ATE344272T1 - Uridinderivate als antibiotika - Google Patents

Uridinderivate als antibiotika

Info

Publication number
ATE344272T1
ATE344272T1 AT01931788T AT01931788T ATE344272T1 AT E344272 T1 ATE344272 T1 AT E344272T1 AT 01931788 T AT01931788 T AT 01931788T AT 01931788 T AT01931788 T AT 01931788T AT E344272 T1 ATE344272 T1 AT E344272T1
Authority
AT
Austria
Prior art keywords
antibiotics
uridine derivatives
uridine
derivatives
formulawhere
Prior art date
Application number
AT01931788T
Other languages
English (en)
Inventor
Jozsef Aszodi
Stanislas Didierlaurent
Christophe Dini
Nathalie Drochon
Jean-Claude Guillot
Jidong Zhang
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Application granted granted Critical
Publication of ATE344272T1 publication Critical patent/ATE344272T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/18Acyclic radicals, substituted by carbocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • A61P31/06Antibacterial agents for tuberculosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06Pyrimidine radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
AT01931788T 2000-05-09 2001-05-04 Uridinderivate als antibiotika ATE344272T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0005858A FR2808797A1 (fr) 2000-05-09 2000-05-09 Nouveaux derives de l'uridine, leur procede de preparation et leur application comme medicaments

Publications (1)

Publication Number Publication Date
ATE344272T1 true ATE344272T1 (de) 2006-11-15

Family

ID=8849999

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01931788T ATE344272T1 (de) 2000-05-09 2001-05-04 Uridinderivate als antibiotika

Country Status (12)

Country Link
US (1) US6875752B2 (de)
EP (1) EP1284984B1 (de)
JP (1) JP4994557B2 (de)
CN (1) CN1191264C (de)
AT (1) ATE344272T1 (de)
AU (1) AU2001258488A1 (de)
CA (1) CA2408453A1 (de)
DE (1) DE60124245T2 (de)
FR (1) FR2808797A1 (de)
IL (1) IL152614A0 (de)
MX (1) MXPA02010961A (de)
WO (1) WO2001085750A1 (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006092808A1 (en) * 2005-03-04 2006-09-08 Dabur Pharma Limited Intermediate and process for preparing of beta- anomer enriched 21deoxy, 21 ,21-difluoro-d-ribofuranosyl nucleosides
MX2011009728A (es) * 2009-03-20 2011-10-14 Alios Biopharma Inc Analogos nucleotido y nucleosido sustituidos.
EA025341B1 (ru) 2010-09-22 2016-12-30 Алиос Биофарма, Инк. Замещенные аналоги нуклеотидов
US8980865B2 (en) 2011-12-22 2015-03-17 Alios Biopharma, Inc. Substituted nucleotide analogs
US8916538B2 (en) 2012-03-21 2014-12-23 Vertex Pharmaceuticals Incorporated Solid forms of a thiophosphoramidate nucleotide prodrug
HK1203356A1 (en) 2012-03-22 2015-10-30 艾丽奥斯生物制药有限公司 Pharmaceutical combinations comprising a thionucleotide analog
IL311727A (en) 2017-07-07 2024-05-01 Epicentrx Inc Preparations for intravenous administration of medical substances
CA3087998A1 (en) 2018-01-12 2019-07-18 California Institute Of Technology Glycosyltransferase inhibitors

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH02306992A (ja) * 1989-05-20 1990-12-20 Rikagaku Kenkyusho 抗生物質rk―1061g及びrk―1061h並びにその製造法
GB9004407D0 (en) * 1990-02-27 1990-04-25 Fujisawa Pharmaceutical Co New uronic acid derivatives,a process for their production and a pharmaceutical composition containing the same
CA2252483A1 (en) * 1996-04-26 1997-11-06 Snow Brand Milk Products Co., Ltd. Novel antibiotic rk-1061s and a method of production thereof

Also Published As

Publication number Publication date
CN1427846A (zh) 2003-07-02
MXPA02010961A (es) 2003-03-27
IL152614A0 (en) 2003-06-24
DE60124245D1 (de) 2006-12-14
US20030130227A1 (en) 2003-07-10
EP1284984B1 (de) 2006-11-02
CN1191264C (zh) 2005-03-02
FR2808797A1 (fr) 2001-11-16
JP4994557B2 (ja) 2012-08-08
CA2408453A1 (fr) 2001-11-15
DE60124245T2 (de) 2007-05-31
JP2003532736A (ja) 2003-11-05
AU2001258488A1 (en) 2001-11-20
US6875752B2 (en) 2005-04-05
EP1284984A1 (de) 2003-02-26
WO2001085750A1 (fr) 2001-11-15

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Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties