ATE349203T1 - Delavirdin tablettenformulierung - Google Patents

Delavirdin tablettenformulierung

Info

Publication number: ATE349203T1
Authority: AT; Austria
Prior art keywords: delavirdine; tablet formulation; amount; superdisintegrant; binder
Prior art date: 1998-06-11

Application number

AT99925951T

Other languages

English (en)

Inventor

Alice C Martino

Ashley H Bates

Walter Morozowich

E John Lee

Original Assignee

Pharmacia & Upjohn Co Llc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-06-11

Filing date

1999-06-07

Publication date

2007-01-15

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22214517&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE349203(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1999-06-07 Application filed by Pharmacia & Upjohn Co Llc filed Critical Pharmacia & Upjohn Co Llc

2007-01-15 Application granted granted Critical

2007-01-15 Publication of ATE349203T1 publication Critical patent/ATE349203T1/de

Links

239000007916 tablet composition Substances 0.000 title abstract 2
WHBIGIKBNXZKFE-UHFFFAOYSA-N delavirdine Chemical compound CC(C)NC1=CC=CN=C1N1CCN(C(=O)C=2NC3=CC=C(NS(C)(=O)=O)C=C3C=2)CC1 WHBIGIKBNXZKFE-UHFFFAOYSA-N 0.000 title 2
229960005319 delavirdine Drugs 0.000 title 1
239000011230 binding agent Substances 0.000 abstract 2
239000003814 drug Substances 0.000 abstract 2
229940079593 drug Drugs 0.000 abstract 2
230000001376 precipitating effect Effects 0.000 abstract 2
238000010438 heat treatment Methods 0.000 abstract 1
239000002904 solvent Substances 0.000 abstract 1
238000013268 sustained release Methods 0.000 abstract 1
239000012730 sustained-release form Substances 0.000 abstract 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin

Landscapes

Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical & Material Sciences (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Medicinal Preparation (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Cephalosporin Compounds (AREA)

AT99925951T 1998-06-11 1999-06-07 Delavirdin tablettenformulierung ATE349203T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US8896098P	1998-06-11	1998-06-11

Publications (1)

Publication Number	Publication Date
ATE349203T1 true ATE349203T1 (de)	2007-01-15

Family

ID=22214517

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT99925951T ATE349203T1 (de)	1998-06-11	1999-06-07	Delavirdin tablettenformulierung

Country Status (20)

Country	Link
US (3)	US6177101B1 (de)
EP (1)	EP1083885B1 (de)
JP (1)	JP4827296B2 (de)
KR (2)	KR100724016B1 (de)
CN (1)	CN1237958C (de)
AT (1)	ATE349203T1 (de)
AU (1)	AU753241C (de)
BR (1)	BR9910481A (de)
CA (1)	CA2328703C (de)
CY (1)	CY1105924T1 (de)
DE (1)	DE69934582T2 (de)
DK (1)	DK1083885T3 (de)
EA (1)	EA004311B1 (de)
ES (1)	ES2277682T3 (de)
HU (1)	HUP0102206A3 (de)
NZ (1)	NZ508762A (de)
PL (1)	PL200163B1 (de)
PT (1)	PT1083885E (de)
WO (1)	WO1999063970A1 (de)
ZA (1)	ZA200006090B (de)

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DE69934582T2 (de) *	1998-06-11	2007-10-04	Pharmacia & Upjohn Co. Llc, Kalamazoo	Delavirdin tablettenformulierung
CN1402629A (zh)	1999-12-23	2003-03-12	辉瑞产品公司	提供提高的药物浓度的药物组合物
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ES2752773T3 (es)	2003-06-13	2020-04-06	Idh Holding Aps	Tratamiento de los síntomas asociados a la vaginosis bacteriana
WO2005004763A1 (en) *	2003-07-01	2005-01-20	Pharmacia & Upjohn Company Llc.	Diffusion layer modulated solids
US7201920B2 (en)	2003-11-26	2007-04-10	Acura Pharmaceuticals, Inc.	Methods and compositions for deterring abuse of opioid containing dosage forms
US20050283146A1 (en) *	2004-06-17	2005-12-22	Lentz David J	Thermally extended spiral cryotip for a cryoablation catheter
US20060099253A1 (en) *	2004-10-20	2006-05-11	Wyeth	Antibiotic product formulation
US20070059359A1 (en) *	2005-06-07	2007-03-15	Thomas Backensfeld	Immediate-release and high-drug-load pharmaceutical formulations of non-micronised (4-chlorophenyl)[4-(4-pyridylmethyl)phthalazin-1-yl] and salts thereof
KR101190335B1 (ko)	2006-07-27	2012-10-11	가부시키가이샤 고베 세이코쇼	접속 장치 및 이 접속 장치를 통해 접속되는 혼련 장치와 구동 장치를 갖는 혼련 설비
CA2617688C (en) *	2007-02-22	2015-08-18	Alpex Pharma S.A.	Solid dosage formulations containing weight-loss drugs
US8696606B2 (en) *	2009-09-28	2014-04-15	Continuous MotionFlow, LLC	Passive motion machine with integrated mechanical DVT prophylactic therapy
AU2010300641B2 (en)	2009-09-30	2016-03-17	Acura Pharmaceuticals, Inc.	Methods and compositions for deterring abuse
JP5226732B2 (ja) *	2010-05-20	2013-07-03	エスエス製薬株式会社	催眠用圧縮成型製剤
US20120010216A1 (en) *	2010-07-06	2012-01-12	Brown Arthur M	Pharmaceutical compositions containing vanoxerine
US10201584B1 (en)	2011-05-17	2019-02-12	Abbvie Inc.	Compositions and methods for treating HCV
WO2014063101A1 (en)	2012-10-18	2014-04-24	Abbvie Inc.	Formulations of pyrimidinedione derivative compounds
MX366159B (es)	2012-11-30	2019-07-01	Acura Pharmaceuticals Inc	Liberacion autorregulada de ingrediente farmaceutico activo.
JP2016521747A (ja)	2013-06-13	2016-07-25	アケビアセラピューティクスインコーポレイテッドＡｋｅｂｉａＴｈｅｒａｐｅｕｔｉｃｓＩｎｃ．	貧血治療のための組成物及び方法
WO2015103490A1 (en)	2014-01-03	2015-07-09	Abbvie, Inc.	Solid antiviral dosage forms
US11103581B2 (en)	2015-08-31	2021-08-31	Acura Pharmaceuticals, Inc.	Methods and compositions for self-regulated release of active pharmaceutical ingredient
CA2937365C (en)	2016-03-29	2018-09-18	F. Hoffmann-La Roche Ag	Granulate formulation of 5-methyl-1-phenyl-2-(1h)-pyridone and method of making the same
KR102942294B1 (ko) *	2018-05-15	2026-03-23	장쑤 한서 파마슈티칼 그룹 캄파니 리미티드	소분자 이지에프알 억제제를 포함하는 약학 조성물 및 그의 제조 방법
CN108619104A (zh) *	2018-06-29	2018-10-09	哈尔滨珍宝制药有限公司	一种基于盐酸克林霉素的药物组合物及其制备方法
CZ309820B6 (cs) *	2021-04-23	2023-11-08	Pro.Med.Cs Praha A.S.	Způsob přípravy pevné lékové formy obsahující kompozici s nízkým obsahem účinné látky

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DE3708916A1 (de)	1987-03-19	1988-09-29	Boehringer Ingelheim Kg	Verfahren zur reinigung resorbierbarer polyester
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UA72207C2 (uk) *	1998-04-07	2005-02-15	Брістол- Майєрс Сквібб Фарма Компані	Фармацевтична композиція ефавіренцу з добавкою дезінтегруючих агентів у вигляді швидкорозчинних капсул або таблеток та спосіб її виготовлення
DE69934582T2 (de) *	1998-06-11	2007-10-04	Pharmacia & Upjohn Co. Llc, Kalamazoo	Delavirdin tablettenformulierung

1999
- 1999-06-07 DE DE69934582T patent/DE69934582T2/de not_active Revoked
- 1999-06-07 PL PL344328A patent/PL200163B1/pl unknown
- 1999-06-07 CA CA002328703A patent/CA2328703C/en not_active Expired - Lifetime
- 1999-06-07 EA EA200100024A patent/EA004311B1/ru not_active IP Right Cessation
- 1999-06-07 CN CNB998062316A patent/CN1237958C/zh not_active Expired - Lifetime
- 1999-06-07 AT AT99925951T patent/ATE349203T1/de active
- 1999-06-07 NZ NZ508762A patent/NZ508762A/en not_active IP Right Cessation
- 1999-06-07 KR KR1020007013985A patent/KR100724016B1/ko not_active Expired - Lifetime
- 1999-06-07 WO PCT/US1999/011798 patent/WO1999063970A1/en not_active Ceased
- 1999-06-07 EP EP99925951A patent/EP1083885B1/de not_active Revoked
- 1999-06-07 HU HU0102206A patent/HUP0102206A3/hu unknown
- 1999-06-07 DK DK99925951T patent/DK1083885T3/da active
- 1999-06-07 US US09/327,135 patent/US6177101B1/en not_active Expired - Lifetime
- 1999-06-07 AU AU42134/99A patent/AU753241C/en not_active Expired
- 1999-06-07 PT PT99925951T patent/PT1083885E/pt unknown
- 1999-06-07 KR KR1020077007572A patent/KR20070040426A/ko not_active Ceased
- 1999-06-07 JP JP2000553039A patent/JP4827296B2/ja not_active Expired - Lifetime
- 1999-06-07 BR BR9910481-4A patent/BR9910481A/pt not_active Application Discontinuation
- 1999-06-07 ES ES99925951T patent/ES2277682T3/es not_active Expired - Lifetime
2000
- 2000-09-06 US US09/656,364 patent/US7108864B1/en not_active Expired - Lifetime
- 2000-10-27 ZA ZA200006090A patent/ZA200006090B/xx unknown
2006
- 2006-07-14 US US11/487,554 patent/US20060257476A1/en not_active Abandoned
2007
- 2007-01-15 CY CY20071100050T patent/CY1105924T1/el unknown

Also Published As

Publication number	Publication date
EA200100024A1 (ru)	2001-06-25
CN1301149A (zh)	2001-06-27
US6177101B1 (en)	2001-01-23
WO1999063970A1 (en)	1999-12-16
EA004311B1 (ru)	2004-02-26
ZA200006090B (en)	2001-10-29
KR20010052717A (ko)	2001-06-25
EP1083885A1 (de)	2001-03-21
HUP0102206A3 (en)	2002-12-28
CN1237958C (zh)	2006-01-25
AU4213499A (en)	1999-12-30
KR20070040426A (ko)	2007-04-16
CA2328703A1 (en)	1999-12-16
HK1036417A1 (en)	2002-01-04
AU753241C (en)	2003-05-08
KR100724016B1 (ko)	2007-05-31
ES2277682T3 (es)	2007-07-16
US7108864B1 (en)	2006-09-19
PL200163B1 (pl)	2008-12-31
NZ508762A (en)	2003-07-25
EP1083885B1 (de)	2006-12-27
DK1083885T3 (da)	2007-02-26
HUP0102206A2 (hu)	2002-03-28
DE69934582D1 (de)	2007-02-08
PT1083885E (pt)	2007-01-31
JP4827296B2 (ja)	2011-11-30
CY1105924T1 (el)	2011-04-06
JP2002517430A (ja)	2002-06-18
DE69934582T2 (de)	2007-10-04
AU753241B2 (en)	2002-10-10
US20060257476A1 (en)	2006-11-16
BR9910481A (pt)	2001-01-09
PL344328A1 (en)	2001-10-22
CA2328703C (en)	2007-10-30

Legal Events

Date

Code

Title

Description

2007-07-15

UEP

Publication of translation of european patent specification

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