ATE349203T1 - Delavirdin tablettenformulierung - Google Patents
Delavirdin tablettenformulierungInfo
- Publication number
- ATE349203T1 ATE349203T1 AT99925951T AT99925951T ATE349203T1 AT E349203 T1 ATE349203 T1 AT E349203T1 AT 99925951 T AT99925951 T AT 99925951T AT 99925951 T AT99925951 T AT 99925951T AT E349203 T1 ATE349203 T1 AT E349203T1
- Authority
- AT
- Austria
- Prior art keywords
- delavirdine
- tablet formulation
- amount
- superdisintegrant
- binder
- Prior art date
Links
- 239000007916 tablet composition Substances 0.000 title abstract 2
- WHBIGIKBNXZKFE-UHFFFAOYSA-N delavirdine Chemical compound CC(C)NC1=CC=CN=C1N1CCN(C(=O)C=2NC3=CC=C(NS(C)(=O)=O)C=C3C=2)CC1 WHBIGIKBNXZKFE-UHFFFAOYSA-N 0.000 title 2
- 229960005319 delavirdine Drugs 0.000 title 1
- 239000011230 binding agent Substances 0.000 abstract 2
- 239000003814 drug Substances 0.000 abstract 2
- 229940079593 drug Drugs 0.000 abstract 2
- 230000001376 precipitating effect Effects 0.000 abstract 2
- 238000010438 heat treatment Methods 0.000 abstract 1
- 239000002904 solvent Substances 0.000 abstract 1
- 238000013268 sustained release Methods 0.000 abstract 1
- 239000012730 sustained-release form Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Cephalosporin Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US8896098P | 1998-06-11 | 1998-06-11 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE349203T1 true ATE349203T1 (de) | 2007-01-15 |
Family
ID=22214517
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT99925951T ATE349203T1 (de) | 1998-06-11 | 1999-06-07 | Delavirdin tablettenformulierung |
Country Status (20)
| Country | Link |
|---|---|
| US (3) | US6177101B1 (de) |
| EP (1) | EP1083885B1 (de) |
| JP (1) | JP4827296B2 (de) |
| KR (2) | KR20070040426A (de) |
| CN (1) | CN1237958C (de) |
| AT (1) | ATE349203T1 (de) |
| AU (1) | AU753241C (de) |
| BR (1) | BR9910481A (de) |
| CA (1) | CA2328703C (de) |
| CY (1) | CY1105924T1 (de) |
| DE (1) | DE69934582T2 (de) |
| DK (1) | DK1083885T3 (de) |
| EA (1) | EA004311B1 (de) |
| ES (1) | ES2277682T3 (de) |
| HU (1) | HUP0102206A3 (de) |
| NZ (1) | NZ508762A (de) |
| PL (1) | PL200163B1 (de) |
| PT (1) | PT1083885E (de) |
| WO (1) | WO1999063970A1 (de) |
| ZA (1) | ZA200006090B (de) |
Families Citing this family (31)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2277682T3 (es) * | 1998-06-11 | 2007-07-16 | PHARMACIA & UPJOHN COMPANY LLC | Formulacion de delavirdina en comprimido. |
| EA006402B1 (ru) | 1999-12-23 | 2005-12-29 | Пфайзер Продактс Инк. | Комбинация лекарства и целлюлозного полимера, повышающего концентрацию; способ введения лекарства и водный раствор (варианты) |
| US7115279B2 (en) * | 2000-08-03 | 2006-10-03 | Curatolo William J | Pharmaceutical compositions of cholesteryl ester transfer protein inhibitors |
| US20040243118A1 (en) * | 2001-06-01 | 2004-12-02 | Ayers Gregory M. | Device and method for positioning a catheter tip for creating a cryogenic lesion |
| BR0212214A (pt) * | 2001-08-28 | 2004-10-19 | Pharmacia Corp | Base livre de clindamicina cristalina |
| DE10164510A1 (de) | 2001-12-20 | 2003-07-10 | Schering Ag | Orale Fludara reinst Formulierung mit schneller Freisetzung des Wirkstoffes |
| JP2004107258A (ja) * | 2002-09-18 | 2004-04-08 | Ss Pharmaceut Co Ltd | 催眠用圧縮成型製剤 |
| US20050163839A1 (en) * | 2003-01-29 | 2005-07-28 | Sun Pharmaceutical Industries Limited | Oral controlled release pharmaceutical composition containing metaxalone as active agent |
| JP2006522099A (ja) * | 2003-04-04 | 2006-09-28 | ファルマシア コーポレーション | 複合粒状体からなる経口徐放性圧縮錠 |
| US9241997B2 (en) | 2003-06-13 | 2016-01-26 | Idh Holding Aps | Treatment of symptoms associated with bacterial vaginosis |
| MXPA06000178A (es) * | 2003-07-01 | 2006-04-11 | Pharmacia & Upjohn Co Llc | Solidos modulados en la fase de difusion. |
| US7201920B2 (en) | 2003-11-26 | 2007-04-10 | Acura Pharmaceuticals, Inc. | Methods and compositions for deterring abuse of opioid containing dosage forms |
| US20050283146A1 (en) * | 2004-06-17 | 2005-12-22 | Lentz David J | Thermally extended spiral cryotip for a cryoablation catheter |
| US20060099253A1 (en) * | 2004-10-20 | 2006-05-11 | Wyeth | Antibiotic product formulation |
| US20070059359A1 (en) * | 2005-06-07 | 2007-03-15 | Thomas Backensfeld | Immediate-release and high-drug-load pharmaceutical formulations of non-micronised (4-chlorophenyl)[4-(4-pyridylmethyl)phthalazin-1-yl] and salts thereof |
| EP2048394B1 (de) | 2006-07-27 | 2014-05-07 | Kabushiki Kaisha Kobe Seiko Sho | Kneteinrichtung mit knetvorrichtung und antriebsvorrichtung, die durch die verbindungsvorrichtung miteinander verbunden sind |
| CA2617688C (en) * | 2007-02-22 | 2015-08-18 | Alpex Pharma S.A. | Solid dosage formulations containing weight-loss drugs |
| US8696606B2 (en) * | 2009-09-28 | 2014-04-15 | Continuous MotionFlow, LLC | Passive motion machine with integrated mechanical DVT prophylactic therapy |
| EP2488029B1 (de) | 2009-09-30 | 2016-03-23 | Acura Pharmaceuticals, Inc. | Verfahren und zusammensetzungen zur abschreckung vor missbrauch |
| JP5226732B2 (ja) * | 2010-05-20 | 2013-07-03 | エスエス製薬株式会社 | 催眠用圧縮成型製剤 |
| US20120010216A1 (en) * | 2010-07-06 | 2012-01-12 | Brown Arthur M | Pharmaceutical compositions containing vanoxerine |
| US10201584B1 (en) | 2011-05-17 | 2019-02-12 | Abbvie Inc. | Compositions and methods for treating HCV |
| EA032913B1 (ru) | 2012-10-18 | 2019-08-30 | Эббви Инк. | Препараты производных пиримидиндиона |
| RU2673818C2 (ru) | 2012-11-30 | 2018-11-30 | Экьюра Фармасьютикалз, Инк. | Саморегулируемое высвобождение фармацевтического ингредиента |
| SG11201509998WA (en) | 2013-06-13 | 2016-01-28 | Akebia Therapeutics Inc | Compositions and methods for treating anemia |
| WO2015103490A1 (en) | 2014-01-03 | 2015-07-09 | Abbvie, Inc. | Solid antiviral dosage forms |
| US11103581B2 (en) | 2015-08-31 | 2021-08-31 | Acura Pharmaceuticals, Inc. | Methods and compositions for self-regulated release of active pharmaceutical ingredient |
| CA2937365C (en) | 2016-03-29 | 2018-09-18 | F. Hoffmann-La Roche Ag | Granulate formulation of 5-methyl-1-phenyl-2-(1h)-pyridone and method of making the same |
| WO2019218958A1 (zh) * | 2018-05-15 | 2019-11-21 | 江苏豪森药业集团有限公司 | 包含小分子egfr抑制剂的药物组合物及其制备方法 |
| CN108619104A (zh) * | 2018-06-29 | 2018-10-09 | 哈尔滨珍宝制药有限公司 | 一种基于盐酸克林霉素的药物组合物及其制备方法 |
| CZ309820B6 (cs) * | 2021-04-23 | 2023-11-08 | Pro.Med.Cs Praha A.S. | Způsob přípravy pevné lékové formy obsahující kompozici s nízkým obsahem účinné látky |
Family Cites Families (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4013785A (en) * | 1975-03-21 | 1977-03-22 | Bristol-Myers Company | Apap tablet containing fumed silica and process for manufacturing same |
| ZA855250B (en) * | 1984-08-17 | 1986-02-26 | Upjohn Co | Stable,high dose,high bulk density ibuprofen granulations for tablet and capsule manufacturing |
| GB8521350D0 (en) * | 1985-08-28 | 1985-10-02 | Euro Celtique Sa | Analgesic composition |
| DE3708916A1 (de) | 1987-03-19 | 1988-09-29 | Boehringer Ingelheim Kg | Verfahren zur reinigung resorbierbarer polyester |
| US5211958A (en) * | 1987-11-30 | 1993-05-18 | Gist-Brocades, N.V. | Pharmaceutical composition and process for its preparation |
| ATE72118T1 (de) * | 1987-11-30 | 1992-02-15 | Gist Brocades Nv | Pharmazeutische zusammensetzung und verfahren zu ihrer herstellung. |
| GB8824392D0 (en) * | 1988-10-18 | 1988-11-23 | Ciba Geigy Ag | Dispersible formulation |
| US5256699A (en) * | 1988-10-18 | 1993-10-26 | Ciba-Geify Corporation | Dispersible tablet formulation of diclofenac acid free base |
| CA2007764C (en) | 1989-02-24 | 1999-11-30 | Joseph Michael Beaurline | Salsalate tablet |
| GB8909793D0 (en) * | 1989-04-28 | 1989-06-14 | Beecham Group Plc | Pharmaceutical formulation |
| NZ236393A (en) | 1989-12-13 | 1992-05-26 | Lilly Co Eli | N-alkylated glycopeptide derivatives prepared from antibiotics a82846 series and pa-42867-a; pharmaceutical compositions |
| US5563142A (en) * | 1989-12-28 | 1996-10-08 | The Upjohn Company | Diaromatic substituted compounds as anti-HIV-1 agents |
| US5519021A (en) * | 1992-08-07 | 1996-05-21 | Merck & Co., Inc. | Benzoxazinones as inhibitors of HIV reverse transcriptase |
| US5358941A (en) | 1992-12-02 | 1994-10-25 | Merck & Co., Inc. | Dry mix formulation for bisphosphonic acids with lactose |
| FR2711524B1 (fr) * | 1993-10-21 | 1995-11-24 | Rhone Dpc Europ | Procédé de préparation de compositions orales contenant des quinolones. |
| KR100364941B1 (ko) | 1994-04-15 | 2003-02-19 | 파마시아 앤드 업존 캄파니 | 1-[5-메탄설폰아미도인돌릴-2-카보닐]-4-[3-(1-메틸에틸아미노)-2-피리디닐]피페라진의신규한결정형태 |
| US5585115A (en) * | 1995-01-09 | 1996-12-17 | Edward H. Mendell Co., Inc. | Pharmaceutical excipient having improved compressability |
| US5837292A (en) | 1996-07-03 | 1998-11-17 | Yamanouchi Europe B.V. | Granulate for the preparation of fast-disintegrating and fast-dissolving compositions containing a high amount of drug |
| US6013280A (en) * | 1997-10-07 | 2000-01-11 | Fuisz Technologies Ltd. | Immediate release dosage forms containing microspheres |
| US5955107A (en) * | 1997-12-12 | 1999-09-21 | Fmc Corporation | Pharmaceutical suspension tablet compositions |
| UA72207C2 (uk) * | 1998-04-07 | 2005-02-15 | Брістол- Майєрс Сквібб Фарма Компані | Фармацевтична композиція ефавіренцу з добавкою дезінтегруючих агентів у вигляді швидкорозчинних капсул або таблеток та спосіб її виготовлення |
| ES2277682T3 (es) * | 1998-06-11 | 2007-07-16 | PHARMACIA & UPJOHN COMPANY LLC | Formulacion de delavirdina en comprimido. |
-
1999
- 1999-06-07 ES ES99925951T patent/ES2277682T3/es not_active Expired - Lifetime
- 1999-06-07 JP JP2000553039A patent/JP4827296B2/ja not_active Expired - Lifetime
- 1999-06-07 NZ NZ508762A patent/NZ508762A/en not_active IP Right Cessation
- 1999-06-07 KR KR1020077007572A patent/KR20070040426A/ko not_active Ceased
- 1999-06-07 EA EA200100024A patent/EA004311B1/ru not_active IP Right Cessation
- 1999-06-07 HU HU0102206A patent/HUP0102206A3/hu unknown
- 1999-06-07 KR KR1020007013985A patent/KR100724016B1/ko not_active Expired - Lifetime
- 1999-06-07 EP EP99925951A patent/EP1083885B1/de not_active Revoked
- 1999-06-07 DE DE69934582T patent/DE69934582T2/de not_active Revoked
- 1999-06-07 WO PCT/US1999/011798 patent/WO1999063970A1/en not_active Ceased
- 1999-06-07 BR BR9910481-4A patent/BR9910481A/pt not_active Application Discontinuation
- 1999-06-07 CN CNB998062316A patent/CN1237958C/zh not_active Expired - Lifetime
- 1999-06-07 AT AT99925951T patent/ATE349203T1/de active
- 1999-06-07 PT PT99925951T patent/PT1083885E/pt unknown
- 1999-06-07 CA CA002328703A patent/CA2328703C/en not_active Expired - Lifetime
- 1999-06-07 DK DK99925951T patent/DK1083885T3/da active
- 1999-06-07 PL PL344328A patent/PL200163B1/pl unknown
- 1999-06-07 US US09/327,135 patent/US6177101B1/en not_active Expired - Lifetime
- 1999-06-07 AU AU42134/99A patent/AU753241C/en not_active Expired
-
2000
- 2000-09-06 US US09/656,364 patent/US7108864B1/en not_active Expired - Lifetime
- 2000-10-27 ZA ZA200006090A patent/ZA200006090B/xx unknown
-
2006
- 2006-07-14 US US11/487,554 patent/US20060257476A1/en not_active Abandoned
-
2007
- 2007-01-15 CY CY20071100050T patent/CY1105924T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AU4213499A (en) | 1999-12-30 |
| ES2277682T3 (es) | 2007-07-16 |
| DK1083885T3 (da) | 2007-02-26 |
| PL200163B1 (pl) | 2008-12-31 |
| CA2328703A1 (en) | 1999-12-16 |
| CA2328703C (en) | 2007-10-30 |
| DE69934582T2 (de) | 2007-10-04 |
| HUP0102206A3 (en) | 2002-12-28 |
| WO1999063970A1 (en) | 1999-12-16 |
| BR9910481A (pt) | 2001-01-09 |
| EA004311B1 (ru) | 2004-02-26 |
| KR100724016B1 (ko) | 2007-05-31 |
| AU753241C (en) | 2003-05-08 |
| HK1036417A1 (en) | 2002-01-04 |
| US6177101B1 (en) | 2001-01-23 |
| EA200100024A1 (ru) | 2001-06-25 |
| JP2002517430A (ja) | 2002-06-18 |
| EP1083885A1 (de) | 2001-03-21 |
| DE69934582D1 (de) | 2007-02-08 |
| AU753241B2 (en) | 2002-10-10 |
| ZA200006090B (en) | 2001-10-29 |
| PL344328A1 (en) | 2001-10-22 |
| HUP0102206A2 (hu) | 2002-03-28 |
| EP1083885B1 (de) | 2006-12-27 |
| KR20070040426A (ko) | 2007-04-16 |
| CN1301149A (zh) | 2001-06-27 |
| US7108864B1 (en) | 2006-09-19 |
| US20060257476A1 (en) | 2006-11-16 |
| CN1237958C (zh) | 2006-01-25 |
| PT1083885E (pt) | 2007-01-31 |
| NZ508762A (en) | 2003-07-25 |
| JP4827296B2 (ja) | 2011-11-30 |
| CY1105924T1 (el) | 2011-04-06 |
| KR20010052717A (ko) | 2001-06-25 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DK1083885T3 (da) | Delavirdintabletformulering | |
| GEP20053420B (en) | Sustained Release Ranolanolazine Formulation | |
| AU3080895A (en) | Novel piperazides derived from arylpiperazine, processes for their preparation, their use as medicaments and pharmaceutical compositions comprising them | |
| KR930016091A (ko) | 거의 수불용성인 약제의 고체 분산액을 제조하는 방법 | |
| HUP0100072A3 (en) | Phenoxazine, phenthiazine derivatives, their use in medicine; process for their preparation and pharmaceutical compositions containing them | |
| IE881916L (en) | Press-coated dihydropyridine tablets | |
| GB2186485B (en) | Slow release formulation | |
| CA2346001A1 (en) | Controlled release nanoparticulate compositions | |
| NO934573L (no) | Farmasoeytiske formuleringer av oste-orgeniske proteiner | |
| HUT75881A (en) | Pharmaceutical composition for 24 hour release of metoprolol | |
| BR9808933A (pt) | Composição sob forma de microcápsulas ou de implantes, processo de preparação de uma substância hidrossolúvel, substância ativa, acetato de triptorelina, acetato de lanreotìdeo, ou acetato de octreotìdeo, e rna de filamento duplo | |
| ATE145132T1 (de) | Therapeutische zusammensetzung und verfahren für ihre herstellung | |
| FR2744449B1 (fr) | Nouvelles piperazines aromatiques derivees de cycloazanes substitues, ainsi que leur procede de preparation, les compositions pharmaceutiques et leur utilisation comme medicaments | |
| TR199901433T2 (xx) | Pirolo$3,4-D] pirimidinon t�revleri ve bunlar�n ila� olarak kullan�mlar�. | |
| AU6404398A (en) | New derivatives of 2-(iminomethyl)amino-phenyl, their preparation, their use as medicaments and the pharmaceutical compositions containing them | |
| GEP20033062B (en) | Pharmaceutical Composition Comprising Entacapone or Nitecapone and Cross-Linked Cellulose Derivative | |
| DE69632194D1 (de) | Galanthamin-derivate, verfahren zu ihrer herstellung, ihre verwendung als arzmittel und diese enthaltende pharmazeutische zusammensetzung | |
| HUP9904210A3 (en) | Analogues of camptothecin,their application as medicine and pharmaceutical compositions containing them | |
| TR200003303T2 (tr) | Astıma, alerjiye, iltihaplanmaya karşı, bağışıklık düzenleyici ve sinirsel koruyucu etkiye sahip yeni 1,5- ve 3-O-ikameli 1H-indazoller, bunların hazırlanması ve tıbbi maddeler olarak kullanımları. | |
| MY120550A (en) | Substituted 1,2,3,4,5,6-hexahydro-2,6-methano-3-benzazocin-10-ols, processes for preparing them and their use as pharmaceutical compositions. | |
| IL127518A (en) | Substituted heterocyclic benzocycloalkenes, their preparation and pharmaceutical compositions having an analgesic effect | |
| AU5139596A (en) | Pharmaceutical matrix pellets, tablets and composition for the preparation thereof | |
| MD970269A (en) | Clavulanates | |
| AU1606997A (en) | Novel naphthylpiperazines derived from substituted cycloazanes, method for preparing same, pharmaceutical compositions and use thereof as drugs | |
| TR199900013T2 (xx) | Yeni bile�ikler. |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification |
Ref document number: 1083885 Country of ref document: EP |