ATE447579T1 - Verfahren zur herstellung von 1-hydroxy-2- substituierten cyclohexylazetidin-2-on- verbindungen - Google Patents

Verfahren zur herstellung von 1-hydroxy-2- substituierten cyclohexylazetidin-2-on- verbindungen

Info

Publication number
ATE447579T1
ATE447579T1 AT06792145T AT06792145T ATE447579T1 AT E447579 T1 ATE447579 T1 AT E447579T1 AT 06792145 T AT06792145 T AT 06792145T AT 06792145 T AT06792145 T AT 06792145T AT E447579 T1 ATE447579 T1 AT E447579T1
Authority
AT
Austria
Prior art keywords
formula
compound
trifluoromethanesulfonate
nucleophile
microwave irradiation
Prior art date
Application number
AT06792145T
Other languages
English (en)
Inventor
Lovro Selic
Gregor Vilfan
Uros Urleb
Original Assignee
Lek Pharmaceuticals
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lek Pharmaceuticals filed Critical Lek Pharmaceuticals
Application granted granted Critical
Publication of ATE447579T1 publication Critical patent/ATE447579T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/18Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804Compounds having Si-O-C linkages
    • C07F7/1872Preparation; Treatments not provided for in C07F7/20
    • C07F7/1892Preparation; Treatments not provided for in C07F7/20 by reactions not provided for in C07F7/1876 - C07F7/1888
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AT06792145T 2005-09-21 2006-09-19 Verfahren zur herstellung von 1-hydroxy-2- substituierten cyclohexylazetidin-2-on- verbindungen ATE447579T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SI200500269 2005-09-21
PCT/EP2006/009101 WO2007039099A1 (en) 2005-09-21 2006-09-19 Process for preparing 1’-hydroxy-2’-substituted cyclohexyl azetidin-2-one compounds

Publications (1)

Publication Number Publication Date
ATE447579T1 true ATE447579T1 (de) 2009-11-15

Family

ID=37498010

Family Applications (1)

Application Number Title Priority Date Filing Date
AT06792145T ATE447579T1 (de) 2005-09-21 2006-09-19 Verfahren zur herstellung von 1-hydroxy-2- substituierten cyclohexylazetidin-2-on- verbindungen

Country Status (10)

Country Link
US (1) US20090234139A1 (de)
EP (1) EP1940853B1 (de)
JP (1) JP2009508898A (de)
CN (1) CN101268086A (de)
AT (1) ATE447579T1 (de)
AU (1) AU2006299169A1 (de)
CA (1) CA2621327A1 (de)
DE (1) DE602006010228D1 (de)
SI (1) SI1940853T1 (de)
WO (1) WO2007039099A1 (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2015527376A (ja) * 2012-09-05 2015-09-17 浙江海正薬業股▲ふん▼有限公司Zhejiang Hisun Pharmaceutical CO.,LTD. アゼチジノン化合物の結晶及びその調製方法
CN109134335B (zh) * 2017-06-27 2022-05-17 苏州引航生物科技有限公司 一种制备手性(1r,2s)-1-苯基-2-(1-吡咯烷基)丙烷-1-醇的方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9104832D0 (en) * 1991-03-07 1991-04-17 Glaxo Spa Heterocyclic compounds
JP4257827B2 (ja) * 2002-12-27 2009-04-22 ミヨシ油脂株式会社 両性界面活性剤の製造方法

Also Published As

Publication number Publication date
CA2621327A1 (en) 2007-04-12
SI1940853T1 (sl) 2010-03-31
CN101268086A (zh) 2008-09-17
DE602006010228D1 (de) 2009-12-17
WO2007039099A1 (en) 2007-04-12
AU2006299169A1 (en) 2007-04-12
EP1940853B1 (de) 2009-11-04
US20090234139A1 (en) 2009-09-17
EP1940853A1 (de) 2008-07-09
JP2009508898A (ja) 2009-03-05

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