente eficaz de un compuesto de formula (1), en la que: M es 0, 1 o 2; n es 0, 1 o 2; p es 0 o 1; cada R es independientemente hidrogeno, halogeno, trifluorometilo, alquilo C1-6, alcoxi C1-6, benciloxi, hidroxi, nitro o amino; cada R1 es independientemente hidrogeno, alquilo C1-6, alquenilo C1-6, alcanoilo C1-6, halogeno, ciano, -C(O)-alquiloC1-6, -alquilenC1-6-CN, -alquilenC1-6-NR'R'' en el que R' y R'' son cada uno independientemente hidrogeno o alquilo C1-6, -alquilenC1-6-OC(O)-alquiloC1-6, o -CH(OH)R4 en el que R4 es hidrogeno o alquilo C1-6; R2 es hidrogeno, alquilo C1-6 opcionalmente sustituido con halogeno, hidroxi o benciloxi, alquenilo C1-6, alquinilo C1-6, -CO2-alquiloC1-6, o -R5-NR'R'' en el que R5 es alquileno C1-6, alquenileno C1-6 o alquinileno C1-6 y R' y R'' son cada uno independientemente hidrogeno, alquilo C1-6 o alternativamente el grupo -NR'R'' como un solo grupo es 1-pirrolidinilo; y R3 es hidrogeno, nitro, amino, halogeno, alcoxi C1-6, hidroxi o alquilo C1-6; o una de sus sales farmacéuticamente aceptable, y el uso de dichos compuestos para la fabricacion de un medicamento. Composiciones farmacéuticas para tratar la esquizofrenia en un ser humano que evita la propension concomitante de anomalías de glucorregulacion asociadas con la administracion de agentes antipsicoticos para administrar a dicho ser humano que comprende i) una cantidad terapéuticamente eficaz de un compuesto o una de sus sales farmacéuticamente aceptable, y ii) una cantidad terapéuticamente eficaz del agente antipsicotico y el uso de dichos compuestos para la fabricacion de un medicamento.
ARP050101275A 2004-04-01 2005-03-31 Metodos para tratar la esquizofrenia y/o anomalias de glucorregulacion AR048197A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US55845104P 2004-04-01 2004-04-01

Publications (1)

Publication Number Publication Date
AR048197A1 true AR048197A1 (es) 2006-04-05

Family

ID=34978926

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP050101275A AR048197A1 (es) 2004-04-01 2005-03-31 Metodos para tratar la esquizofrenia y/o anomalias de glucorregulacion

Country Status (26)

Country Link
US (1) US20070129403A1 (es)
EP (2) EP1734959B1 (es)
JP (1) JP2007531730A (es)
KR (1) KR20070010161A (es)
CN (1) CN1946399A (es)
AR (1) AR048197A1 (es)
AT (1) ATE446754T1 (es)
AU (1) AU2005231446A1 (es)
BR (1) BRPI0509512A (es)
CA (1) CA2561162A1 (es)
CL (1) CL2009001605A1 (es)
CY (1) CY1109734T1 (es)
DE (1) DE602005017373D1 (es)
DK (1) DK1734959T3 (es)
DO (1) DOP2005000050A (es)
ES (1) ES2334241T3 (es)
GT (1) GT200500063A (es)
IL (1) IL178168A0 (es)
MX (1) MXPA06011222A (es)
PA (1) PA8628601A1 (es)
PL (1) PL1734959T3 (es)
PT (1) PT1734959E (es)
SI (1) SI1734959T1 (es)
SV (1) SV2006002069A (es)
TW (1) TW200602040A (es)
WO (1) WO2005097122A2 (es)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR053710A1 (es) 2005-04-11 2007-05-16 Xenon Pharmaceuticals Inc Compuestos espiroheterociclicos y sus usos como agentes terapeuticos
AR056968A1 (es) 2005-04-11 2007-11-07 Xenon Pharmaceuticals Inc Compuestos espiro-oxindol y composiciones farmacéuticas
US20110294842A9 (en) * 2006-10-12 2011-12-01 Xenon Pharmaceuticals Inc. Spiro (furo [3, 2-c] pyridine-3-3' -indol) -2' (1'h)-one derivatives and related compounds for the treatment of sodium-channel mediated diseases, such as pain
WO2008060789A2 (en) 2006-10-12 2008-05-22 Xenon Pharmaceuticals Inc. Use of spiro-oxindole compounds as therapeutic agents
CA2741024A1 (en) 2008-10-17 2010-04-22 Xenon Pharmaceuticals Inc. Spiro-oxindole compounds and their use as therapeutic agents
JO3032B1 (ar) 2008-10-17 2016-09-05 Xenon Pharmaceuticals Inc مركبات سبيرو – اوكسندول وإستعمالاتها كعوامل علاجية.
WO2010068750A2 (en) * 2008-12-11 2010-06-17 Board Of Trustees Of Leland Stanford Junior University Compositons and method for treatment of mood and cognitive impairments
EP2437744B1 (en) * 2009-06-03 2015-06-03 Marquette University Modulation of kcnq potassium channel activity for treatment of psychiatric disorders and the symptoms thereof
AR077252A1 (es) 2009-06-29 2011-08-10 Xenon Pharmaceuticals Inc Enantiomeros de compuestos de espirooxindol y sus usos como agentes terapeuticos
KR20120099429A (ko) 2009-10-14 2012-09-10 제논 파마슈티칼스 인크. 스피로-옥스인돌 화합물의 합성 방법
WO2011106729A2 (en) 2010-02-26 2011-09-01 Xenon Pharmaceuticals Inc. Pharmaceutical compositions of spiro-oxindole compound for topical administration and their use as therapeutic agents
US11090297B2 (en) 2013-06-21 2021-08-17 Prilenia Neurotherapeutics Ltd. Pridopidine for treating huntington's disease
CN103512972A (zh) * 2013-07-29 2014-01-15 上海交通大学 精神分裂症的生物标志物及其使用方法和应用
WO2016127068A1 (en) 2015-02-05 2016-08-11 Teva Pharmaceuticals International Gmbh Methods of treating postherpetic neuralgia with a topical formulation of a spiro-oxindole compound
KR101759122B1 (ko) 2015-08-07 2017-07-18 계명대학교 산학협력단 오렉신 a를 함유하는 당뇨병 치료용 약학 조성물
EP4516356A3 (en) 2016-08-24 2025-05-14 Prilenia Neurotherapeutics Ltd. Use of pridopidine for treating functional decline
EP3941352A1 (en) 2019-03-19 2022-01-26 Cambridge Cognition Limited Method and uses of diagnosing and recommending treatment for a psychotic disorder

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0287982B1 (en) * 1987-04-24 1994-12-07 Hoechst-Roussel Pharmaceuticals Incorporated N-(Pyridinyl)-1H-indol-1-amines, a process for their preparation and their use as medicaments
US4970218A (en) 1987-04-24 1990-11-13 Hoechst-Roussel Pharmaceuticals Inc. N-(pyridinyl)-1H-indol-1-amines
US4880822A (en) * 1987-04-24 1989-11-14 Hoechst-Roussel Pharmaceuticals, Inc. N-(pyridinyl)-1H-indol-1-amines
US5102891A (en) * 1990-07-23 1992-04-07 Hoechst-Roussel Pharmaceuticals Inc. 1-(substituted pyridinylamino)-1H-indol-5-yl substituted carbamates
US5214038A (en) * 1991-04-15 1993-05-25 Hoechst-Roussel Pharmaceuticals Inc. 1-(pyrido[3,4-b]-1,4-oxazinyl-4-yl)-1H-indoles and intermediates for the preparation thereof
US5356910A (en) * 1993-07-19 1994-10-18 Hoechst-Roussel Pharmaceuticals Inc. Use of N-(pyridinyl)-1H-indol-1-amines for the treatment of obsessive-compulsive disorder
DE69621617T2 (de) * 1995-07-27 2003-01-02 Aventis Pharmaceuticals Inc., Bridgewater Verwendung von substituierten und nichtsubstituierten n-(pyrrol-1-yl)pyridinaminen als antikonvulsiva
EP0876379A1 (en) 1996-01-17 1998-11-11 Novo Nordisk A/S Fused 1,2,4-thiadiazine and fused 1,4-thiazine derivatives, their preparation and use
IL128332A0 (en) 1996-08-30 2000-01-31 Novo Nordisk As GLP-1 derivatives
DE19726167B4 (de) 1997-06-20 2008-01-24 Sanofi-Aventis Deutschland Gmbh Insulin, Verfahren zu seiner Herstellung und es enthaltende pharmazeutische Zubereitung
RU2215004C2 (ru) 1997-07-16 2003-10-27 Ново Нордиск А/С Конденсированное производное 1,2,4-тиадиазина, фармацевтическая композиция и способ получения лекарственного препарата
GB0119435D0 (en) * 2001-02-15 2001-10-03 Aventis Pharm Prod Inc Method of treating of demyelinating diseases or conditions

Also Published As

Publication number Publication date
GT200500063A (es) 2005-10-14
SI1734959T1 (sl) 2010-02-26
ATE446754T1 (de) 2009-11-15
PL1734959T3 (pl) 2010-03-31
US20070129403A1 (en) 2007-06-07
CY1109734T1 (el) 2014-09-10
CN1946399A (zh) 2007-04-11
DE602005017373D1 (de) 2009-12-10
EP1734959A2 (en) 2006-12-27
ES2334241T3 (es) 2010-03-08
IL178168A0 (en) 2006-12-31
CA2561162A1 (en) 2005-10-20
DOP2005000050A (es) 2005-11-30
WO2005097122A2 (en) 2005-10-20
EP2138176A1 (en) 2009-12-30
MXPA06011222A (es) 2007-01-16
PA8628601A1 (es) 2006-05-16
PT1734959E (pt) 2009-12-24
JP2007531730A (ja) 2007-11-08
AU2005231446A1 (en) 2005-10-20
WO2005097122A3 (en) 2006-02-02
EP1734959B1 (en) 2009-10-28
SV2006002069A (es) 2006-05-24
TW200602040A (en) 2006-01-16
CL2009001605A1 (es) 2009-11-27
KR20070010161A (ko) 2007-01-22
DK1734959T3 (da) 2010-03-08
BRPI0509512A (pt) 2007-09-11

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