ATE465741T1 - 9a-carbamoyl-y-aminopropyl- und 9a-thiocarbamoyl- y-aminopropyl-azalide mit antimalaria-aktivität - Google Patents

9a-carbamoyl-y-aminopropyl- und 9a-thiocarbamoyl- y-aminopropyl-azalide mit antimalaria-aktivität

Info

Publication number: ATE465741T1
Authority: AT; Austria
Prior art keywords: aminopropyl; thiocarbamoyl; carbamoyl; azalides; homoerythromycin
Prior art date: 2005-01-14

Application number

AT06727593T

Other languages

English (en)

Inventor

Krajacic Mirjana Bukvic

Nedjeljko Kujundzic

Zrinka Ivezic

Sulejman Alihodzic

Antun Hutinec

Andrea Fajdetic

Original Assignee

Glaxosmithkline Zagreb

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2005-01-14

Filing date

2006-01-13

Publication date

2010-05-15

2006-01-13 Application filed by Glaxosmithkline Zagreb filed Critical Glaxosmithkline Zagreb

2010-05-15 Application granted granted Critical

2010-05-15 Publication of ATE465741T1 publication Critical patent/ATE465741T1/de

Links

230000000078 anti-malarial effect Effects 0.000 title abstract 3
150000001875 compounds Chemical class 0.000 abstract 2

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/06—Antimalarials
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Organic Chemistry (AREA)
Medicinal Chemistry (AREA)
Molecular Biology (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Tropical Medicine & Parasitology (AREA)
Epidemiology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
Genetics & Genomics (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

AT06727593T 2005-01-14 2006-01-13 9a-carbamoyl-y-aminopropyl- und 9a-thiocarbamoyl- y-aminopropyl-azalide mit antimalaria-aktivität ATE465741T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US64436005P	2005-01-14	2005-01-14
PCT/IB2006/001227 WO2006085228A2 (en)	2005-01-14	2006-01-13	9a-carbamoyl-y-aminopropyl and 9a-thiocarbamoyl-y-aminopropyl-azalides with antimalarial activity

Publications (1)

Publication Number	Publication Date
ATE465741T1 true ATE465741T1 (de)	2010-05-15

Family

ID=36793417

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT06727593T ATE465741T1 (de)	2005-01-14	2006-01-13	9a-carbamoyl-y-aminopropyl- und 9a-thiocarbamoyl- y-aminopropyl-azalide mit antimalaria-aktivität

Country Status (7)

Country	Link
US (1)	US20080200404A1 (de)
EP (1)	EP1855696B1 (de)
JP (1)	JP2008526949A (de)
AT (1)	ATE465741T1 (de)
DE (1)	DE602006013953D1 (de)
ES (1)	ES2344518T3 (de)
WO (1)	WO2006085228A2 (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP1835921B1 (de) *	2005-01-14	2010-08-18	GlaxoSmithKline istrazivacki centar Zagreb d.o.o.	9a-carbamoyl-y-aminopropyl- und 9a-thiocarbamoyl-y-aminopropyl-azalide mit antimalaria-aktivität
EP2012776A2 (de) *	2006-05-03	2009-01-14	GlaxoSmithKline istrazivacki centar Zagreb d.o.o.	9a-substituierte azalide
PE20090879A1 (es) *	2007-07-30	2009-07-25	Glaxosmithkline Zagreb	DERIVADOS 9-DESOXO-9a-METIL-9a-AZA-9a-HOMOERITROMICINA A COMO AGENTES ANTIMALARICOS
TWI486451B (zh) *	2013-12-11	2015-06-01	Ind Tech Res Inst	經分離之人類肝癌細胞株及化合物篩選方法
TWI461535B (zh) *	2013-12-11	2014-11-21	Ind Tech Res Inst	經分離之人類肝癌細胞株及化合物篩選方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
HRP20020991A2 (en) *	2002-12-12	2005-02-28	Pliva-Istra�iva�ki institut d.o.o.	N"-Substituted 9a-N-(N'-carbamoyl-Gamma-aminopropyl), 9a-N-(N'? -thiocarbamoyl-Gamma-aminopropyl), 9a-N-(N'-((Beta-cyanoethyl)-N'-carbamoyl-Gamma? -aminopropyl) and 9a-N-(N'-(Beta-cyanoethyl)-N'-thiocarbamoyl-Gamma? -aminopropyl) derivatives of 9-de
EP1835921B1 (de) *	2005-01-14	2010-08-18	GlaxoSmithKline istrazivacki centar Zagreb d.o.o.	9a-carbamoyl-y-aminopropyl- und 9a-thiocarbamoyl-y-aminopropyl-azalide mit antimalaria-aktivität

2006
- 2006-01-13 ES ES06727593T patent/ES2344518T3/es not_active Expired - Lifetime
- 2006-01-13 US US11/813,875 patent/US20080200404A1/en not_active Abandoned
- 2006-01-13 JP JP2007550878A patent/JP2008526949A/ja not_active Withdrawn
- 2006-01-13 EP EP06727593A patent/EP1855696B1/de not_active Expired - Lifetime
- 2006-01-13 AT AT06727593T patent/ATE465741T1/de not_active IP Right Cessation
- 2006-01-13 WO PCT/IB2006/001227 patent/WO2006085228A2/en not_active Ceased
- 2006-01-13 DE DE602006013953T patent/DE602006013953D1/de not_active Expired - Lifetime

Also Published As

Publication number	Publication date
US20080200404A1 (en)	2008-08-21
WO2006085228A2 (en)	2006-08-17
JP2008526949A (ja)	2008-07-24
EP1855696A2 (de)	2007-11-21
WO2006085228A3 (en)	2007-01-04
DE602006013953D1 (de)	2010-06-10
ES2344518T3 (es)	2010-08-30
EP1855696B1 (de)	2010-04-28

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Legal Events

Date	Code	Title	Description
2010-10-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties