ATE315382T1 - Pharmazeutische zusammensetzungen zur oralen verabreichung, die einen magensaftresistenten überzug auf der basis von acrylatpolymeren enthalten - Google Patents
Pharmazeutische zusammensetzungen zur oralen verabreichung, die einen magensaftresistenten überzug auf der basis von acrylatpolymeren enthaltenInfo
- Publication number
- ATE315382T1 ATE315382T1 AT99122470T AT99122470T ATE315382T1 AT E315382 T1 ATE315382 T1 AT E315382T1 AT 99122470 T AT99122470 T AT 99122470T AT 99122470 T AT99122470 T AT 99122470T AT E315382 T1 ATE315382 T1 AT E315382T1
- Authority
- AT
- Austria
- Prior art keywords
- pharmaceutical compositions
- oral administration
- entericial
- resistant coating
- acrylate polymers
- Prior art date
Links
- 239000011248 coating agent Substances 0.000 title abstract 2
- 238000000576 coating method Methods 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 229920000058 polyacrylate Polymers 0.000 title 1
- 239000004480 active ingredient Substances 0.000 abstract 3
- BAPJBEWLBFYGME-UHFFFAOYSA-N Methyl acrylate Chemical compound COC(=O)C=C BAPJBEWLBFYGME-UHFFFAOYSA-N 0.000 abstract 2
- CERQOIWHTDAKMF-UHFFFAOYSA-N Methacrylic acid Chemical compound CC(=C)C(O)=O CERQOIWHTDAKMF-UHFFFAOYSA-N 0.000 abstract 1
- VVQNEPGJFQJSBK-UHFFFAOYSA-N Methyl methacrylate Chemical compound COC(=O)C(C)=C VVQNEPGJFQJSBK-UHFFFAOYSA-N 0.000 abstract 1
- 230000002757 inflammatory effect Effects 0.000 abstract 1
- 208000028774 intestinal disease Diseases 0.000 abstract 1
- 210000000936 intestine Anatomy 0.000 abstract 1
- 230000000622 irritating effect Effects 0.000 abstract 1
- KBOPZPXVLCULAV-UHFFFAOYSA-N mesalamine Chemical compound NC1=CC=C(O)C(C(O)=O)=C1 KBOPZPXVLCULAV-UHFFFAOYSA-N 0.000 abstract 1
- 229960004963 mesalazine Drugs 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 229920001897 terpolymer Polymers 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/60—Salicylic acid; Derivatives thereof
- A61K31/606—Salicylic acid; Derivatives thereof having amino groups
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
- A61K9/2846—Poly(meth)acrylates
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT1998MI002467A IT1303753B1 (it) | 1998-11-13 | 1998-11-13 | Composizioni farmaceutiche somministrabili per via orale contenentiun rivestimento gastroresistente a base di polimeri acrilici. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE315382T1 true ATE315382T1 (de) | 2006-02-15 |
Family
ID=11381056
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT99122470T ATE315382T1 (de) | 1998-11-13 | 1999-11-11 | Pharmazeutische zusammensetzungen zur oralen verabreichung, die einen magensaftresistenten überzug auf der basis von acrylatpolymeren enthalten |
Country Status (4)
| Country | Link |
|---|---|
| EP (1) | EP1004297B1 (de) |
| AT (1) | ATE315382T1 (de) |
| DE (1) | DE69929387D1 (de) |
| IT (1) | IT1303753B1 (de) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10013030A1 (de) * | 2000-03-17 | 2001-09-20 | Roehm Gmbh | Verwendung eines Copolymers zur Herstellung einer Arzneiform zur Therapie von Colitis ulcerosa und verwendungsgemäße Arzneiform |
| RU2286156C2 (ru) * | 2001-10-15 | 2006-10-27 | Ферринг Бв | Способ приготовления фармацевтической композиции, включающей в себя 5-аминосалициловую кислоту, для применения в лечении неспецифического язвенного колита и болезни крона |
| ES2288999T3 (es) * | 2001-10-15 | 2008-02-01 | Ferring Bv | Metodo para la preparacion de una composicion farmaceutica que comprende acido 5-aminosalicilico para su uso en el tratamiento de la colitis ulcerosa y la enfermedad de crohn. |
| US8282955B2 (en) | 2001-10-15 | 2012-10-09 | Ferring B.V. | Method for the preparation of a pharmaceutical composition comprising 5-aminosalicylic acid for use in treatment of ulcerative colitis and Crohn's disease |
| BG65471B1 (bg) * | 2002-04-02 | 2008-09-30 | "Софарма" Ад | Лекарствена форма на мезалазин и метод за нейнотополучаване |
| CA2520197A1 (en) * | 2003-04-23 | 2004-11-04 | Ferring B.V. | Sachet for a pharmaceutical composition |
| ITMI20032087A1 (it) | 2003-10-27 | 2005-04-28 | Pharmafilm S R L | Film autosupportanti per uso farmaceutico ed alimentare. |
| ITUB20160203A1 (it) * | 2016-01-19 | 2017-07-19 | Valpharma Int Spa | Formulazioni in compresse a rilascio modificato contenenti Mesalazina ad alto dosaggio, processo per la loro preparazione e loro uso. |
| ITUA20162293A1 (it) * | 2016-04-05 | 2017-10-05 | Sofar Spa | Processo per formulazioni solide di mesalazina |
| IT201800005908A1 (it) * | 2018-05-31 | 2019-12-01 | Compressa gastroresistente rivestita con film per il rilascio protratto di acido butirrico |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZA825384B (en) * | 1981-07-31 | 1983-05-25 | Tillott J B Ltd | Orally administrable pharmaceutical compositions |
| DE9414066U1 (de) * | 1994-08-31 | 1994-11-03 | Röhm GmbH & Co. KG, 64293 Darmstadt | Überzugs- und Bindemittel für Arzneiformen sowie damit hergestellte Arzneiform |
-
1998
- 1998-11-13 IT IT1998MI002467A patent/IT1303753B1/it active
-
1999
- 1999-11-11 EP EP99122470A patent/EP1004297B1/de not_active Expired - Lifetime
- 1999-11-11 AT AT99122470T patent/ATE315382T1/de not_active IP Right Cessation
- 1999-11-11 DE DE69929387T patent/DE69929387D1/de not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| IT1303753B1 (it) | 2001-02-23 |
| DE69929387D1 (de) | 2006-04-06 |
| EP1004297B1 (de) | 2006-01-11 |
| EP1004297A1 (de) | 2000-05-31 |
| ITMI982467A1 (it) | 2000-05-13 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |