ATE377605T1 - 6-oxygenierte steroid-estrogene mit aromatischen a- und b-ringen - Google Patents

6-oxygenierte steroid-estrogene mit aromatischen a- und b-ringen

Info

Publication number: ATE377605T1
Authority: AT; Austria
Prior art keywords: hydrogen; group; hydroxy; esters; sulfate
Prior art date: 2000-03-10

Application number

AT01920261T

Other languages

English (en)

Inventor

Edward Hill

Frederick Sancilio

Robert Whittle

Original Assignee

Barr Lab Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-03-10

Filing date

2001-03-09

Publication date

2007-11-15

2001-03-09 Application filed by Barr Lab Inc filed Critical Barr Lab Inc

2007-11-15 Application granted granted Critical

2007-11-15 Publication of ATE377605T1 publication Critical patent/ATE377605T1/de

Links

239000000262 estrogen Substances 0.000 title abstract 2
229940011871 estrogen Drugs 0.000 title 1
150000003431 steroids Chemical class 0.000 title 1
150000002148 esters Chemical class 0.000 abstract 4
QAOWNCQODCNURD-UHFFFAOYSA-N Sulfuric acid Chemical group OS(O)(=O)=O QAOWNCQODCNURD-UHFFFAOYSA-N 0.000 abstract 3
125000000217 alkyl group Chemical group 0.000 abstract 2
150000001875 compounds Chemical class 0.000 abstract 2
125000004356 hydroxy functional group Chemical group O* 0.000 abstract 2
241000124008 Mammalia Species 0.000 abstract 1
125000003545 alkoxy group Chemical group 0.000 abstract 1
BVKZGUZCCUSVTD-UHFFFAOYSA-N carbonic acid Chemical compound OC(O)=O BVKZGUZCCUSVTD-UHFFFAOYSA-N 0.000 abstract 1
125000002915 carbonyl group Chemical group [*:2]C([*:1])=O 0.000 abstract 1
229930182480 glucuronide Natural products 0.000 abstract 1
150000008134 glucuronides Chemical class 0.000 abstract 1
229910052736 halogen Inorganic materials 0.000 abstract 1
150000002367 halogens Chemical class 0.000 abstract 1
229910052739 hydrogen Inorganic materials 0.000 abstract 1
239000001257 hydrogen Substances 0.000 abstract 1
125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 1
239000000203 mixture Substances 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
- C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/30—Oestrogens
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0059—Estrane derivatives substituted in position 17 by a keto group
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0066—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
- C07J1/007—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa the substituent being an OH group free esterified or etherified

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Diabetes (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Endocrinology (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

AT01920261T 2000-03-10 2001-03-09 6-oxygenierte steroid-estrogene mit aromatischen a- und b-ringen ATE377605T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US18853300P	2000-03-10	2000-03-10

Publications (1)

Publication Number	Publication Date
ATE377605T1 true ATE377605T1 (de)	2007-11-15

Family

ID=22693557

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT01920261T ATE377605T1 (de)	2000-03-10	2001-03-09	6-oxygenierte steroid-estrogene mit aromatischen a- und b-ringen

Country Status (6)

Country	Link
EP (1)	EP1263770B1 (de)
AT (1)	ATE377605T1 (de)
AU (1)	AU2001247337A1 (de)
CA (1)	CA2402667C (de)
DE (1)	DE60131253T2 (de)
WO (1)	WO2001068669A1 (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US7235539B2 (en)	2002-01-23	2007-06-26	Wyeth	6-Hydroxyequilenins as estrogenic agents
US6956126B2 (en) *	2002-07-02	2005-10-18	Wyeth	Preparation of 6-hydroxyequilenins

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IL25265A (en) *	1966-02-28	1969-12-31	Harnik M	Estrane derivatives and their preparation
GB1399162A (en) *	1972-06-29	1975-06-25	Schering Ag	6-keto-delta1,3,5-10-steroids and process for the manufacture of 6-keto-delta1,3,5-10-steroids

2001
- 2001-03-09 CA CA2402667A patent/CA2402667C/en not_active Expired - Fee Related
- 2001-03-09 EP EP01920261A patent/EP1263770B1/de not_active Expired - Lifetime
- 2001-03-09 DE DE60131253T patent/DE60131253T2/de not_active Expired - Lifetime
- 2001-03-09 AU AU2001247337A patent/AU2001247337A1/en not_active Abandoned
- 2001-03-09 AT AT01920261T patent/ATE377605T1/de not_active IP Right Cessation
- 2001-03-09 WO PCT/US2001/007544 patent/WO2001068669A1/en not_active Ceased

Also Published As

Publication number	Publication date
EP1263770A1 (de)	2002-12-11
WO2001068669A1 (en)	2001-09-20
DE60131253T2 (de)	2008-08-28
AU2001247337A1 (en)	2001-09-24
EP1263770B1 (de)	2007-11-07
DE60131253D1 (de)	2007-12-20
CA2402667C (en)	2010-05-25
CA2402667A1 (en)	2001-09-20

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Legal Events

Date	Code	Title	Description
2008-05-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties