ATE255896T1 - Tetrahydropteridine und pyridylpiperazine zur behandlung von neurologischen störungen - Google Patents

Tetrahydropteridine und pyridylpiperazine zur behandlung von neurologischen störungen

Info

Publication number
ATE255896T1
ATE255896T1 AT97926590T AT97926590T ATE255896T1 AT E255896 T1 ATE255896 T1 AT E255896T1 AT 97926590 T AT97926590 T AT 97926590T AT 97926590 T AT97926590 T AT 97926590T AT E255896 T1 ATE255896 T1 AT E255896T1
Authority
AT
Austria
Prior art keywords
neurological disorders
pyridylpiperazine
tetrahydropteridine
treatment
crf
Prior art date
Application number
AT97926590T
Other languages
English (en)
Inventor
Richard Gerald Wilde
Original Assignee
Bristol Myers Squibb Pharma Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Pharma Co filed Critical Bristol Myers Squibb Pharma Co
Application granted granted Critical
Publication of ATE255896T1 publication Critical patent/ATE255896T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D475/00—Heterocyclic compounds containing pteridine ring systems
    • C07D475/06—Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Immunology (AREA)
  • Psychiatry (AREA)
  • Transplantation (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Addiction (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AT97926590T 1996-05-23 1997-05-19 Tetrahydropteridine und pyridylpiperazine zur behandlung von neurologischen störungen ATE255896T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US1819896P 1996-05-23 1996-05-23
PCT/US1997/008448 WO1997044038A1 (en) 1996-05-23 1997-05-19 Tetrahydropteridines and pyridylpiperazines for treatment of neurological disorders

Publications (1)

Publication Number Publication Date
ATE255896T1 true ATE255896T1 (de) 2003-12-15

Family

ID=21786748

Family Applications (1)

Application Number Title Priority Date Filing Date
AT97926590T ATE255896T1 (de) 1996-05-23 1997-05-19 Tetrahydropteridine und pyridylpiperazine zur behandlung von neurologischen störungen

Country Status (14)

Country Link
US (3) US6083948A (de)
EP (1) EP0901374B1 (de)
JP (1) JP2000511183A (de)
AT (1) ATE255896T1 (de)
AU (1) AU739269B2 (de)
CA (1) CA2255650A1 (de)
DE (1) DE69726724T2 (de)
DK (1) DK0901374T3 (de)
ES (1) ES2213216T3 (de)
IL (1) IL127170A0 (de)
NZ (1) NZ332704A (de)
PT (1) PT901374E (de)
WO (1) WO1997044038A1 (de)
ZA (1) ZA973884B (de)

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AU2001255673A1 (en) * 2000-05-01 2001-11-12 Dupont Pharmaceuticals Company Tricyclic fused pyridine and pyrimidine derivatives as crf receptor antagonists
EP1287002A1 (de) 2000-05-18 2003-03-05 Neurocrine Biosciences, Inc. Crf rezeptor-antagonisten
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US20090137550A1 (en) * 2005-03-25 2009-05-28 Glaxo Group Limited Novel Compounds
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AU2006275694A1 (en) * 2005-07-28 2007-02-08 Bristol-Myers Squibb Company Substituted tetrahydro-1H-pyrido(4,3,b)indoles as serotonin receptor agonists and antagonists
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AR060432A1 (es) * 2006-04-12 2008-06-18 Vertex Pharma Tetrahidropteridinas utiles como inhibidores de las proteinas quinasas
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Also Published As

Publication number Publication date
PT901374E (pt) 2004-04-30
WO1997044038A1 (en) 1997-11-27
ZA973884B (en) 1998-11-06
US6083948A (en) 2000-07-04
ES2213216T3 (es) 2004-08-16
DE69726724D1 (de) 2004-01-22
US6399609B1 (en) 2002-06-04
NZ332704A (en) 2000-05-26
EP0901374A1 (de) 1999-03-17
DE69726724T2 (de) 2004-12-09
IL127170A0 (en) 1999-09-22
JP2000511183A (ja) 2000-08-29
US20030064993A1 (en) 2003-04-03
DK0901374T3 (da) 2004-04-05
AU3131697A (en) 1997-12-09
EP0901374A4 (de) 2001-05-09
AU739269B2 (en) 2001-10-11
CA2255650A1 (en) 1997-11-27
US6869955B2 (en) 2005-03-22
EP0901374B1 (de) 2003-12-10

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