ATE400179T1 - Verwendung von pyrimidinetrion-derivaten als acetylcholinesterase-hemmer, diese enthaltende zusammensetzungen und deren verwendungen - Google Patents

Verwendung von pyrimidinetrion-derivaten als acetylcholinesterase-hemmer, diese enthaltende zusammensetzungen und deren verwendungen

Info

Publication number
ATE400179T1
ATE400179T1 AT06755417T AT06755417T ATE400179T1 AT E400179 T1 ATE400179 T1 AT E400179T1 AT 06755417 T AT06755417 T AT 06755417T AT 06755417 T AT06755417 T AT 06755417T AT E400179 T1 ATE400179 T1 AT E400179T1
Authority
AT
Austria
Prior art keywords
acetylcholinesterase
optionally substituted
acetylcholinesterase inhibitors
derivatives
pyrimidinetrion
Prior art date
Application number
AT06755417T
Other languages
English (en)
Inventor
Mylene Weill
Philippe Fort
Jean-Paul Leonetti
Original Assignee
Centre Nat Rech Scient
Univ Montpellier Ii
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Centre Nat Rech Scient, Univ Montpellier Ii filed Critical Centre Nat Rech Scient
Application granted granted Critical
Publication of ATE400179T1 publication Critical patent/ATE400179T1/de

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Agronomy & Crop Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Plant Pathology (AREA)
  • Biomedical Technology (AREA)
  • Epidemiology (AREA)
  • Pest Control & Pesticides (AREA)
  • General Chemical & Material Sciences (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AT06755417T 2005-02-10 2006-02-10 Verwendung von pyrimidinetrion-derivaten als acetylcholinesterase-hemmer, diese enthaltende zusammensetzungen und deren verwendungen ATE400179T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0501328A FR2881618B1 (fr) 2005-02-10 2005-02-10 Utilisation de composes derives de pyrimidinetrione en tant qu'inhibiteurs de l'acetylcholinesterase, compositions contenant ces derives et leurs utilisations en tant qu'insecticides

Publications (1)

Publication Number Publication Date
ATE400179T1 true ATE400179T1 (de) 2008-07-15

Family

ID=35406144

Family Applications (1)

Application Number Title Priority Date Filing Date
AT06755417T ATE400179T1 (de) 2005-02-10 2006-02-10 Verwendung von pyrimidinetrion-derivaten als acetylcholinesterase-hemmer, diese enthaltende zusammensetzungen und deren verwendungen

Country Status (8)

Country Link
US (1) US8309556B2 (de)
EP (1) EP1845781B1 (de)
AT (1) ATE400179T1 (de)
CA (1) CA2597349C (de)
DE (1) DE602006001731D1 (de)
ES (1) ES2312134T3 (de)
FR (1) FR2881618B1 (de)
WO (1) WO2006097588A1 (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2011215870B2 (en) 2010-02-09 2016-01-28 The Johns Hopkins University Methods and compositions for improving cognitive function
US20140206667A1 (en) 2012-11-14 2014-07-24 Michela Gallagher Methods and compositions for treating schizophrenia
JP6433482B2 (ja) 2013-03-15 2018-12-05 エージンバイオ, インコーポレイテッド 認知機能を改善するための方法および組成物
WO2014144663A1 (en) 2013-03-15 2014-09-18 The Johns Hopkins University Methods and compositions for improving cognitive function
WO2016191288A1 (en) 2015-05-22 2016-12-01 Agenebio, Inc. Extended release pharmaceutical compositions of levetiracetam

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR382112A (fr) 1907-09-20 1908-01-30 Juan Puig Y Marco Appareil indiquant à tout instant la longueur de tissu fabriqué par un métier
FR455300A (fr) 1913-03-08 1913-07-26 Deutsche Maschf Ag Chariot de coulée
DE3903404A1 (de) * 1989-02-06 1990-08-09 Hoechst Ag Pyrimidintrionderivate, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als schaedlingsbekaempfungsmittel
NL9001075A (de) * 1990-05-04 1991-12-02 Duphar Int Res
US20050049267A1 (en) * 2002-03-01 2005-03-03 Pintex Pharmaceuticals, Inc. Pin1-modulating compounds and methods of use thereof

Also Published As

Publication number Publication date
WO2006097588A1 (fr) 2006-09-21
EP1845781A1 (de) 2007-10-24
CA2597349C (fr) 2015-05-26
EP1845781B1 (de) 2008-07-09
US8309556B2 (en) 2012-11-13
ES2312134T3 (es) 2009-02-16
FR2881618A1 (fr) 2006-08-11
FR2881618B1 (fr) 2007-04-13
CA2597349A1 (fr) 2006-09-21
DE602006001731D1 (de) 2008-08-21
US20080269252A1 (en) 2008-10-30

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Legal Events

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