ATE209204T1 - Piperidinderivate. - Google Patents

Piperidinderivate.

Info

Publication number
ATE209204T1
ATE209204T1 AT96907664T AT96907664T ATE209204T1 AT E209204 T1 ATE209204 T1 AT E209204T1 AT 96907664 T AT96907664 T AT 96907664T AT 96907664 T AT96907664 T AT 96907664T AT E209204 T1 ATE209204 T1 AT E209204T1
Authority
AT
Austria
Prior art keywords
piperidine derivatives
represents hydrogen
lower alkyl
antagonism
vomiting
Prior art date
Application number
AT96907664T
Other languages
English (en)
Inventor
Yoshihiro Tanoue
Koichi Beppu
Akira Okayama
Osami Sakamoto
Original Assignee
Hisamitsu Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hisamitsu Pharmaceutical Co filed Critical Hisamitsu Pharmaceutical Co
Application granted granted Critical
Publication of ATE209204T1 publication Critical patent/ATE209204T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pulmonology (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
AT96907664T 1995-03-27 1996-03-27 Piperidinderivate. ATE209204T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP9315095 1995-03-27
PCT/JP1996/000796 WO1996030367A1 (en) 1995-03-27 1996-03-27 Piperidine derivatives

Publications (1)

Publication Number Publication Date
ATE209204T1 true ATE209204T1 (de) 2001-12-15

Family

ID=14074519

Family Applications (1)

Application Number Title Priority Date Filing Date
AT96907664T ATE209204T1 (de) 1995-03-27 1996-03-27 Piperidinderivate.

Country Status (9)

Country Link
US (1) US5886011A (de)
EP (1) EP0826684B1 (de)
JP (1) JP3992733B2 (de)
KR (1) KR19980703354A (de)
AT (1) ATE209204T1 (de)
AU (1) AU696948B2 (de)
CA (1) CA2216701A1 (de)
DE (1) DE69617226T2 (de)
WO (1) WO1996030367A1 (de)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW340842B (en) 1995-08-24 1998-09-21 Pfizer Substituted benzylaminopiperidine compounds
TW426667B (en) * 1997-11-19 2001-03-21 Pfizer Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance P antagonists
TW537894B (en) * 1998-05-26 2003-06-21 Novartis Ag A spontaneously dispersible pharmaceutical composition comprising a piperidine substance P antagonist
EP1029456B1 (de) 1998-09-09 2005-11-09 Kewpie Kabushiki Kaisha Brechreizunterdrueckende nahrungsmittel
IL145949A0 (en) * 1999-05-21 2002-07-25 Pfizer Prod Inc 1-trifluoromethyl-4-hydroxy-7-piperidinyl-aminomethylchroman derivatives
AU7557000A (en) * 1999-10-07 2001-05-10 Hisamitsu Pharmaceutical Co. Inc. Piperidine derivatives
PT1095939E (pt) * 1999-10-18 2004-04-30 Pfizer Prod Inc Processo para a preparacao de eteres ciclicos de compostos com piperidinilaminometilo
EP1170006B8 (de) * 1999-12-14 2008-03-19 Teikoku Seiyaku Co., Ltd. Arzneimittel zur behandlung der hemicrania
US7728155B2 (en) 2003-10-24 2010-06-01 Wyeth Llc Dihydrobenzofuranyl alkanamines and methods for using same as cns agents
US7435837B2 (en) 2003-10-24 2008-10-14 Wyeth Dihydrobenzofuranyl alkanamine derivatives and methods for using same
US20070218143A1 (en) * 2006-03-20 2007-09-20 Chong Mok T M Topical preparation
WO2013004766A1 (en) 2011-07-04 2013-01-10 Ferrari Giulio Nk-1 receptor antagonists for treating corneal neovascularisation
RU2020131446A (ru) 2018-02-26 2022-03-28 Оспедале Сан Раффаэле С.Р.Л. Антагонисты nk-1 для применения в лечении глазной боли
EP4117673A1 (de) 2020-03-11 2023-01-18 Ospedale San Raffaele S.r.l. Behandlung von stammzellenmangel

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5232929A (en) * 1990-11-28 1993-08-03 Pfizer Inc. 3-aminopiperidine derivatives and related nitrogen containing heterocycles and pharmaceutical compositions and use
AU647592B2 (en) * 1991-03-26 1994-03-24 Pfizer Inc. Stereoselective preparation of substituted piperidines
ES2147759T3 (es) * 1992-12-10 2000-10-01 Pfizer Heterociclos no aromaticos sustituidos con aminometileno y uso como antagonistas de la sustancia p.
US5393762A (en) * 1993-06-04 1995-02-28 Pfizer Inc. Pharmaceutical agents for treatment of emesis

Also Published As

Publication number Publication date
CA2216701A1 (en) 1996-10-03
DE69617226T2 (de) 2002-07-25
EP0826684A4 (de) 1998-07-08
AU5120296A (en) 1996-10-16
US5886011A (en) 1999-03-23
AU696948B2 (en) 1998-09-24
EP0826684B1 (de) 2001-11-21
JP3992733B2 (ja) 2007-10-17
WO1996030367A1 (en) 1996-10-03
DE69617226D1 (de) 2002-01-03
EP0826684A1 (de) 1998-03-04
KR19980703354A (ko) 1998-10-15

Similar Documents

Publication Publication Date Title
AU696948B2 (en) Piperidine derivatives
CA2124680A1 (en) Piperazine derivatives as 5-ht1a antagonists
NO953305D0 (no) Antranilsyrederivat
AU9281198A (en) Benzofuran derivatives
DE69717970D1 (de) Chinolin carbonsaure-derivate und ihre salze
DK0695755T3 (da) Pyrrolocarbazoler
DE69122941D1 (de) Piperazinderivate
ATE252074T1 (de) Phenylalkylcarbonsäure-derivate
DE69621469D1 (de) Phenylpiperidin-derivate
DE69019293D1 (de) Naphthyloxazolidon-Derivate.
ATE231487T1 (de) 2-phenoxyanilin-derivate
PT1122253E (pt) Derivados de quinazolinona
EP1219619A4 (de) Piperidinderivate
AU4370489A (en) The use of oxidized polyamines, especially nn'-bis-(3- propionaldehyde)-1-4-diaminobutane (sperminedialdehyde) as immunosuppressive agents
DE60103732D1 (de) Pyrimidinderivate mit antitumor-wirkung

Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties