ATE205505T1 - Basische oxazolinamid-derivate von ge2270 und ge2270-änlichen antibiotika - Google Patents

Basische oxazolinamid-derivate von ge2270 und ge2270-änlichen antibiotika

Info

Publication number
ATE205505T1
ATE205505T1 AT96901344T AT96901344T ATE205505T1 AT E205505 T1 ATE205505 T1 AT E205505T1 AT 96901344 T AT96901344 T AT 96901344T AT 96901344 T AT96901344 T AT 96901344T AT E205505 T1 ATE205505 T1 AT E205505T1
Authority
AT
Austria
Prior art keywords
pct
antibiotics
basic
derivatives
oxazolinamide
Prior art date
Application number
AT96901344T
Other languages
English (en)
Inventor
Sergio Lociuro
Pierfausto Seneci
Romeo Ciabatti
Original Assignee
Biosearch Italia Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biosearch Italia Spa filed Critical Biosearch Italia Spa
Application granted granted Critical
Publication of ATE205505T1 publication Critical patent/ATE205505T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06139Dipeptides with the first amino acid being heterocyclic
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/05Dipeptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
AT96901344T 1995-02-07 1996-02-01 Basische oxazolinamid-derivate von ge2270 und ge2270-änlichen antibiotika ATE205505T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP95101596 1995-02-07
PCT/EP1996/000425 WO1996024608A1 (en) 1995-02-07 1996-02-01 Basic oxazoline-amide derivatives of ge 2270 and ge 2270-like antibiotics

Publications (1)

Publication Number Publication Date
ATE205505T1 true ATE205505T1 (de) 2001-09-15

Family

ID=8218960

Family Applications (1)

Application Number Title Priority Date Filing Date
AT96901344T ATE205505T1 (de) 1995-02-07 1996-02-01 Basische oxazolinamid-derivate von ge2270 und ge2270-änlichen antibiotika

Country Status (13)

Country Link
US (1) US5891869A (de)
EP (1) EP0808326B1 (de)
JP (1) JP3518606B2 (de)
KR (1) KR100394930B1 (de)
AT (1) ATE205505T1 (de)
AU (1) AU693989B2 (de)
CA (1) CA2212437A1 (de)
DE (1) DE69615155T2 (de)
DK (1) DK0808326T3 (de)
ES (1) ES2161344T3 (de)
PT (1) PT808326E (de)
SI (1) SI0808326T1 (de)
WO (1) WO1996024608A1 (de)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100381688B1 (ko) * 1995-02-07 2003-12-11 바이오써치 이탈리아 에스.피.에이. Ge2270및ge2270-유사항생제의염기성프롤린-아미드유도체
CA2242067A1 (en) * 1996-02-14 1997-08-21 Versicor Inc. Derivatives of antibiotic ge2270 factors c2a, d2 and e
US6632812B2 (en) * 2000-04-11 2003-10-14 Dupont Pharmaceuticals Company Substituted lactams as inhibitors of Aβ protein production
US20060074014A1 (en) * 2002-11-18 2006-04-06 Vicuron Pharmaceuticals Inc. Dalbavancin compositions for treatment of bacterial infections
US20050090433A1 (en) * 2002-11-18 2005-04-28 Vicuron Pharmaceuticals, Inc Dalbavancin compositions for treatment of bacterial infections
US7119061B2 (en) * 2002-11-18 2006-10-10 Vicuron Pharmaceuticals, Inc. Dalbavancin compositions for treatment of bacterial infections
CA2455024A1 (en) * 2003-01-30 2004-07-30 Endicott Interconnect Technologies, Inc. Stacked chip electronic package having laminate carrier and method of making same
US7023707B2 (en) * 2003-01-30 2006-04-04 Endicott Interconnect Technologies, Inc. Information handling system
US7035113B2 (en) * 2003-01-30 2006-04-25 Endicott Interconnect Technologies, Inc. Multi-chip electronic package having laminate carrier and method of making same
US6828514B2 (en) * 2003-01-30 2004-12-07 Endicott Interconnect Technologies, Inc. High speed circuit board and method for fabrication
AR060977A1 (es) * 2006-05-31 2008-07-23 Novartis Ag Aminotiazoles y sus usos
ATE500259T1 (de) * 2006-12-20 2011-03-15 Novartis Ag Aminothiazolmakrocyclen, ihre verwendung als antibakterielle verbindungen und verfahren zu ihrer herstellung
NZ585788A (en) 2007-12-12 2011-07-29 Novartis Ag Aminothiazoles and their uses

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5202241A (en) * 1988-09-09 1993-04-13 Gruppo Lepetit S.P.A. Antibiotic GE 2270
DK0406745T3 (da) 1989-07-04 1995-02-27 Lepetit Spa Antibiotiske GE 2270 faktorer A1, A2, A3 og H
DK0451486T3 (da) * 1990-03-08 1995-05-08 Lepetit Spa Antibiotikum GE 2270 faktorer B1, B2, C1, C2, D1, D2, E og T
IL100572A (en) * 1991-01-03 1997-01-10 Lepetit Spa Amides of antibiotic ge 2270 factors their preparation and pharmaceutical compositions containing them
ES2113391T3 (es) * 1991-08-30 1998-05-01 Biosearch Italia Spa Factor c2a de antibiotico ge 2270.
KR100381688B1 (ko) * 1995-02-07 2003-12-11 바이오써치 이탈리아 에스.피.에이. Ge2270및ge2270-유사항생제의염기성프롤린-아미드유도체
CA2242067A1 (en) * 1996-02-14 1997-08-21 Versicor Inc. Derivatives of antibiotic ge2270 factors c2a, d2 and e

Also Published As

Publication number Publication date
KR19980701995A (ko) 1998-06-25
AU4540096A (en) 1996-08-27
AU693989B2 (en) 1998-07-09
US5891869A (en) 1999-04-06
CA2212437A1 (en) 1996-08-15
PT808326E (pt) 2002-02-28
JP3518606B2 (ja) 2004-04-12
WO1996024608A1 (en) 1996-08-15
DE69615155D1 (de) 2001-10-18
ES2161344T3 (es) 2001-12-01
EP0808326A1 (de) 1997-11-26
KR100394930B1 (ko) 2003-12-18
EP0808326B1 (de) 2001-09-12
DE69615155T2 (de) 2002-01-17
DK0808326T3 (da) 2001-10-01
JPH10513461A (ja) 1998-12-22
SI0808326T1 (en) 2001-12-31

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Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification
EEIH Change in the person of patent owner
REN Ceased due to non-payment of the annual fee