ATE418543T1 - Substituierte 1,4-dipiperidin-4-yl- piperazinderivate und deren verwendung als neurokininantagonisten - Google Patents

Substituierte 1,4-dipiperidin-4-yl- piperazinderivate und deren verwendung als neurokininantagonisten

Info

Publication number: ATE418543T1
Authority: AT; Austria
Prior art keywords: dipiperidine; substituted; piperazine derivatives; neurokin antagonists; neurokin
Prior art date: 2002-10-08

Application number

AT03773731T

Other languages

German (de)

English (en)

Inventor

Frans Eduard Janssens

Francois Maria Sommen

Boeck Benoit Christian Albert De

Joseph Elisabeth Leenaerts

Roosbroeck Yves Emiel Maria Van

Gaston Stanislas Marcella Diels

Original Assignee

Janssen Pharmaceutica Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-10-08

Filing date

2003-10-07

Publication date

2009-01-15

2002-12-23 Priority claimed from PCT/EP2002/014836 external-priority patent/WO2004056772A1/fr

2003-10-07 Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv

2009-01-15 Application granted granted Critical

2009-01-15 Publication of ATE418543T1 publication Critical patent/ATE418543T1/de

Links

TYYZPUUMIWNDKS-UHFFFAOYSA-N 1,4-di(piperidin-4-yl)piperazine Chemical class C1CNCCC1N1CCN(C2CCNCC2)CC1 TYYZPUUMIWNDKS-UHFFFAOYSA-N 0.000 title 1
239000005557 antagonist Substances 0.000 title 1

Classifications

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- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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AT03773731T 2002-10-08 2003-10-07 Substituierte 1,4-dipiperidin-4-yl- piperazinderivate und deren verwendung als neurokininantagonisten ATE418543T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP0211328		2002-10-08
PCT/EP2002/014836 WO2004056772A1 (fr)	2002-12-23	2002-12-23	Derives de 1,4-di-piperidin-4-yl-piperazine substitues et leur utilisation comme antagonistes de la tachykinine

Publications (1)

Publication Number	Publication Date
ATE418543T1 true ATE418543T1 (de)	2009-01-15

Family

ID=32094938

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT03773731T ATE418543T1 (de)	2002-10-08	2003-10-07	Substituierte 1,4-dipiperidin-4-yl- piperazinderivate und deren verwendung als neurokininantagonisten

Country Status (18)

Country	Link
US (1)	US7410970B2 (fr)
EP (1)	EP1551804B1 (fr)
JP (1)	JP4674086B2 (fr)
KR (1)	KR101049074B1 (fr)
AR (1)	AR041545A1 (fr)
AT (1)	ATE418543T1 (fr)
AU (1)	AU2003282115B2 (fr)
BR (1)	BR0315098A (fr)
CA (1)	CA2499903C (fr)
DE (1)	DE60325493D1 (fr)
EA (1)	EA009217B1 (fr)
ES (1)	ES2319642T3 (fr)
HR (1)	HRP20050309A2 (fr)
IL (1)	IL167885A (fr)
MY (1)	MY141736A (fr)
PA (1)	PA8584901A1 (fr)
TW (1)	TWI324995B (fr)
WO (1)	WO2004033428A1 (fr)

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JP2013503908A (ja) *	2009-09-04	2013-02-04	ユナイテッドパラゴンアソシエイツインコーポレイテッド	ニューロキニン２受容体活性に関連する障害または疾患を治療するための化合物
CA2900710C (fr)	2013-02-08	2023-08-08	General Mills, Inc.	Produit alimentaire a teneur reduite en sodium
KR101472916B1 (ko)	2013-06-27	2014-12-16	한국과학기술연구원	모르폴린 또는 피페라진 화합물, 및 도네페질을 포함하는 인지 장애 관련 질병의 예방 또는 치료용 약학적 조성물
EP3915560A1 (fr)	2014-06-25	2021-12-01	Emory University	Procédés de gestion d'une peur conditionnée à l'aide d'antagonistes du récepteur de la neurokinine
RU2617694C1 (ru) *	2015-12-24	2017-04-26	Федеральное государственное бюджетное учреждение науки Институт элементоорганических соединений им. А.Н. Несмеянова Российской академии наук (ИНЭОС РАН)	Амиды акриловой и метакриловой кислот с олигопиперидинами и способ их получения
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2003
- 2003-10-06 MY MYPI20033797A patent/MY141736A/en unknown
- 2003-10-07 WO PCT/EP2003/050697 patent/WO2004033428A1/fr not_active Ceased
- 2003-10-07 AR ARP030103649A patent/AR041545A1/es unknown
- 2003-10-07 US US10/527,821 patent/US7410970B2/en not_active Expired - Fee Related
- 2003-10-07 TW TW092127724A patent/TWI324995B/zh active
- 2003-10-07 EA EA200500616A patent/EA009217B1/ru not_active IP Right Cessation
- 2003-10-07 AU AU2003282115A patent/AU2003282115B2/en not_active Ceased
- 2003-10-07 BR BR0315098-4A patent/BR0315098A/pt not_active IP Right Cessation
- 2003-10-07 EP EP03773731A patent/EP1551804B1/fr not_active Expired - Lifetime
- 2003-10-07 DE DE60325493T patent/DE60325493D1/de not_active Expired - Lifetime
- 2003-10-07 CA CA2499903A patent/CA2499903C/fr not_active Expired - Fee Related
- 2003-10-07 ES ES03773731T patent/ES2319642T3/es not_active Expired - Lifetime
- 2003-10-07 AT AT03773731T patent/ATE418543T1/de not_active IP Right Cessation
- 2003-10-07 JP JP2004542503A patent/JP4674086B2/ja not_active Expired - Fee Related
- 2003-10-07 HR HR20050309A patent/HRP20050309A2/xx not_active Application Discontinuation
- 2003-10-07 KR KR1020057003472A patent/KR101049074B1/ko not_active Expired - Fee Related
- 2003-10-08 PA PA20038584901A patent/PA8584901A1/es unknown
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Also Published As

Publication number	Publication date
AU2003282115B2 (en)	2009-10-01
CA2499903C (fr)	2011-06-14
ES2319642T3 (es)	2009-05-11
EP1551804A1 (fr)	2005-07-13
MY141736A (en)	2010-06-15
EP1551804B1 (fr)	2008-12-24
US20060167008A1 (en)	2006-07-27
IL167885A (en)	2010-04-29
TW200413319A (en)	2004-08-01
JP4674086B2 (ja)	2011-04-20
US7410970B2 (en)	2008-08-12
CA2499903A1 (fr)	2004-04-22
EA009217B1 (ru)	2007-12-28
KR101049074B1 (ko)	2011-07-15
WO2004033428A1 (fr)	2004-04-22
HK1084394A1 (zh)	2006-07-28
TWI324995B (en)	2010-05-21
BR0315098A (pt)	2005-08-16
KR20050059164A (ko)	2005-06-17
EA200500616A1 (ru)	2005-10-27
AR041545A1 (es)	2005-05-18
JP2006510602A (ja)	2006-03-30
PA8584901A1 (es)	2005-10-28
DE60325493D1 (de)	2009-02-05
AU2003282115A1 (en)	2004-05-04
HRP20050309A2 (en)	2006-07-31

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2009-06-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties

Publication	Publication Date	Title
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DE60106607D1 (de)	2004-11-25	Substituierte 1-aminoalkyl-lactame und ihre verwendung als muscarinrezeptor antagonisten
DE50111690D1 (de)	2007-02-01	2-acyl-indolderivate und deren verwendung als antitumormittel
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DE60114413D1 (de)	2005-12-01	Substituierte 1-aminoalkyl-lactame und deren verwendung als muscarinrezeptor-antagonisten
DE602005011593D1 (de)	2009-01-22	Substituierte diazaspiroä5.5üundecanderivate und deren verwendung als neurokininantagonisten
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ATE353083T1 (de)	2007-02-15	Naphthyridin-derivate und ihre verwendung als fungizide
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ATE361295T1 (de)	2007-05-15	Substituierte diketopiperazine und deren verwendung als oxytocynantagonisten
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DE50313185D1 (de)	2010-11-25	2-pyrrolidin-2-yl-ä1,3,4ü -oxadiazol-derivate und ihre verwendung als antidepressiva
DE60324586D1 (de)	2008-12-18	Substituierte pyridyloxyalkylamide und ihre verwendung als fungizide
ATE430733T1 (de)	2009-05-15	6-(1,1-difluoralkyl)-4-aminopicolinate und deren verwendung als herbizide