ATE501147T1 - Dipeptidylpeptidase-iv-inhibitoren auf azolopyrimidinbasis und verfahren - Google Patents

Dipeptidylpeptidase-iv-inhibitoren auf azolopyrimidinbasis und verfahren

Info

Publication number
ATE501147T1
ATE501147T1 AT05855291T AT05855291T ATE501147T1 AT E501147 T1 ATE501147 T1 AT E501147T1 AT 05855291 T AT05855291 T AT 05855291T AT 05855291 T AT05855291 T AT 05855291T AT E501147 T1 ATE501147 T1 AT E501147T1
Authority
AT
Austria
Prior art keywords
azolopyrimidine
dipeptidylpeptidase
inhibitors
methods
based dipeptidylpeptidase
Prior art date
Application number
AT05855291T
Other languages
English (en)
Inventor
Wei Meng
Lawrence G Hamann
Robert Paul Brigance
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Application granted granted Critical
Publication of ATE501147T1 publication Critical patent/ATE501147T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Hematology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Obesity (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AT05855291T 2004-12-29 2005-12-23 Dipeptidylpeptidase-iv-inhibitoren auf azolopyrimidinbasis und verfahren ATE501147T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US64013504P 2004-12-29 2004-12-29
PCT/US2005/046706 WO2006071752A1 (en) 2004-12-29 2005-12-23 Azolopyrimidine-based inhibitors of dipeptidyl peptidase iv and methods

Publications (1)

Publication Number Publication Date
ATE501147T1 true ATE501147T1 (de) 2011-03-15

Family

ID=36177846

Family Applications (1)

Application Number Title Priority Date Filing Date
AT05855291T ATE501147T1 (de) 2004-12-29 2005-12-23 Dipeptidylpeptidase-iv-inhibitoren auf azolopyrimidinbasis und verfahren

Country Status (9)

Country Link
US (1) US7635699B2 (de)
EP (1) EP1836206B1 (de)
AR (1) AR052658A1 (de)
AT (1) ATE501147T1 (de)
DE (1) DE602005026864D1 (de)
ES (1) ES2360937T3 (de)
PE (1) PE20060835A1 (de)
TW (1) TW200634018A (de)
WO (1) WO2006071752A1 (de)

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Also Published As

Publication number Publication date
TW200634018A (en) 2006-10-01
DE602005026864D1 (de) 2011-04-21
AR052658A1 (es) 2007-03-28
ES2360937T3 (es) 2011-06-10
PE20060835A1 (es) 2006-08-23
WO2006071752A1 (en) 2006-07-06
US7635699B2 (en) 2009-12-22
US20060178377A1 (en) 2006-08-10
EP1836206A1 (de) 2007-09-26
EP1836206B1 (de) 2011-03-09

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