ATE209204T1 - Piperidinderivate. - Google Patents

Piperidinderivate.

Info

Publication number
ATE209204T1
ATE209204T1 AT96907664T AT96907664T ATE209204T1 AT E209204 T1 ATE209204 T1 AT E209204T1 AT 96907664 T AT96907664 T AT 96907664T AT 96907664 T AT96907664 T AT 96907664T AT E209204 T1 ATE209204 T1 AT E209204T1
Authority
AT
Austria
Prior art keywords
piperidine derivatives
represents hydrogen
lower alkyl
antagonism
vomiting
Prior art date
Application number
AT96907664T
Other languages
English (en)
Inventor
Yoshihiro Tanoue
Koichi Beppu
Akira Okayama
Osami Sakamoto
Original Assignee
Hisamitsu Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hisamitsu Pharmaceutical Co filed Critical Hisamitsu Pharmaceutical Co
Application granted granted Critical
Publication of ATE209204T1 publication Critical patent/ATE209204T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Otolaryngology (AREA)
  • Hospice & Palliative Care (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
AT96907664T 1995-03-27 1996-03-27 Piperidinderivate. ATE209204T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP9315095 1995-03-27
PCT/JP1996/000796 WO1996030367A1 (en) 1995-03-27 1996-03-27 Piperidine derivatives

Publications (1)

Publication Number Publication Date
ATE209204T1 true ATE209204T1 (de) 2001-12-15

Family

ID=14074519

Family Applications (1)

Application Number Title Priority Date Filing Date
AT96907664T ATE209204T1 (de) 1995-03-27 1996-03-27 Piperidinderivate.

Country Status (9)

Country Link
US (1) US5886011A (de)
EP (1) EP0826684B1 (de)
JP (1) JP3992733B2 (de)
KR (1) KR19980703354A (de)
AT (1) ATE209204T1 (de)
AU (1) AU696948B2 (de)
CA (1) CA2216701A1 (de)
DE (1) DE69617226T2 (de)
WO (1) WO1996030367A1 (de)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW340842B (en) 1995-08-24 1998-09-21 Pfizer Substituted benzylaminopiperidine compounds
TW426667B (en) * 1997-11-19 2001-03-21 Pfizer Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance P antagonists
TW537894B (en) * 1998-05-26 2003-06-21 Novartis Ag A spontaneously dispersible pharmaceutical composition comprising a piperidine substance P antagonist
ES2251217T3 (es) 1998-09-09 2006-04-16 Kewpie Kabushiki Kaisha Alimentos para la prevencion de vomitos.
EP1178984B1 (de) * 1999-05-21 2003-03-19 Pfizer Products Inc. 1-trifluorotmethyl-4-hydroxy-7-piperidinyl-aminomethylchroman-derivate
WO2001025233A1 (en) * 1999-10-07 2001-04-12 Hisamitsu Pharmaceutical Co., Inc. Piperidine derivatives
EP1095939B1 (de) * 1999-10-18 2004-01-07 Pfizer Products Inc. Verfahren zur Herstellung von zyklischen Piperidinylaminomethyl-trifluoromethyl-etherderivaten
EP1170006B8 (de) * 1999-12-14 2008-03-19 Teikoku Seiyaku Co., Ltd. Arzneimittel zur behandlung der hemicrania
US7728155B2 (en) 2003-10-24 2010-06-01 Wyeth Llc Dihydrobenzofuranyl alkanamines and methods for using same as cns agents
US7435837B2 (en) 2003-10-24 2008-10-14 Wyeth Dihydrobenzofuranyl alkanamine derivatives and methods for using same
US20070218143A1 (en) * 2006-03-20 2007-09-20 Chong Mok T M Topical preparation
ES2672099T3 (es) 2011-07-04 2018-06-12 Irbm - Science Park S.P.A. Antagonistas del receptor NK-1 para el tratamiento de la neovascularización corneal
EP3758688B1 (de) 2018-02-26 2024-03-27 Ospedale San Raffaele S.r.l. Nk-1-antagonisten zur verwendung bei der behandlung von augenschmerzen
EP4117673A1 (de) 2020-03-11 2023-01-18 Ospedale San Raffaele S.r.l. Behandlung von stammzellenmangel

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5232929A (en) * 1990-11-28 1993-08-03 Pfizer Inc. 3-aminopiperidine derivatives and related nitrogen containing heterocycles and pharmaceutical compositions and use
JPH0794440B2 (ja) * 1991-03-26 1995-10-11 フアイザー・インコーポレイテツド 置換ピペリジンの立体選択的製造
EP0675886B1 (de) * 1992-12-10 2000-07-05 Pfizer Inc. Aminomethylen substituierte heterocyclische verbindungen und ihre verwendung alssubstanz p antagonisten
US5393762A (en) * 1993-06-04 1995-02-28 Pfizer Inc. Pharmaceutical agents for treatment of emesis

Also Published As

Publication number Publication date
US5886011A (en) 1999-03-23
KR19980703354A (ko) 1998-10-15
EP0826684B1 (de) 2001-11-21
DE69617226D1 (de) 2002-01-03
DE69617226T2 (de) 2002-07-25
AU5120296A (en) 1996-10-16
JP3992733B2 (ja) 2007-10-17
EP0826684A1 (de) 1998-03-04
EP0826684A4 (de) 1998-07-08
WO1996030367A1 (en) 1996-10-03
AU696948B2 (en) 1998-09-24
CA2216701A1 (en) 1996-10-03

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Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties