ATE242631T1 - Transdermale verabreichung von risperidon mit kontrollierter geschwindigkeit - Google Patents

Transdermale verabreichung von risperidon mit kontrollierter geschwindigkeit

Info

Publication number
ATE242631T1
ATE242631T1 AT96908146T AT96908146T ATE242631T1 AT E242631 T1 ATE242631 T1 AT E242631T1 AT 96908146 T AT96908146 T AT 96908146T AT 96908146 T AT96908146 T AT 96908146T AT E242631 T1 ATE242631 T1 AT E242631T1
Authority
AT
Austria
Prior art keywords
risperidone
transdermal administration
controlled rate
controlled
rate
Prior art date
Application number
AT96908146T
Other languages
English (en)
Inventor
Jean Louis Mesens
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Application granted granted Critical
Publication of ATE242631T1 publication Critical patent/ATE242631T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
    • A61K9/7053—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
    • A61K9/7061—Polyacrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Dermatology (AREA)
  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AT96908146T 1995-04-06 1996-03-29 Transdermale verabreichung von risperidon mit kontrollierter geschwindigkeit ATE242631T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP95200867 1995-04-06
PCT/EP1996/001421 WO1996031201A1 (en) 1995-04-06 1996-03-29 Rate-controlled transdermal administration of risperidone

Publications (1)

Publication Number Publication Date
ATE242631T1 true ATE242631T1 (de) 2003-06-15

Family

ID=8220172

Family Applications (1)

Application Number Title Priority Date Filing Date
AT96908146T ATE242631T1 (de) 1995-04-06 1996-03-29 Transdermale verabreichung von risperidon mit kontrollierter geschwindigkeit

Country Status (16)

Country Link
EP (1) EP0879051B9 (de)
JP (1) JPH11503138A (de)
KR (1) KR100437672B1 (de)
AR (1) AR003413A1 (de)
AT (1) ATE242631T1 (de)
CA (1) CA2214420A1 (de)
CY (1) CY2388B1 (de)
DE (1) DE69628672T2 (de)
DK (1) DK0879051T3 (de)
ES (1) ES2201176T3 (de)
HR (1) HRP960154A2 (de)
IL (1) IL117809A (de)
PT (1) PT879051E (de)
TW (1) TW592729B (de)
WO (1) WO1996031201A1 (de)
ZA (1) ZA962752B (de)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10042412B4 (de) * 2000-08-30 2005-12-22 Lts Lohmann Therapie-Systeme Ag Transdermales therapeutisches System zur Abgabe von Venlafaxin, und seine Verwendung
US20050232995A1 (en) 2002-07-29 2005-10-20 Yam Nyomi V Methods and dosage forms for controlled delivery of paliperidone and risperidone
DE602005010812D1 (de) * 2004-11-22 2008-12-18 Hisamitsu Pharmaceutical Co Transdermales Pflaster enthaltend einen schmelzpunktsenkenden Hilfsstoff
JP4914826B2 (ja) * 2005-02-28 2012-04-11 久光製薬株式会社 経皮吸収製剤
WO2007035942A2 (en) * 2005-09-23 2007-03-29 Alza Corporation Transdermal risperidone delivery system
AU2007255724B2 (en) 2006-06-09 2012-05-10 Dainippon Sumitomo Pharma Co., Ltd. Novel tape preparation
DE102007006244B4 (de) 2007-02-08 2012-03-15 Lts Lohmann Therapie-Systeme Ag Transdermales Therapeutisches System zur Verabreichung wasserlöslicher Wirkstoffe
EP2230911A4 (de) * 2007-12-21 2013-07-03 Zars Pharma Inc Patches, Formulierungen und entsprechende Verfahren für die perkutane Applikation von Alprazolam und anderen Arzeneimitteln
JPWO2010098261A1 (ja) * 2009-02-24 2012-08-30 久光製薬株式会社 リスペリドン含有経皮吸収型製剤及びこれを用いた貼付剤
JP2025528758A (ja) * 2023-01-04 2025-09-02 新領医薬技術(深▲せん▼)有限公司 リスペリドン経皮投与システム及びその製造方法と用途

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3854480A (en) * 1969-04-01 1974-12-17 Alza Corp Drug-delivery system
US4804663A (en) * 1985-03-27 1989-02-14 Janssen Pharmaceutica N.V. 3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles
US4710191A (en) * 1985-12-16 1987-12-01 Jonergin, Inc. Therapeutic device for the administration of medicaments
US4938759A (en) * 1986-09-02 1990-07-03 Alza Corporation Transdermal delivery device having a rate controlling adhesive
US5788983A (en) * 1989-04-03 1998-08-04 Rutgers, The State University Of New Jersey Transdermal controlled delivery of pharmaceuticals at variable dosage rates and processes
WO1991002527A1 (en) * 1989-08-21 1991-03-07 Beth Israel Hospital Association Method and composition for the treatment of cutaneous, ocular, and mucosal hypersensitivity, inflammation, and hyperproliferative conditions using topical preparations of serotonin antagonists

Also Published As

Publication number Publication date
CY2388B1 (en) 2004-09-10
AR003413A1 (es) 1998-08-05
HRP960154A2 (en) 1997-08-31
ZA962752B (en) 1997-10-06
JPH11503138A (ja) 1999-03-23
EP0879051A1 (de) 1998-11-25
WO1996031201A1 (en) 1996-10-10
ES2201176T3 (es) 2004-03-16
IL117809A0 (en) 1996-08-04
AU696789B2 (en) 1998-09-17
TW592729B (en) 2004-06-21
DK0879051T3 (da) 2003-09-29
AU5149296A (en) 1996-10-23
EP0879051B9 (de) 2004-03-03
KR100437672B1 (ko) 2004-09-10
PT879051E (pt) 2003-10-31
HK1015681A1 (en) 1999-10-22
EP0879051B1 (de) 2003-06-11
DE69628672D1 (de) 2003-07-17
IL117809A (en) 2000-10-31
DE69628672T2 (de) 2004-04-29
CA2214420A1 (en) 1996-10-10

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