AR211547A1 - Procedimiento para la preparacion de derivados de 3-fluor-5-fenil-1,4-benzodiazepina - Google Patents

Procedimiento para la preparacion de derivados de 3-fluor-5-fenil-1,4-benzodiazepina

Info

Publication number
AR211547A1
AR211547A1 AR264001A AR26400176A AR211547A1 AR 211547 A1 AR211547 A1 AR 211547A1 AR 264001 A AR264001 A AR 264001A AR 26400176 A AR26400176 A AR 26400176A AR 211547 A1 AR211547 A1 AR 211547A1
Authority
AR
Argentina
Prior art keywords
benzodiazepine
fluor
phenyl
derivatives
procedure
Prior art date
Application number
AR264001A
Other languages
English (en)
Original Assignee
Du Pont
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/687,318 external-priority patent/US4246270A/en
Application filed by Du Pont filed Critical Du Pont
Application granted granted Critical
Publication of AR211547A1 publication Critical patent/AR211547A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24—Oxygen atoms

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AR264001A 1975-07-21 1976-07-20 Procedimiento para la preparacion de derivados de 3-fluor-5-fenil-1,4-benzodiazepina AR211547A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US59750275A 1975-07-21 1975-07-21
US05/687,318 US4246270A (en) 1976-05-26 1976-05-26 3-Fluorobenzodiazepines and compositions and uses thereof

Publications (1)

Publication Number Publication Date
AR211547A1 true AR211547A1 (es) 1978-01-30

Family

ID=27082840

Family Applications (1)

Application Number Title Priority Date Filing Date
AR264001A AR211547A1 (es) 1975-07-21 1976-07-20 Procedimiento para la preparacion de derivados de 3-fluor-5-fenil-1,4-benzodiazepina

Country Status (22)

Country Link
JP (1) JPS5231087A (es)
AR (1) AR211547A1 (es)
AU (1) AU512991B2 (es)
CH (1) CH598234A5 (es)
DD (1) DD126767A5 (es)
DE (1) DE2632539A1 (es)
DK (1) DK326576A (es)
ES (1) ES449960A1 (es)
FI (1) FI762079A7 (es)
FR (1) FR2318643A1 (es)
GB (1) GB1553599A (es)
GR (1) GR60850B (es)
IL (1) IL50072A0 (es)
LU (1) LU75411A1 (es)
MX (1) MX3412E (es)
NL (1) NL7608074A (es)
NO (1) NO762525L (es)
NZ (1) NZ181516A (es)
PH (1) PH12173A (es)
PT (1) PT65383B (es)
SE (1) SE7606676L (es)
SU (1) SU683618A3 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4182760A (en) * 1977-06-16 1980-01-08 E. I. Du Pont De Nemours And Company Benzophenone anti-oximes, diazepin-N-oxides, and their use as pharmaceutical agents and as intermediates for pharmaceutical agents
JP2527717Y2 (ja) * 1991-07-19 1997-03-05 株式会社デンソー 車両用計器の取付け構造

Also Published As

Publication number Publication date
GB1553599A (en) 1979-09-26
LU75411A1 (es) 1978-02-08
NL7608074A (nl) 1977-01-25
AU1598876A (en) 1978-01-26
IL50072A0 (en) 1976-09-30
PT65383B (en) 1978-06-08
AU512991B2 (en) 1980-11-06
SE7606676L (sv) 1977-01-22
FR2318643A1 (fr) 1977-02-18
PH12173A (en) 1978-11-21
NZ181516A (en) 1978-04-28
FI762079A7 (es) 1977-01-22
DD126767A5 (es) 1977-08-10
DK326576A (da) 1977-01-22
CH598234A5 (es) 1978-04-28
NO762525L (es) 1977-01-24
GR60850B (en) 1978-08-31
PT65383A (en) 1976-08-01
DE2632539A1 (de) 1977-02-10
FR2318643B1 (es) 1980-10-17
MX3412E (es) 1980-11-06
JPS5231087A (en) 1977-03-09
ES449960A1 (es) 1977-12-01
SU683618A3 (ru) 1979-08-30

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