ATE330960T1 - Beta-lactamase hemmende verbindungen - Google Patents

Beta-lactamase hemmende verbindungen

Info

Publication number
ATE330960T1
ATE330960T1 AT03015238T AT03015238T ATE330960T1 AT E330960 T1 ATE330960 T1 AT E330960T1 AT 03015238 T AT03015238 T AT 03015238T AT 03015238 T AT03015238 T AT 03015238T AT E330960 T1 ATE330960 T1 AT E330960T1
Authority
AT
Austria
Prior art keywords
beta
formula
compounds
inhibiting compounds
lactamase inhibiting
Prior art date
Application number
AT03015238T
Other languages
English (en)
Inventor
John D Buynak
Sirishkumar D Nidamarthy
Greg C Adam
Srinivasa A Rao
Original Assignee
Res Corp Technologies Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Res Corp Technologies Inc filed Critical Res Corp Technologies Inc
Application granted granted Critical
Publication of ATE330960T1 publication Critical patent/ATE330960T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Cephalosporin Compounds (AREA)
AT03015238T 1999-04-15 2000-04-14 Beta-lactamase hemmende verbindungen ATE330960T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US12948299P 1999-04-15 1999-04-15

Publications (1)

Publication Number Publication Date
ATE330960T1 true ATE330960T1 (de) 2006-07-15

Family

ID=22440183

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03015238T ATE330960T1 (de) 1999-04-15 2000-04-14 Beta-lactamase hemmende verbindungen

Country Status (8)

Country Link
EP (1) EP1169323A1 (de)
JP (1) JP2002542249A (de)
AT (1) ATE330960T1 (de)
AU (1) AU773013B2 (de)
CA (1) CA2371389A1 (de)
DE (1) DE60029023T2 (de)
MX (1) MXPA01010409A (de)
WO (1) WO2000063213A1 (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2282461C (en) 1997-12-29 2004-04-20 John D. Buynak 2-.beta.-substituted-6-alkylidene penicillanic acid derivatives as .beta.-lactamase inhibitors
US6407091B1 (en) 1999-04-15 2002-06-18 Research Corporation Technologies, Inc. β-lactamase inhibiting compounds
JP2002356427A (ja) * 2001-05-30 2002-12-13 Shionogi & Co Ltd β−ラクタマーゼ阻害剤
CA2454413A1 (en) 2001-07-24 2003-03-13 Alamx, L.L.C. 7-alkylidene-3-substituted-3-cephem-4-carboxylates as beta-lactamase inhibitors
US7022691B2 (en) 2002-04-04 2006-04-04 John D. Buynak Inhibitors of serine and metallo-β-lactamases
CN102731530B (zh) * 2011-04-07 2016-05-04 天津市医药集团技术发展有限公司 头孢菌素化合物及其合成方法与应用
CN107021893A (zh) * 2017-05-05 2017-08-08 贵州师范学院 一类硫代酰铵盐离子液体及其制备方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5629306A (en) * 1994-12-09 1997-05-13 Research Corporation Technologies, Inc. 7-alkylidene cephalosporanic acid derivatives and methods of using the same
US5760027A (en) * 1996-12-06 1998-06-02 Research Corporation Technologies, Inc. Use of 7-alkylidene cephalosporins to inhibit elastase activity

Also Published As

Publication number Publication date
AU773013B2 (en) 2004-05-13
JP2002542249A (ja) 2002-12-10
DE60029023T2 (de) 2007-01-18
AU4238600A (en) 2000-11-02
WO2000063213A1 (en) 2000-10-26
EP1169323A1 (de) 2002-01-09
DE60029023D1 (de) 2006-08-03
MXPA01010409A (es) 2003-12-11
CA2371389A1 (en) 2000-10-26

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Legal Events

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RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties