ATE328609T1 - Zusammensetzungen zur behandlung von parkinson's krankheit, welche antagonisten der cb1-rezeptoren und aktivierungssubstanzen der dopamin- neurotransmission im gehirn enthalten - Google Patents

Zusammensetzungen zur behandlung von parkinson's krankheit, welche antagonisten der cb1-rezeptoren und aktivierungssubstanzen der dopamin- neurotransmission im gehirn enthalten

Info

Publication number
ATE328609T1
ATE328609T1 AT02772514T AT02772514T ATE328609T1 AT E328609 T1 ATE328609 T1 AT E328609T1 AT 02772514 T AT02772514 T AT 02772514T AT 02772514 T AT02772514 T AT 02772514T AT E328609 T1 ATE328609 T1 AT E328609T1
Authority
AT
Austria
Prior art keywords
parkinson
receptors
brain
disease
compositions
Prior art date
Application number
AT02772514T
Other languages
English (en)
Inventor
Jesus Benavides
Daniel Boccio
Yvette Henin
Odile Piot-Grosjean
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Application granted granted Critical
Publication of ATE328609T1 publication Critical patent/ATE328609T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
AT02772514T 2001-08-29 2002-08-28 Zusammensetzungen zur behandlung von parkinson's krankheit, welche antagonisten der cb1-rezeptoren und aktivierungssubstanzen der dopamin- neurotransmission im gehirn enthalten ATE328609T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0111200A FR2829028B1 (fr) 2001-08-29 2001-08-29 Association d'un antagoniste du recepteur cb1 et d'un produit qui active la neurotransmission dopaminergique dans le cerveau, les compositions pharmaceutiques les contenant et leur utilisation pour le traitement de la maladie de

Publications (1)

Publication Number Publication Date
ATE328609T1 true ATE328609T1 (de) 2006-06-15

Family

ID=8866792

Family Applications (1)

Application Number Title Priority Date Filing Date
AT02772514T ATE328609T1 (de) 2001-08-29 2002-08-28 Zusammensetzungen zur behandlung von parkinson's krankheit, welche antagonisten der cb1-rezeptoren und aktivierungssubstanzen der dopamin- neurotransmission im gehirn enthalten

Country Status (16)

Country Link
US (2) US7217705B2 (de)
EP (2) EP1423145B1 (de)
JP (2) JP2005505551A (de)
AR (1) AR036302A1 (de)
AT (1) ATE328609T1 (de)
AU (2) AU2002337277B2 (de)
CA (1) CA2458348A1 (de)
CY (1) CY1105341T1 (de)
DE (1) DE60212148T2 (de)
DK (1) DK1423145T3 (de)
ES (1) ES2263816T3 (de)
FR (1) FR2829028B1 (de)
IL (2) IL160557A0 (de)
MX (1) MXPA04001645A (de)
PT (1) PT1423145E (de)
WO (1) WO2003020314A1 (de)

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DE10359528A1 (de) 2003-12-18 2005-07-28 Schwarz Pharma Ag (S)-2-N-Propylamino-5-hydroxytetralin als D3-agonistisches Therapeutikum
EP1547592A1 (de) * 2003-12-23 2005-06-29 Schwarz Pharma Ag Intranasale formulierung enthaltend
DE10361258A1 (de) * 2003-12-24 2005-07-28 Schwarz Pharma Ag Verwendung von substituierten 2-Aminotetralinen zur vorbeugenden Behandlung von Morbus Parkinson
JP2007522255A (ja) * 2004-02-17 2007-08-09 ラボラトリオス・デル・ドクトル・エステベ・ソシエダッド・アノニマ 置換アゼチジン化合物、その製造および医薬品としての使用
ES2244314B1 (es) * 2004-02-17 2007-02-01 Laboratorios Del Dr. Esteve, S.A. Compuestos azetidinicos sustituidos, su preparacion y su aplicacion como medicamentos.
US20050197385A1 (en) * 2004-02-20 2005-09-08 Schwarz Pharma Ag Use of rotigotine for treatment or prevention of dopaminergic neuron loss
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Also Published As

Publication number Publication date
AU2002337277B2 (en) 2008-06-05
US20040209861A1 (en) 2004-10-21
IL160557A0 (en) 2004-07-25
EP1649849A3 (de) 2006-11-02
ES2263816T3 (es) 2006-12-16
CY1105341T1 (el) 2010-03-03
IL193325A0 (en) 2009-02-11
US7217705B2 (en) 2007-05-15
PT1423145E (pt) 2006-09-29
EP1423145A1 (de) 2004-06-02
DE60212148D1 (de) 2006-07-20
WO2003020314A1 (fr) 2003-03-13
EP1649849A2 (de) 2006-04-26
FR2829028A1 (fr) 2003-03-07
EP1423145B1 (de) 2006-06-07
CA2458348A1 (en) 2003-03-13
JP2005505551A (ja) 2005-02-24
US20070197654A1 (en) 2007-08-23
FR2829028B1 (fr) 2004-12-17
JP2010053153A (ja) 2010-03-11
MXPA04001645A (es) 2004-05-31
DK1423145T3 (da) 2006-10-02
AU2008212039A1 (en) 2008-10-09
AR036302A1 (es) 2004-08-25
DE60212148T2 (de) 2007-04-19

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