AT348523B - PROCESS FOR THE PRODUCTION OF NEW TETRAHYDROPYRIDINE AND PIPERIDINE DERIVATIVES AND THEIR ACID ADDITION SALTS - Google Patents

PROCESS FOR THE PRODUCTION OF NEW TETRAHYDROPYRIDINE AND PIPERIDINE DERIVATIVES AND THEIR ACID ADDITION SALTS

Info

Publication number
AT348523B
AT348523B AT667875A AT667875A AT348523B AT 348523 B AT348523 B AT 348523B AT 667875 A AT667875 A AT 667875A AT 667875 A AT667875 A AT 667875A AT 348523 B AT348523 B AT 348523B
Authority
AT
Austria
Prior art keywords
production
acid addition
addition salts
piperidine derivatives
tetrahydropyridine
Prior art date
Application number
AT667875A
Other languages
German (de)
Other versions
ATA667875A (en
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of ATA667875A publication Critical patent/ATA667875A/en
Application granted granted Critical
Publication of AT348523B publication Critical patent/AT348523B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/44Radicals substituted by doubly-bound oxygen, sulfur, or nitrogen atoms, or by two such atoms singly-bound to the same carbon atom
    • C07D213/46Oxygen atoms
    • C07D213/50Ketonic radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
AT667875A 1974-08-30 1975-08-29 PROCESS FOR THE PRODUCTION OF NEW TETRAHYDROPYRIDINE AND PIPERIDINE DERIVATIVES AND THEIR ACID ADDITION SALTS AT348523B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH1183774A CH605925A5 (en) 1974-08-30 1974-08-30
CH1511677A CH609980A5 (en) 1974-08-30 1974-08-30 Process for the preparation of novel piperidine derivatives

Publications (2)

Publication Number Publication Date
ATA667875A ATA667875A (en) 1978-07-15
AT348523B true AT348523B (en) 1979-02-26

Family

ID=25709012

Family Applications (1)

Application Number Title Priority Date Filing Date
AT667875A AT348523B (en) 1974-08-30 1975-08-29 PROCESS FOR THE PRODUCTION OF NEW TETRAHYDROPYRIDINE AND PIPERIDINE DERIVATIVES AND THEIR ACID ADDITION SALTS

Country Status (11)

Country Link
JP (1) JPS5148673A (en)
AT (1) AT348523B (en)
AU (1) AU499372B2 (en)
BE (1) BE832885A (en)
CA (1) CA1076118A (en)
CH (2) CH609980A5 (en)
DE (1) DE2537837A1 (en)
FR (1) FR2282887A1 (en)
GB (1) GB1510977A (en)
NL (1) NL7510142A (en)
SE (1) SE7508897L (en)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0006524A1 (en) * 1978-06-22 1980-01-09 Ciba-Geigy Ag Tetrahydropyridine and tetrahydropiperidine derivatives, their acid addition salts, processes for their preparation and pharmaceutical compositions containing them
US4490531A (en) * 1981-07-01 1984-12-25 The Upjohn Company Pyridyl-substituted-benzofurans
US4495357A (en) * 1981-07-01 1985-01-22 The Upjohn Company Pyridyl-substituted-benzofurans
US4455427A (en) * 1981-07-01 1984-06-19 The Upjohn Company Pyridyl-substituted-benzofurans
US4447620A (en) * 1982-06-08 1984-05-08 The Upjohn Company Imidazolyl-substituted benzothiophenes
US4452986A (en) * 1982-06-08 1984-06-05 The Upjohn Company Imidazolyl-substituted benzofurans
US4430502A (en) 1982-08-13 1984-02-07 The Upjohn Company Pyridinyl substituted benzimidazoles and quinoxalines
US4855435A (en) * 1982-10-12 1989-08-08 The Upjohn Company Pyridyl-substituted benzothiophenes
US4611059A (en) * 1982-10-12 1986-09-09 The Upjohn Company Pyridyl-substituted benzothiophenes
AU579647B2 (en) * 1985-02-21 1988-12-01 Asahi Kasei Kogyo Kabushiki Kaisha Process for adsorption treatment of dissolved fluorine
TW266206B (en) * 1993-04-28 1995-12-21 Takeda Pharm Industry Co Ltd
ATE189814T1 (en) * 1996-04-15 2000-03-15 Takeda Chemical Industries Ltd HYDROXYPYRIDINE DERIVATIVES, THEIR PREPARATION AND THEIR PHARMACEUTICAL USE
CA3240990A1 (en) * 2021-12-01 2023-06-08 Pfizer Inc. 3-phenyl-1-benzothiophene-2-carboxylic acid derivatives as branched-chain alpha keto acid dehydrogenase kinase inhibitors for the treatment of diabetes, kidney diseases, nash and heart failure

Also Published As

Publication number Publication date
CH605925A5 (en) 1978-10-13
FR2282887A1 (en) 1976-03-26
CA1076118A (en) 1980-04-22
JPS5148673A (en) 1976-04-26
NL7510142A (en) 1976-03-02
AU499372B2 (en) 1979-04-12
FR2282887B1 (en) 1980-04-18
GB1510977A (en) 1978-05-17
CH609980A5 (en) 1979-03-30
SE7508897L (en) 1976-03-01
DE2537837A1 (en) 1976-03-18
ATA667875A (en) 1978-07-15
AU8435675A (en) 1977-03-03
BE832885A (en) 1976-03-01

Similar Documents

Publication Publication Date Title
AT321912B (en) PROCESS FOR THE PRODUCTION OF NEW SUBSTITUTED PIPERIDINE DERIVATIVES AND THEIR ACID ADDITION SALTS
AT336000B (en) PROCESS FOR THE PRODUCTION OF NEW 3-PHENOXY-3-PHENYLPROPYLAMINES AND THEIR ACID ADDITIONAL SALTS
AT345833B (en) METHOD FOR PRODUCING NEW BENZIMIDAZOLINONE DERIVATIVES AND THEIR ACID ADDITION SALTS
AT348523B (en) PROCESS FOR THE PRODUCTION OF NEW TETRAHYDROPYRIDINE AND PIPERIDINE DERIVATIVES AND THEIR ACID ADDITION SALTS
AT336014B (en) PROCESS FOR THE PRODUCTION OF NEW TETRAHYDROPYRIDINE AND PIPERIDINE DERIVATIVES AND THEIR ACID ADDITION SALTS
ATA612476A (en) METHOD FOR THE PRODUCTION OF NEW PHENOXYAL CYCARBONIC ACID DERIVATIVES AND THEIR SALTS
ATA182577A (en) PROCESS FOR THE PRODUCTION OF NEW PIPERIDINE DERIVATIVES AND THEIR SALTS
ATA341575A (en) PROCESS FOR THE PRODUCTION OF NEW MORPHOLINE DERIVATIVES AND THEIR ACID ADDITION SALTS
AT340417B (en) PROCESS FOR THE PRODUCTION OF NEW XANTHENDER DERIVATIVES AND THEIR ACID ADDITION SALTS
ATA46475A (en) PROCESS FOR THE PRODUCTION OF NEW PHENTIAZINE DERIVATIVES AND THEIR ACID ADDITION SALTS
AT352728B (en) METHOD FOR PRODUCING NEW TETRAHYDROPYRIDINE AND PIPERIDINE DERIVATIVES AND THEIR ACID ADDITION SALTS
ATA404674A (en) PROCESS FOR THE PRODUCTION OF NEW PIPERIDINO ALCANONE DERIVATIVES AND THEIR ACID ADDITION SALTS
ATA307175A (en) METHOD FOR PRODUCING NEW PROSTANIC ACID DERIVATIVES AND THEIR SALTS
ATA606175A (en) METHOD FOR PRODUCING NEW PROSTANIC ACID DERIVATIVES AND THEIR SALTS
ATA224875A (en) PROCESS FOR THE PRODUCTION OF NEW INDOLOBENZA ACEPINES AND THEIR ACID ADDITIONAL SALTS
ATA419076A (en) PROCESS FOR THE PRODUCTION OF NEW TETRAHYDROPYRIDINE AND PIPERIDINE DERIVATIVES AND THEIR ACID ADDITION SALTS
ATA418876A (en) PROCESS FOR THE PRODUCTION OF NEW TETRAHYDROPYRIDINE AND PIPERIDINE DERIVATIVES AND THEIR ACID ADDITION SALTS
ATA419176A (en) PROCESS FOR THE PRODUCTION OF NEW TETRAHYDROPYRIDINE AND PIPERIDINE DERIVATIVES AND THEIR ACID ADDITION SALTS
AT289116B (en) PROCESS FOR THE PRODUCTION OF NEW PIPERIDINE DERIVATIVES AND THEIR ACID ADDITION SALTS
AT342594B (en) PROCESS FOR THE PRODUCTION OF NEW N- (P-FLUOROBENZOYLPROPYL) -4-PIPERIDYLAMIDES AND THEIR ACID ADDITION SALTS
ATA418976A (en) PROCESS FOR THE PRODUCTION OF NEW TETRAHYDROPYRIDE DERIVATIVES AND THEIR ACID ADDITION SALTS
AT352134B (en) PROCESS FOR THE PRODUCTION OF NEW TETRAHYDROPYRIDINE AND PIPERIDINE DERIVATIVES
ATA266877A (en) PROCESS FOR THE PRODUCTION OF NEW MORPHOLINE DERIVATIVES AND THEIR ACID ADDITION SALTS
ATA467278A (en) PROCESS FOR THE PRODUCTION OF NEW 2- (3-C3-C4- BRANCHED ALKYLAMINO-2-HYDROXY-PROPOXY) -3-CYANPYRIDINES AND THEIR ACID ADDITIONAL SALTS
ATA753676A (en) PROCESS FOR THE PRODUCTION OF NEW XANTHENDER DERIVATIVES AND THEIR ACID ADDITION SALTS

Legal Events

Date Code Title Description
ELJ Ceased due to non-payment of the annual fee