ATA212290A - Verfahren zur grossproduktion von 1-((1-(2- (trifluormethyl)-4-pyrimidinyl)-4-piperidinyl)- methyl)-2-pyrrolidinon - Google Patents

Verfahren zur grossproduktion von 1-((1-(2- (trifluormethyl)-4-pyrimidinyl)-4-piperidinyl)- methyl)-2-pyrrolidinon

Info

Publication number
ATA212290A
ATA212290A AT0212290A AT212290A ATA212290A AT A212290 A ATA212290 A AT A212290A AT 0212290 A AT0212290 A AT 0212290A AT 212290 A AT212290 A AT 212290A AT A212290 A ATA212290 A AT A212290A
Authority
AT
Austria
Prior art keywords
trifluormethyl
pyrrolidinone
piperidinyl
pyrimidinyl
methyl
Prior art date
Application number
AT0212290A
Other languages
English (en)
Other versions
AT397961B (de
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of ATA212290A publication Critical patent/ATA212290A/de
Application granted granted Critical
Publication of AT397961B publication Critical patent/AT397961B/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Catalysts (AREA)
  • Silicon Polymers (AREA)
  • Macromonomer-Based Addition Polymer (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
AT0212290A 1989-10-27 1990-10-22 Verfahren zur grossproduktion von 1-((1-(2- (trifluormethyl)-4-pyrimidinyl)-4-piperidinyl)- methyl)-2-pyrrolidinon AT397961B (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/427,546 US4963678A (en) 1989-10-27 1989-10-27 Process for large-scale production of BMY 21502

Publications (2)

Publication Number Publication Date
ATA212290A true ATA212290A (de) 1993-12-15
AT397961B AT397961B (de) 1994-08-25

Family

ID=23695332

Family Applications (1)

Application Number Title Priority Date Filing Date
AT0212290A AT397961B (de) 1989-10-27 1990-10-22 Verfahren zur grossproduktion von 1-((1-(2- (trifluormethyl)-4-pyrimidinyl)-4-piperidinyl)- methyl)-2-pyrrolidinon

Country Status (12)

Country Link
US (1) US4963678A (de)
KR (1) KR910007917A (de)
CN (1) CN1032916C (de)
AT (1) AT397961B (de)
EG (1) EG19764A (de)
ES (1) ES2026059A6 (de)
FI (1) FI95467C (de)
GR (1) GR1001125B (de)
HU (1) HU206878B (de)
NO (1) NO177303C (de)
PT (1) PT95711B (de)
YU (1) YU203290A (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI95468C (fi) * 1989-10-27 1996-02-12 Squibb Bristol Myers Co Parannettu menetelmä käyttökelpoisten piperidiinijohdannaisten valmistamiseksi
HU206878B (en) * 1989-10-27 1993-01-28 Bristol Myers Squibb Co Process for producing 1-//1-/2-/trifluoromethyl/-4-pyrimidinyl/-4-piperidinyl/-methyl/-2-pirrolidinone
US5098904A (en) * 1990-06-27 1992-03-24 Bristol-Myers Squibb Company Cerebral function enhancing pyrimidinyl derivatives
US5401744A (en) * 1993-10-04 1995-03-28 Bristol-Myers Squibb Company Useful hemi-hydrate form of a cerebral function enhancing agent
US5538985A (en) * 1994-01-27 1996-07-23 Mitsui Toatsu Chemicals, Inc. Pyrrolidinone derivatives
BR0207975A (pt) 2001-03-15 2004-06-15 Basf Ag Composto, processo para preparar 5 fenilpiridinas, produto intermediário, agente adequado para combater fungos nocivos fitopatogênicos, e, processo para combater fungos nocivos fitopatogênicos
US7073271B2 (en) * 2002-02-14 2006-07-11 Faro Technologies Inc. Portable coordinate measurement machine
CN106883185B (zh) * 2015-12-15 2021-07-09 重庆博腾制药科技股份有限公司 一种4-氯-2-三氟甲基嘧啶的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4826843A (en) * 1985-07-08 1989-05-02 Bristol-Myers Cerebral function enhancing diazinylpiperidine derivatives
NZ216720A (en) * 1985-07-08 1990-09-26 Bristol Myers Co Diazinylpiperidine derivatives and pharmaceutical compositions
DE3703103A1 (de) * 1987-02-03 1988-08-11 Bayer Ag Mittel gegen fischparsiten
HU206878B (en) * 1989-10-27 1993-01-28 Bristol Myers Squibb Co Process for producing 1-//1-/2-/trifluoromethyl/-4-pyrimidinyl/-4-piperidinyl/-methyl/-2-pirrolidinone

Also Published As

Publication number Publication date
GR1001125B (el) 1993-04-28
FI95467C (fi) 1996-02-12
HU910050D0 (en) 1991-08-28
AT397961B (de) 1994-08-25
EG19764A (en) 1996-01-31
CN1032916C (zh) 1996-10-02
FI905225A0 (fi) 1990-10-24
NO177303B (no) 1995-05-15
NO904587D0 (no) 1990-10-24
NO904587L (no) 1991-04-29
ES2026059A6 (es) 1992-04-01
YU203290A (sh) 1993-10-20
NO177303C (no) 1995-08-23
PT95711B (pt) 1997-12-31
PT95711A (pt) 1991-09-13
US4963678A (en) 1990-10-16
KR910007917A (ko) 1991-05-30
FI95467B (fi) 1995-10-31
HU206878B (en) 1993-01-28
CN1051175A (zh) 1991-05-08
GR900100776A (en) 1992-03-20

Similar Documents

Publication Publication Date Title
DK8985A (da) 4-((bicyklisk heterocyclyl)-methyl og -hetero)-piperidin-derivater ogfremgangsmaade til fremstilling deraf
DE69407638D1 (de) Verfahren zur Fraktionierung von Blutmaterial
ATE181326T1 (de) Verfahren zu diastereoselektiven herstellung von nucleosid analoga
DE69322498D1 (de) Verfahren zur identifizierung von normalen biomedizinischen proben
ATE164079T1 (de) Verfahren zur behandlung von parasitären infektionen unter verwendung von ige-antagonisten
DE69807157D1 (de) Verfahren zur Rückgewinnung von Acrylsäure
DE69613770D1 (de) Verfahren zur Herstellung von Ethylen-Propylen-Copolymeren
DE59305971D1 (de) Verfahren zur entölung von rohlecithin
DE69305323D1 (de) Verfahren zur Herstellung von Äthylen-Propylen-Blockcopolymeren
DE69634457D1 (de) Verfahren zur Gewinnung von Butylacrylat das im wesentlichen keine Acrylsäure mehr enthält
ATE212380T1 (de) Verfahren zur herstellung von nikotinsäureamid
ATA212290A (de) Verfahren zur grossproduktion von 1-((1-(2- (trifluormethyl)-4-pyrimidinyl)-4-piperidinyl)- methyl)-2-pyrrolidinon
ATE207898T1 (de) Verfahren zur herstellung von acryl-piperidin- carbinolen
DE69414652D1 (de) Verbessertes Verfahren zur Bildung von Siliconkristallen
DE59607103D1 (de) Verfahren zur gewinnung von 2-hydroxy-4-methylthiobuttersäure (mha)
DE69409040D1 (de) Verfahren zur Entfärbung von Alkanolaminen
DE59604829D1 (de) Kontinuierliches Verfahren zur Herstellung von 4-Amino-2,2,6,6-tetramethylpiperidin
DE69806074D1 (de) Verfahren zur Rückgewinnung von Acrylsäure
DE59104247D1 (de) Verfahren zur Racemisierung von optisch aktiven 1-Aryl-alkylaminen.
DE68903228D1 (de) Verfahren zur fluoreszenzverbesserung von ti:al2o3-laser-kristallen.
DE69834276D1 (de) Verfahren zur Verbesserung der optischen Aktivität von Azetidin-2-carbonsäure
DE69514535D1 (de) Verfahren zur raffinierung von methylal
DE69937365D1 (de) Verfahren zur verwendung von aralkylsiloxanen
DE59007763D1 (de) Verfahren zur asymmetrischen Hydrierung von alpha-Ketocarbonyl-verbindungen zu optisch aktiven alpha-Hydroxycarbonylverbindungen.
DE59409261D1 (de) Verfahren zur Aufarbeitung von Dünnsäure

Legal Events

Date Code Title Description
ELJ Ceased due to non-payment of the annual fee