ATE260272T1 - Beta-aminsäure-derivate zur verwendung als matrix-metalloproteasen- und tna-alpha-inhibitoren - Google Patents

Beta-aminsäure-derivate zur verwendung als matrix-metalloproteasen- und tna-alpha-inhibitoren

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Publication number
ATE260272T1
ATE260272T1 AT01924171T AT01924171T ATE260272T1 AT E260272 T1 ATE260272 T1 AT E260272T1 AT 01924171 T AT01924171 T AT 01924171T AT 01924171 T AT01924171 T AT 01924171T AT E260272 T1 ATE260272 T1 AT E260272T1
Authority
AT
Austria
Prior art keywords
tna
beta
amino acid
acid derivatives
matrix metalloproteases
Prior art date
Application number
AT01924171T
Other languages
English (en)
Inventor
Jingwu Duan
Bryan W King
Carl Decicco
Thomas P Maduskuie Jr
Matthew E Voss
Original Assignee
Bristol Myers Squibb Pharma Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Pharma Co filed Critical Bristol Myers Squibb Pharma Co
Application granted granted Critical
Publication of ATE260272T1 publication Critical patent/ATE260272T1/de

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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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AT01924171T 2000-03-17 2001-03-15 Beta-aminsäure-derivate zur verwendung als matrix-metalloproteasen- und tna-alpha-inhibitoren ATE260272T1 (de)

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US19018300P 2000-03-17 2000-03-17
US23546700P 2000-09-26 2000-09-26
US25206200P 2000-11-20 2000-11-20
PCT/US2001/008336 WO2001070734A2 (en) 2000-03-17 2001-03-15 Beta-amino acid derivatives as inhibitors of matrix metalloproteases and tnf-alpha

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DE60102137D1 (de) 2004-04-01
ES2215893T3 (es) 2004-10-16
US20020013341A1 (en) 2002-01-31
BR0109469A (pt) 2003-04-29
NZ521245A (en) 2004-04-30
CA2400168A1 (en) 2001-09-27
WO2001070734A2 (en) 2001-09-27
CN1420881A (zh) 2003-05-28
HK1049334A1 (en) 2003-05-09
EP1263756A2 (de) 2002-12-11
WO2001070734A3 (en) 2002-03-14
US6495565B2 (en) 2002-12-17
AU2001250850A1 (en) 2001-10-03
IL151018A0 (en) 2003-02-12
AR035174A1 (es) 2004-05-05
HK1049334B (en) 2004-07-16
DE60102137T2 (de) 2004-10-21
EP1263756B1 (de) 2004-02-25
JP2003528097A (ja) 2003-09-24

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