AT383736B - METHOD FOR PRODUCING WATER-SOLUBLE PHARMACEUTICAL COMPOSITIONS - Google Patents

METHOD FOR PRODUCING WATER-SOLUBLE PHARMACEUTICAL COMPOSITIONS

Info

Publication number
AT383736B
AT383736B AT0287185A AT287185A AT383736B AT 383736 B AT383736 B AT 383736B AT 0287185 A AT0287185 A AT 0287185A AT 287185 A AT287185 A AT 287185A AT 383736 B AT383736 B AT 383736B
Authority
AT
Austria
Prior art keywords
pharmaceutical compositions
producing water
soluble pharmaceutical
soluble
producing
Prior art date
Application number
AT0287185A
Other languages
German (de)
Other versions
ATA287185A (en
Inventor
Stefania Meola
Original Assignee
Schering Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Spa filed Critical Schering Spa
Publication of ATA287185A publication Critical patent/ATA287185A/en
Application granted granted Critical
Publication of AT383736B publication Critical patent/AT383736B/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/08—Solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18—Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • A61K47/183—Amino acids, e.g. glycine, EDTA or aspartame
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/655—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having oxygen atoms, with or without sulfur, selenium, or tellurium atoms, as the only ring hetero atoms
    • C07F9/65502—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having oxygen atoms, with or without sulfur, selenium, or tellurium atoms, as the only ring hetero atoms the oxygen atom being part of a three-membered ring
    • C07F9/65505—Phosphonic acids containing oxirane groups; esters thereof

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Dermatology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AT0287185A 1984-10-05 1985-10-03 METHOD FOR PRODUCING WATER-SOLUBLE PHARMACEUTICAL COMPOSITIONS AT383736B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH4792/84A CH660306A5 (en) 1984-10-05 1984-10-05 WATER-SOLUBLE PHARMACEUTICAL COMPOSITIONS BASED ON SALTS OF (-)CIS-1,2-EPOXYPROPYLPHOSPHONIC ACID WITH AMINO ACIDS.

Publications (2)

Publication Number Publication Date
ATA287185A ATA287185A (en) 1987-01-15
AT383736B true AT383736B (en) 1987-08-10

Family

ID=4282621

Family Applications (1)

Application Number Title Priority Date Filing Date
AT0287185A AT383736B (en) 1984-10-05 1985-10-03 METHOD FOR PRODUCING WATER-SOLUBLE PHARMACEUTICAL COMPOSITIONS

Country Status (11)

Country Link
JP (1) JPS62223121A (en)
KR (1) KR860003012A (en)
AT (1) AT383736B (en)
BE (1) BE903369A (en)
CH (1) CH660306A5 (en)
DE (1) DE3535356A1 (en)
ES (1) ES8609351A1 (en)
FR (1) FR2571255B1 (en)
GB (1) GB2165152B (en)
IT (1) IT1201479B (en)
NL (1) NL8502712A (en)

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1311956A (en) * 1969-10-02 1973-03-28 Merck & Co Inc Method of potentiating the activity of phosphonomycin antibiotics

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH310498A (en) * 1951-11-14 1955-10-31 Waldhof Zellstoff Fab Process for stabilizing alkali salts of adenosine polyphosphoric acids.
DE1767212B1 (en) * 1967-04-13 1971-05-06 Sumitomo Chemical Co Process for making injectable drugs
US3639590A (en) * 1967-07-25 1972-02-01 Merck & Co Inc Antibacterial composition containing (-) (cis-1 2-epoxypropyl) phosphoric acid
IT1161974B (en) * 1978-02-02 1987-03-18 Italchemi Spa CIS.I 2 EPOXYPROPYLPHOSPHONIC ACID DERIVATIVES THEIR PREPARATION PROCEDURE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
DE2813814A1 (en) * 1978-03-31 1979-10-18 Boehringer Mannheim Gmbh Increasing the enteral reabsorption of pharmaceuticals - by administration together with an aminoacid or a peptide
IT1112282B (en) * 1978-07-19 1986-01-13 Zambon Spa Bis- (2-AMMONIUM-2-hydroxymethyl-1,3-propanediol) (2R-CIS) - (3-METILOSSIRANIL) phosphonate
IT1097578B (en) * 1978-07-31 1985-08-31 Italchemi Spa METHOD FOR PREPARING ACID SALTS (-)
US4235900A (en) * 1978-11-15 1980-11-25 E. R. Squibb & Sons, Inc. Cephradine compositions

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1311956A (en) * 1969-10-02 1973-03-28 Merck & Co Inc Method of potentiating the activity of phosphonomycin antibiotics

Also Published As

Publication number Publication date
BE903369A (en) 1986-02-03
GB2165152B (en) 1988-03-16
NL8502712A (en) 1986-05-01
IT1201479B (en) 1989-02-02
ATA287185A (en) 1987-01-15
GB8524550D0 (en) 1985-11-06
CH660306A5 (en) 1987-04-15
FR2571255A1 (en) 1986-04-11
IT8522367A0 (en) 1985-10-04
ES8609351A1 (en) 1986-09-01
FR2571255B1 (en) 1988-09-16
JPS62223121A (en) 1987-10-01
DE3535356A1 (en) 1986-04-24
GB2165152A (en) 1986-04-09
ES547625A0 (en) 1986-09-01
KR860003012A (en) 1986-05-19

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Legal Events

Date Code Title Description
EIH Change in the person of patent owner
ELJ Ceased due to non-payment of the annual fee