ATE389405T1 - Fexofenadine hydrochlorid polymorph - Google Patents
Fexofenadine hydrochlorid polymorphInfo
- Publication number
- ATE389405T1 ATE389405T1 AT02751479T AT02751479T ATE389405T1 AT E389405 T1 ATE389405 T1 AT E389405T1 AT 02751479 T AT02751479 T AT 02751479T AT 02751479 T AT02751479 T AT 02751479T AT E389405 T1 ATE389405 T1 AT E389405T1
- Authority
- AT
- Austria
- Prior art keywords
- polymorpho
- fexofenadine hydrochloride
- polymorph
- fexofenadine
- hydrochloride
- Prior art date
Links
- RRJFVPUCXDGFJB-UHFFFAOYSA-N Fexofenadine hydrochloride Chemical compound Cl.C1=CC(C(C)(C(O)=O)C)=CC=C1C(O)CCCN1CCC(C(O)(C=2C=CC=CC=2)C=2C=CC=CC=2)CC1 RRJFVPUCXDGFJB-UHFFFAOYSA-N 0.000 title abstract 2
- 229960000354 fexofenadine hydrochloride Drugs 0.000 title abstract 2
- GUGOEEXESWIERI-UHFFFAOYSA-N Terfenadine Chemical compound C1=CC(C(C)(C)C)=CC=C1C(O)CCCN1CCC(C(O)(C=2C=CC=CC=2)C=2C=CC=CC=2)CC1 GUGOEEXESWIERI-UHFFFAOYSA-N 0.000 abstract 1
- 230000001387 anti-histamine Effects 0.000 abstract 1
- 239000000043 antiallergic agent Substances 0.000 abstract 1
- 239000000739 antihistaminic agent Substances 0.000 abstract 1
- 229940124630 bronchodilator Drugs 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
- C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pulmonology (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP01610081 | 2001-07-31 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE389405T1 true ATE389405T1 (de) | 2008-04-15 |
Family
ID=8183555
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT02751479T ATE389405T1 (de) | 2001-07-31 | 2002-07-29 | Fexofenadine hydrochlorid polymorph |
Country Status (7)
| Country | Link |
|---|---|
| US (2) | US20040248935A1 (de) |
| EP (1) | EP1414453B1 (de) |
| AT (1) | ATE389405T1 (de) |
| DE (1) | DE60225694T2 (de) |
| ES (1) | ES2301662T3 (de) |
| PT (1) | PT1414453E (de) |
| WO (1) | WO2003011295A1 (de) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL158334A0 (en) * | 2001-04-09 | 2004-05-12 | Teva Pharma | Polymorphs of fexofenadine hydrochloride |
| US20040044038A1 (en) | 2002-06-10 | 2004-03-04 | Barnaba Krochmal | Polymorphic form XVI of fexofenadine hydrochloride |
| GB0319935D0 (en) | 2003-08-26 | 2003-09-24 | Cipla Ltd | Polymorphs |
| JP2007532687A (ja) * | 2004-04-26 | 2007-11-15 | テバ ファーマシューティカル インダストリーズ リミティド | フェキソフェナジン塩酸塩の結晶形およびその製造方法 |
| ITMI20041143A1 (it) * | 2004-06-08 | 2004-09-08 | Dipharma Spa | Polimorfi di fexofenadina e procedimento per la loro preparazione |
| WO2007052310A2 (en) * | 2005-11-03 | 2007-05-10 | Morepen Laboratories Limited | Polymorphs of fexofenadine hydrochloride and process for their preparation |
| DOP2006000274A (es) | 2005-12-14 | 2007-10-15 | Sanofi Aventis Us Llc | Formulación de suspensión de fexofenadina |
| US20080095843A1 (en) * | 2006-07-11 | 2008-04-24 | Nutalapati Siva R K | Controlled-release formulations |
| US20090306135A1 (en) | 2008-03-24 | 2009-12-10 | Mukesh Kumar Sharma | Stable amorphous fexofenadine hydrochloride |
| WO2010083360A2 (en) * | 2009-01-16 | 2010-07-22 | Mutual Pharmaceutical Company, Inc. | Controlled-release formulations |
| ES2403130B1 (es) | 2010-06-15 | 2014-09-29 | Chemelectiva S.R.L. | Forma polimórfica de clorhidrato de fexofenadina, compuestos intermedios y procedimiento para su preparación |
| CN104072402B (zh) * | 2014-07-16 | 2016-08-17 | 昆山龙灯瑞迪制药有限公司 | 一种新结晶形式的盐酸非索非那定化合物及其制备方法 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1178041A1 (de) * | 1994-05-18 | 2002-02-06 | Aventis Pharmaceuticals Inc. | Verfahren zur Herstellung von wasserfreien und Hydrat-Formen von antihistaminischen Piperidinderivaten |
| DK0812195T3 (da) * | 1995-02-28 | 2003-03-03 | Aventis Pharma Inc | Farmaceutisk sammensætning til piperidinoalkanolforbindelser |
-
2002
- 2002-07-29 WO PCT/IB2002/002954 patent/WO2003011295A1/en not_active Ceased
- 2002-07-29 ES ES02751479T patent/ES2301662T3/es not_active Expired - Lifetime
- 2002-07-29 AT AT02751479T patent/ATE389405T1/de not_active IP Right Cessation
- 2002-07-29 EP EP02751479A patent/EP1414453B1/de not_active Expired - Lifetime
- 2002-07-29 US US10/485,391 patent/US20040248935A1/en not_active Abandoned
- 2002-07-29 DE DE60225694T patent/DE60225694T2/de not_active Expired - Fee Related
- 2002-07-29 PT PT02751479T patent/PT1414453E/pt unknown
-
2009
- 2009-09-18 US US12/562,725 patent/US20100010229A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| EP1414453B1 (de) | 2008-03-19 |
| DE60225694T2 (de) | 2008-06-26 |
| WO2003011295B1 (en) | 2003-04-03 |
| ES2301662T3 (es) | 2008-07-01 |
| EP1414453A1 (de) | 2004-05-06 |
| US20040248935A1 (en) | 2004-12-09 |
| WO2003011295A1 (en) | 2003-02-13 |
| DE60225694D1 (de) | 2008-04-30 |
| PT1414453E (pt) | 2008-05-29 |
| US20100010229A1 (en) | 2010-01-14 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification |
Ref document number: 1414453 Country of ref document: EP |
|
| REN | Ceased due to non-payment of the annual fee |