ATE344272T1 - Uridinderivate als antibiotika - Google Patents

Uridinderivate als antibiotika

Info

Publication number
ATE344272T1
ATE344272T1 AT01931788T AT01931788T ATE344272T1 AT E344272 T1 ATE344272 T1 AT E344272T1 AT 01931788 T AT01931788 T AT 01931788T AT 01931788 T AT01931788 T AT 01931788T AT E344272 T1 ATE344272 T1 AT E344272T1
Authority
AT
Austria
Prior art keywords
antibiotics
uridine derivatives
uridine
derivatives
formulawhere
Prior art date
Application number
AT01931788T
Other languages
English (en)
Inventor
Jozsef Aszodi
Stanislas Didierlaurent
Christophe Dini
Nathalie Drochon
Jean-Claude Guillot
Jidong Zhang
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Application granted granted Critical
Publication of ATE344272T1 publication Critical patent/ATE344272T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/18—Acyclic radicals, substituted by carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/06—Antibacterial agents for tuberculosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06—Pyrimidine radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
AT01931788T 2000-05-09 2001-05-04 Uridinderivate als antibiotika ATE344272T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0005858A FR2808797A1 (fr) 2000-05-09 2000-05-09 Nouveaux derives de l'uridine, leur procede de preparation et leur application comme medicaments

Publications (1)

Publication Number Publication Date
ATE344272T1 true ATE344272T1 (de) 2006-11-15

Family

ID=8849999

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01931788T ATE344272T1 (de) 2000-05-09 2001-05-04 Uridinderivate als antibiotika

Country Status (12)

Country Link
US (1) US6875752B2 (de)
EP (1) EP1284984B1 (de)
JP (1) JP4994557B2 (de)
CN (1) CN1191264C (de)
AT (1) ATE344272T1 (de)
AU (1) AU2001258488A1 (de)
CA (1) CA2408453A1 (de)
DE (1) DE60124245T2 (de)
FR (1) FR2808797A1 (de)
IL (1) IL152614A0 (de)
MX (1) MXPA02010961A (de)
WO (1) WO2001085750A1 (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE602005019626D1 (de) * 2005-03-04 2010-04-08 Fresenius Kabi Oncology Ltd Zwischenprodukt und verfahren zur herstellung von an beta-anomeren angereicherten 2'-desoxy,2',2'-difluor-d-ribufuranosylnukleosiden
WO2010108140A1 (en) * 2009-03-20 2010-09-23 Alios Biopharma, Inc. Substituted nucleoside and nucleotide analogs
WO2012040127A1 (en) 2010-09-22 2012-03-29 Alios Biopharma, Inc. Substituted nucleotide analogs
EP2794630A4 (de) 2011-12-22 2015-04-01 Alios Biopharma Inc Substituierte phosphorthioat-nukleotidanaloga
NZ631601A (en) 2012-03-21 2016-06-24 Alios Biopharma Inc Solid forms of a thiophosphoramidate nucleotide prodrug
NZ630805A (en) 2012-03-22 2016-01-29 Alios Biopharma Inc Pharmaceutical combinations comprising a thionucleotide analog
MX2020000265A (es) 2017-07-07 2020-07-22 Epicentrx Inc Composiciones para la administración parenteral de agentes terapéuticos.
CA3087998A1 (en) * 2018-01-12 2019-07-18 California Institute Of Technology Glycosyltransferase inhibitors

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH02306992A (ja) * 1989-05-20 1990-12-20 Rikagaku Kenkyusho 抗生物質rk―1061g及びrk―1061h並びにその製造法
GB9004407D0 (en) * 1990-02-27 1990-04-25 Fujisawa Pharmaceutical Co New uronic acid derivatives,a process for their production and a pharmaceutical composition containing the same
US6455694B1 (en) * 1996-04-26 2002-09-24 Daiichi Pharmaceutical Co., Ltd. Antibiotics RK-1061 and process for preparing the same

Also Published As

Publication number Publication date
EP1284984B1 (de) 2006-11-02
FR2808797A1 (fr) 2001-11-16
IL152614A0 (en) 2003-06-24
CN1191264C (zh) 2005-03-02
CA2408453A1 (fr) 2001-11-15
CN1427846A (zh) 2003-07-02
DE60124245T2 (de) 2007-05-31
US20030130227A1 (en) 2003-07-10
US6875752B2 (en) 2005-04-05
MXPA02010961A (es) 2003-03-27
JP2003532736A (ja) 2003-11-05
JP4994557B2 (ja) 2012-08-08
WO2001085750A1 (fr) 2001-11-15
AU2001258488A1 (en) 2001-11-20
EP1284984A1 (de) 2003-02-26
DE60124245D1 (de) 2006-12-14

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Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties