ATE431341T1 - P-toluenosulfonatsalz des n-methyl-n-(3,5- dimatoxy-2,4,6-triazinyl-1-)-morpholins und verwandte verbindungen zur verwendung als kondensationsreagenz in der peptidsynthese - Google Patents
P-toluenosulfonatsalz des n-methyl-n-(3,5- dimatoxy-2,4,6-triazinyl-1-)-morpholins und verwandte verbindungen zur verwendung als kondensationsreagenz in der peptidsyntheseInfo
- Publication number
- ATE431341T1 ATE431341T1 AT05006473T AT05006473T ATE431341T1 AT E431341 T1 ATE431341 T1 AT E431341T1 AT 05006473 T AT05006473 T AT 05006473T AT 05006473 T AT05006473 T AT 05006473T AT E431341 T1 ATE431341 T1 AT E431341T1
- Authority
- AT
- Austria
- Prior art keywords
- group
- anion
- substituted
- heterocyclic
- toluenosulfonate
- Prior art date
Links
- 239000003153 chemical reaction reagent Substances 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 title abstract 2
- 238000009833 condensation Methods 0.000 title 1
- 230000005494 condensation Effects 0.000 title 1
- 238000010647 peptide synthesis reaction Methods 0.000 title 1
- 150000003839 salts Chemical class 0.000 title 1
- 150000001450 anions Chemical class 0.000 abstract 7
- 125000000623 heterocyclic group Chemical group 0.000 abstract 5
- -1 arylsulfonate anion Chemical class 0.000 abstract 3
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 125000003118 aryl group Chemical group 0.000 abstract 2
- 125000004104 aryloxy group Chemical group 0.000 abstract 2
- 150000002148 esters Chemical class 0.000 abstract 2
- 125000000547 substituted alkyl group Chemical group 0.000 abstract 2
- 125000003107 substituted aryl group Chemical group 0.000 abstract 2
- 238000003786 synthesis reaction Methods 0.000 abstract 2
- QAOWNCQODCNURD-UHFFFAOYSA-L Sulfate Chemical compound [O-]S([O-])(=O)=O QAOWNCQODCNURD-UHFFFAOYSA-L 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 150000001408 amides Chemical class 0.000 abstract 1
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 abstract 1
- 229910052757 nitrogen Inorganic materials 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- 102000004196 processed proteins & peptides Human genes 0.000 abstract 1
- 108090000765 processed proteins & peptides Proteins 0.000 abstract 1
- 125000005415 substituted alkoxy group Chemical group 0.000 abstract 1
- 125000005338 substituted cycloalkoxy group Chemical group 0.000 abstract 1
- 125000005346 substituted cycloalkyl group Chemical group 0.000 abstract 1
- 150000003460 sulfonic acids Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D251/00—Heterocyclic compounds containing 1,3,5-triazine rings
- C07D251/02—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings
- C07D251/12—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D251/26—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with only hetero atoms directly attached to ring carbon atoms
- C07D251/40—Nitrogen atoms
- C07D251/42—One nitrogen atom
- C07D251/46—One nitrogen atom with oxygen or sulfur atoms attached to the two other ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
- C07K1/08—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using activating agents
- C07K1/084—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using activating agents containing nitrogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/10—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using coupling agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Analytical Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PL366673A PL211025B1 (pl) | 2004-03-29 | 2004-03-29 | Czwartorzędowe sole N-(3,5-dipodstawionych-2,4,6-triazynylo-1-)amoniowych kwasów sulfonowych i ich zastosowanie |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE431341T1 true ATE431341T1 (de) | 2009-05-15 |
Family
ID=34934485
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT05006473T ATE431341T1 (de) | 2004-03-29 | 2005-03-24 | P-toluenosulfonatsalz des n-methyl-n-(3,5- dimatoxy-2,4,6-triazinyl-1-)-morpholins und verwandte verbindungen zur verwendung als kondensationsreagenz in der peptidsynthese |
Country Status (4)
| Country | Link |
|---|---|
| EP (1) | EP1586566B9 (de) |
| AT (1) | ATE431341T1 (de) |
| DE (1) | DE602005014413D1 (de) |
| PL (2) | PL211025B1 (de) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2006107963A2 (en) * | 2005-04-06 | 2006-10-12 | Novartis Ag | Process for preparing dipeptide amides |
| PL391832A1 (pl) | 2010-07-14 | 2012-01-16 | Politechnika Łódzka | Sole N-triazynyloamoniowe, sposób ich wytwarzania oraz ich zastosowanie |
| CZ306115B6 (cs) * | 2012-12-04 | 2016-08-10 | Zentiva, K.S. | Způsob přípravy derivátů kyseliny 3-amino-4-(2,4,5-trifluorfenyl)-butanové |
| JP6705111B2 (ja) * | 2016-02-25 | 2020-06-03 | 国立大学法人金沢大学 | トリアジノン化合物 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10029139A1 (de) * | 2000-06-14 | 2002-01-03 | Sueddeutsche Kalkstickstoff | Verfahren zur Herstellung von Amiden oder Estern |
-
2004
- 2004-03-29 PL PL366673A patent/PL211025B1/pl not_active IP Right Cessation
-
2005
- 2005-03-24 DE DE602005014413T patent/DE602005014413D1/de not_active Expired - Lifetime
- 2005-03-24 AT AT05006473T patent/ATE431341T1/de not_active IP Right Cessation
- 2005-03-24 PL PL05006473T patent/PL1586566T3/pl unknown
- 2005-03-24 EP EP05006473A patent/EP1586566B9/de not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| EP1586566B1 (de) | 2009-05-13 |
| PL211025B1 (pl) | 2012-03-30 |
| EP1586566A1 (de) | 2005-10-19 |
| PL366673A1 (en) | 2005-10-03 |
| EP1586566B9 (de) | 2009-11-18 |
| PL1586566T3 (pl) | 2009-10-30 |
| DE602005014413D1 (de) | 2009-06-25 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |