ATE467616T1 - Verbindungen mit aktivität an der 11beta- hydroxasteroiddehydrogenase - Google Patents

Verbindungen mit aktivität an der 11beta- hydroxasteroiddehydrogenase

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Publication number
ATE467616T1
ATE467616T1 AT07102177T AT07102177T ATE467616T1 AT E467616 T1 ATE467616 T1 AT E467616T1 AT 07102177 T AT07102177 T AT 07102177T AT 07102177 T AT07102177 T AT 07102177T AT E467616 T1 ATE467616 T1 AT E467616T1
Authority
AT
Austria
Prior art keywords
compounds
activity
hydroxasteroid
11beta
dehydrogenase
Prior art date
Application number
AT07102177T
Other languages
English (en)
Inventor
Anette Gundertofte
Anker Steen Jorgensen
Gita Camilla Tejlgaard Kampen
Henrik Sune Andersen
Inge Thoger Christensen
John Paul Kilburn
Original Assignee
High Point Pharmaceuticals Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by High Point Pharmaceuticals Llc filed Critical High Point Pharmaceuticals Llc
Application granted granted Critical
Publication of ATE467616T1 publication Critical patent/ATE467616T1/de

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
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    • A61K31/16—Amides, e.g. hydroxamic acids
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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WO2004089896A1 (en) 2004-10-21
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EP1615698A2 (de) 2006-01-18
JP2006522748A (ja) 2006-10-05
JP4629657B2 (ja) 2011-02-09
US20090264414A1 (en) 2009-10-22
EP1787982A3 (de) 2007-05-30
EP1787982B1 (de) 2010-05-12
EP2239012A2 (de) 2010-10-13
EP1618090A1 (de) 2006-01-25
ATE482747T1 (de) 2010-10-15
JP2006522746A (ja) 2006-10-05
EP2239012A3 (de) 2011-06-15
DE602004027171D1 (de) 2010-06-24
EP1615698B1 (de) 2010-09-29

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