ATE205505T1 - Basische oxazolinamid-derivate von ge2270 und ge2270-änlichen antibiotika - Google Patents

Basische oxazolinamid-derivate von ge2270 und ge2270-änlichen antibiotika

Info

Publication number
ATE205505T1
ATE205505T1 AT96901344T AT96901344T ATE205505T1 AT E205505 T1 ATE205505 T1 AT E205505T1 AT 96901344 T AT96901344 T AT 96901344T AT 96901344 T AT96901344 T AT 96901344T AT E205505 T1 ATE205505 T1 AT E205505T1
Authority
AT
Austria
Prior art keywords
pct
antibiotics
basic
derivatives
oxazolinamide
Prior art date
Application number
AT96901344T
Other languages
English (en)
Inventor
Sergio Lociuro
Pierfausto Seneci
Romeo Ciabatti
Original Assignee
Biosearch Italia Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biosearch Italia Spa filed Critical Biosearch Italia Spa
Application granted granted Critical
Publication of ATE205505T1 publication Critical patent/ATE205505T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/05—Dipeptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
AT96901344T 1995-02-07 1996-02-01 Basische oxazolinamid-derivate von ge2270 und ge2270-änlichen antibiotika ATE205505T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP95101596 1995-02-07
PCT/EP1996/000425 WO1996024608A1 (en) 1995-02-07 1996-02-01 Basic oxazoline-amide derivatives of ge 2270 and ge 2270-like antibiotics

Publications (1)

Publication Number Publication Date
ATE205505T1 true ATE205505T1 (de) 2001-09-15

Family

ID=8218960

Family Applications (1)

Application Number Title Priority Date Filing Date
AT96901344T ATE205505T1 (de) 1995-02-07 1996-02-01 Basische oxazolinamid-derivate von ge2270 und ge2270-änlichen antibiotika

Country Status (13)

Country Link
US (1) US5891869A (de)
EP (1) EP0808326B1 (de)
JP (1) JP3518606B2 (de)
KR (1) KR100394930B1 (de)
AT (1) ATE205505T1 (de)
AU (1) AU693989B2 (de)
CA (1) CA2212437A1 (de)
DE (1) DE69615155T2 (de)
DK (1) DK0808326T3 (de)
ES (1) ES2161344T3 (de)
PT (1) PT808326E (de)
SI (1) SI0808326T1 (de)
WO (1) WO1996024608A1 (de)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE165101T1 (de) * 1995-02-07 1998-05-15 Biosearch Italia Spa Basische prolinamid derivate von ge2270 und ge2270-ahnlichten antibiotika
EP0880541B1 (de) * 1996-02-14 2003-01-15 Biosearch Italia S.p.A. Derivate des antibiotisch wirkenden faktors ge2270
WO2001077086A1 (en) * 2000-04-11 2001-10-18 Dupont Pharmaceuticals Company SUBSTITUTED LACTAMS AS INHIBITORS OF Aβ PROTEIN PRODUCTION
EP1565201B1 (de) * 2002-11-18 2018-10-31 Vicuron Pharmaceuticals, Inc. Methoden zur verabreichung von dalbavancin zur behandung bakterieller infektionen
US20060074014A1 (en) * 2002-11-18 2006-04-06 Vicuron Pharmaceuticals Inc. Dalbavancin compositions for treatment of bacterial infections
US7119061B2 (en) * 2002-11-18 2006-10-10 Vicuron Pharmaceuticals, Inc. Dalbavancin compositions for treatment of bacterial infections
US7023707B2 (en) * 2003-01-30 2006-04-04 Endicott Interconnect Technologies, Inc. Information handling system
US6828514B2 (en) * 2003-01-30 2004-12-07 Endicott Interconnect Technologies, Inc. High speed circuit board and method for fabrication
US7035113B2 (en) * 2003-01-30 2006-04-25 Endicott Interconnect Technologies, Inc. Multi-chip electronic package having laminate carrier and method of making same
CA2455024A1 (en) * 2003-01-30 2004-07-30 Endicott Interconnect Technologies, Inc. Stacked chip electronic package having laminate carrier and method of making same
PE20080103A1 (es) * 2006-05-31 2008-04-03 Novartis Ag AMINOTIAZOLES COMO MODULADORES DEL FACTOR DE ELONGACION EF-Tu
WO2008082562A2 (en) * 2006-12-20 2008-07-10 Novartis Ag Aminothiazole macrocycles, their use as antibacterial compounds and processes for their production
CA2708793C (en) 2007-12-12 2016-06-21 Novartis Ag Aminothiazoles and their uses

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5202241A (en) * 1988-09-09 1993-04-13 Gruppo Lepetit S.P.A. Antibiotic GE 2270
ES2066914T3 (es) * 1989-07-04 1995-03-16 Lepetit Spa Factores a1, a2, a3 y h del antibiotico ge 2270.
DK0451486T3 (da) * 1990-03-08 1995-05-08 Lepetit Spa Antibiotikum GE 2270 faktorer B1, B2, C1, C2, D1, D2, E og T
IL100572A (en) * 1991-01-03 1997-01-10 Lepetit Spa Amides of antibiotic ge 2270 factors their preparation and pharmaceutical compositions containing them
DE69224497T2 (de) * 1991-08-30 1998-07-02 Biosearch Italia Spa Faktor C2a des Antibiotikums CE 2270
ATE165101T1 (de) * 1995-02-07 1998-05-15 Biosearch Italia Spa Basische prolinamid derivate von ge2270 und ge2270-ahnlichten antibiotika
EP0880541B1 (de) * 1996-02-14 2003-01-15 Biosearch Italia S.p.A. Derivate des antibiotisch wirkenden faktors ge2270

Also Published As

Publication number Publication date
DK0808326T3 (da) 2001-10-01
KR19980701995A (ko) 1998-06-25
EP0808326A1 (de) 1997-11-26
KR100394930B1 (ko) 2003-12-18
CA2212437A1 (en) 1996-08-15
JPH10513461A (ja) 1998-12-22
WO1996024608A1 (en) 1996-08-15
DE69615155T2 (de) 2002-01-17
AU4540096A (en) 1996-08-27
PT808326E (pt) 2002-02-28
ES2161344T3 (es) 2001-12-01
US5891869A (en) 1999-04-06
AU693989B2 (en) 1998-07-09
JP3518606B2 (ja) 2004-04-12
EP0808326B1 (de) 2001-09-12
DE69615155D1 (de) 2001-10-18
SI0808326T1 (en) 2001-12-31

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Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification
EEIH Change in the person of patent owner
REN Ceased due to non-payment of the annual fee