ATE449102T1 - Kristallines azithromycin-l-malat-monohydrat und pharmazeutische zusammensetzung, die dieses enthält - Google Patents

Kristallines azithromycin-l-malat-monohydrat und pharmazeutische zusammensetzung, die dieses enthält

Info

Publication number
ATE449102T1
ATE449102T1 AT06747495T AT06747495T ATE449102T1 AT E449102 T1 ATE449102 T1 AT E449102T1 AT 06747495 T AT06747495 T AT 06747495T AT 06747495 T AT06747495 T AT 06747495T AT E449102 T1 ATE449102 T1 AT E449102T1
Authority
AT
Austria
Prior art keywords
pharmaceutical composition
composition containing
containing same
crystalline azithromycin
malate monohydrate
Prior art date
Application number
AT06747495T
Other languages
English (en)
Inventor
Bo Sung Kwon
Eun Sook Kim
Hee Cheol Kim
Sangmin Yun
Myoung-Sil Ko
Tae Hun Song
Han Kyong Kim
Kwee Hyun Suh
Gwansun Lee
Original Assignee
Hanmi Pharm Ind Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hanmi Pharm Ind Co Ltd filed Critical Hanmi Pharm Ind Co Ltd
Application granted granted Critical
Publication of ATE449102T1 publication Critical patent/ATE449102T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Genetics & Genomics (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
AT06747495T 2005-06-08 2006-06-05 Kristallines azithromycin-l-malat-monohydrat und pharmazeutische zusammensetzung, die dieses enthält ATE449102T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
KR1020050048923A KR100666091B1 (ko) 2005-06-08 2005-06-08 아지스로마이신 ｌ-말산염 일수화물 및 이를 포함하는 약학조성물
PCT/KR2006/002157 WO2006132486A1 (en) 2005-06-08 2006-06-05 Crystalline azithromycin l-malate monohydrate and pharmaceutical composition containing same

Publications (1)

Publication Number Publication Date
ATE449102T1 true ATE449102T1 (de) 2009-12-15

Family

ID=37498652

Family Applications (1)

Application Number Title Priority Date Filing Date
AT06747495T ATE449102T1 (de) 2005-06-08 2006-06-05 Kristallines azithromycin-l-malat-monohydrat und pharmazeutische zusammensetzung, die dieses enthält

Country Status (13)

Country Link
US (1) US20090318375A1 (de)
EP (1) EP1910392B1 (de)
JP (1) JP2008543749A (de)
KR (1) KR100666091B1 (de)
CN (1) CN101193904A (de)
AT (1) ATE449102T1 (de)
AU (1) AU2006255914B2 (de)
CA (1) CA2610449A1 (de)
DE (1) DE602006010565D1 (de)
ES (1) ES2333610T3 (de)
IL (1) IL187639A0 (de)
RU (1) RU2348644C1 (de)
WO (1) WO2006132486A1 (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8106111B2 (en) 2009-05-15 2012-01-31 Eastman Chemical Company Antimicrobial effect of cycloaliphatic diol antimicrobial agents in coating compositions
RU2512683C2 (ru) 2012-06-08 2014-04-10 Общество с ограниченной ответственностью "ВИК-здоровье животных" Антибактериальная инъекционная фармацевтическая композиция
CN115057814A (zh) * 2021-12-07 2022-09-16 山东新时代药业有限公司 一种米力农苹果酸盐晶体
CN120842284B (zh) * 2025-09-24 2025-12-02 济南大学 一种低溶剂残留的小粒度富马酸阿奇霉素结晶工艺
CN120842293B (zh) * 2025-09-24 2025-12-02 济南大学 一种低引湿性富马酸阿奇霉素新晶型b及其制备方法

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI8110592A8 (en) * 1981-03-06 1996-06-30 Pliva Pharm & Chem Works Process for preparing of n-methyl-11-aza-10-deoxo-10-dihydroerythromycine a and derivatives thereof
US4474768A (en) * 1982-07-19 1984-10-02 Pfizer Inc. N-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates therefor
CA2245398C (en) * 1998-08-21 2002-01-29 Apotex Inc. Azithromycin monohydrate isopropanol clathrate and methods for the manufacture thereof
SI20639A (sl) * 1998-11-30 2002-02-28 Teva Pharmaceutical Industries Ltd. Etanolat azitromicina, postopek za njegovo pripravo in njegovi farmacevtski sestavki
EP1246831B1 (de) * 2000-01-04 2008-03-05 Teva Pharmaceutical Industries Ltd. Verfahren zur herstellung von azithromycin-dihydrat
ES2162764B1 (es) * 2000-05-17 2003-04-01 Ercros Ind Sa Forma polimorfica del dihidrato de azitromicina, y su procedimiento deobtencion.
HRP20030430B1 (hr) * 2000-11-27 2011-11-30 Biochemie S.A. Makrolidni solvati
CN100341886C (zh) * 2000-11-27 2007-10-10 桑多斯股份公司 大环内酯类化合物的溶剂化物
IN190080B (de) * 2001-01-29 2003-06-07 Alembic Ltd
KR100491183B1 (ko) * 2001-03-21 2005-05-25 한미약품 주식회사 아지트로마이신의 제조방법 및 이 방법에 사용되는9-데옥소-9에이-아자-9에이-호모에리트로마이신 에이의결정성 수화물
KR100431431B1 (ko) * 2001-04-25 2004-05-14 한미약품 주식회사 아지트로마이신 수화물의 1,2-프로필렌글리콜 내포화합물,그의 제조방법 및 그의 약학적 조성물
US6855813B2 (en) * 2002-07-19 2005-02-15 Alembic Limited Process for the preparation of azithromycin monohydrate
HRP20020614A2 (en) * 2002-07-22 2004-06-30 PLIVA-ISTRAŽIVAČKI INSTITUT d.o.o. Rhombic pseudopolymorph of 9-deoxo-9a-aza-9a-methyl-9a-homoerythromycin a
ES2220229B1 (es) 2003-05-29 2005-10-16 Quimica Sintetica, S.A. Sales de adicion de azitromicina y acido citrico y procedimiento para su obtencion.
GB2395482A (en) * 2003-07-03 2004-05-26 Jubilant Organosys Ltd Process for preparing non-hygroscopic azithromycin dihydrate
US20050013835A1 (en) * 2003-07-15 2005-01-20 Pfizer Inc. Stable non-dihydrate azithromycin oral suspensions

Also Published As

Publication number Publication date
CN101193904A (zh) 2008-06-04
KR20060128066A (ko) 2006-12-14
AU2006255914A1 (en) 2006-12-14
WO2006132486A1 (en) 2006-12-14
DE602006010565D1 (de) 2009-12-31
ES2333610T3 (es) 2010-02-24
KR100666091B1 (ko) 2007-01-10
IL187639A0 (en) 2008-03-20
RU2348644C1 (ru) 2009-03-10
CA2610449A1 (en) 2006-12-14
JP2008543749A (ja) 2008-12-04
EP1910392A1 (de) 2008-04-16
US20090318375A1 (en) 2009-12-24
EP1910392A4 (de) 2008-10-29
EP1910392B1 (de) 2009-11-18
AU2006255914B2 (en) 2009-09-03

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