ATE502930T1 - Antibakterielle mittel - Google Patents
Antibakterielle mittelInfo
- Publication number
- ATE502930T1 ATE502930T1 AT08806355T AT08806355T ATE502930T1 AT E502930 T1 ATE502930 T1 AT E502930T1 AT 08806355 T AT08806355 T AT 08806355T AT 08806355 T AT08806355 T AT 08806355T AT E502930 T1 ATE502930 T1 AT E502930T1
- Authority
- AT
- Austria
- Prior art keywords
- radical
- hydrogen
- antibacterial agents
- optionally substituted
- ring atoms
- Prior art date
Links
- 239000003242 anti bacterial agent Substances 0.000 title 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- 125000006413 ring segment Chemical group 0.000 abstract 2
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 1
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 abstract 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- CIUQDSCDWFSTQR-UHFFFAOYSA-N [C]1=CC=CC=C1 Chemical compound [C]1=CC=CC=C1 CIUQDSCDWFSTQR-UHFFFAOYSA-N 0.000 abstract 1
- 230000000844 anti-bacterial effect Effects 0.000 abstract 1
- 125000001309 chloro group Chemical group Cl* 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000001153 fluoro group Chemical group F* 0.000 abstract 1
- 150000002431 hydrogen Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/08—1,2,4-Thiadiazoles; Hydrogenated 1,2,4-thiadiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0718335.3A GB0718335D0 (en) | 2007-09-20 | 2007-09-20 | Antibacterial agents |
| PCT/GB2008/003200 WO2009037485A1 (en) | 2007-09-20 | 2008-09-22 | Antibacterial agents |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE502930T1 true ATE502930T1 (de) | 2011-04-15 |
Family
ID=38670209
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT08806355T ATE502930T1 (de) | 2007-09-20 | 2008-09-22 | Antibakterielle mittel |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US8492414B2 (de) |
| EP (1) | EP2200991B1 (de) |
| AT (1) | ATE502930T1 (de) |
| DE (1) | DE602008005777D1 (de) |
| ES (1) | ES2364959T3 (de) |
| GB (1) | GB0718335D0 (de) |
| WO (1) | WO2009037485A1 (de) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5996532B2 (ja) | 2010-07-15 | 2016-09-21 | バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングBayer Intellectual Property GmbH | 有害生物防除剤としての新規複素環式化合物 |
| WO2012142671A1 (en) | 2011-04-20 | 2012-10-26 | Biota Scientific Management Pty Ltd | Aromatic amides and uses thereof |
| CN102276554B (zh) * | 2011-06-28 | 2013-10-30 | 四川大学 | 4-((2-氨基-5-巯基-1,3,4-噻二唑)-甲基)-苯甲酰胺衍生物及其制备方法和用途 |
| US9282738B2 (en) | 2011-07-11 | 2016-03-15 | Wisconsin Alumni Research Foundation | Antimicrobial compositions and methods of use thereof |
| US9822108B2 (en) | 2012-01-13 | 2017-11-21 | Rutgers, The State University Of New Jersey | Antimicrobial agents |
| US9475783B2 (en) | 2012-03-21 | 2016-10-25 | Rutgers, The State University Of New Jersey | Antimicrobial agents |
| US9458150B2 (en) | 2013-11-08 | 2016-10-04 | Rutgers, The State University Of New Jersey | Antimicrobial agents |
| WO2015179697A1 (en) | 2014-05-21 | 2015-11-26 | Taxis Pharmaceuticals, Inc. | Compounds for the treatment of bacterial infections |
| WO2017147316A1 (en) | 2016-02-25 | 2017-08-31 | Taxis Pharmaceuticals, Inc. | Synthetic processes and intermediates |
| US10774093B2 (en) | 2017-03-30 | 2020-09-15 | Taxis Pharmaceuticals, Inc. | Synthetic processes and synthetic intermediates |
| CN112341506B (zh) * | 2020-11-11 | 2022-05-06 | 铜仁学院 | 乙酰葡萄糖噻二唑苯甲酰胺类化合物及其合成方法和应用 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2003220935A1 (en) | 2002-04-03 | 2003-10-13 | Sumitomo Pharmaceuticals Company, Limited. | Benzamide derivatives |
| WO2007107758A1 (en) | 2006-03-23 | 2007-09-27 | Prolysis Ltd | Antibacterial agents |
-
2007
- 2007-09-20 GB GBGB0718335.3A patent/GB0718335D0/en not_active Ceased
-
2008
- 2008-09-22 DE DE200860005777 patent/DE602008005777D1/de active Active
- 2008-09-22 EP EP20080806355 patent/EP2200991B1/de not_active Not-in-force
- 2008-09-22 US US12/678,767 patent/US8492414B2/en active Active
- 2008-09-22 ES ES08806355T patent/ES2364959T3/es active Active
- 2008-09-22 WO PCT/GB2008/003200 patent/WO2009037485A1/en not_active Ceased
- 2008-09-22 AT AT08806355T patent/ATE502930T1/de not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| DE602008005777D1 (de) | 2011-05-05 |
| ES2364959T3 (es) | 2011-09-19 |
| EP2200991B1 (de) | 2011-03-23 |
| GB0718335D0 (en) | 2007-10-31 |
| US20100273837A1 (en) | 2010-10-28 |
| EP2200991A1 (de) | 2010-06-30 |
| US8492414B2 (en) | 2013-07-23 |
| WO2009037485A1 (en) | 2009-03-26 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| ATE502930T1 (de) | Antibakterielle mittel | |
| CR20140392A (es) | Dihidropirazolonas sustituidas | |
| CY1111481T1 (el) | Υποκατεστημενα αρυλοκυκλοπροπυλακεταμιδια ως ενεργοποιητες γλυκοκινασης | |
| PE20081888A1 (es) | ANALOGOS DE PIRAZOLOPIRIMIDINA Y SU USO COMO INHIBIDORES DE CINASA mTOR Y CINASA PI3 | |
| MX2017010735A (es) | Inhibidores de inhibidores del factor beta de crecimiento de transformacion (tgf-beta). | |
| MD4582B1 (ro) | Derivaţi ai 1-fenil-1H-benzimidazolului ca inhibitori ai protein kinazei | |
| PE20211782A1 (es) | Compuestos de 5-cloro-2-difluorometoxifenil pirazolopirimidina, composiciones y metodos de uso de los mismos | |
| EA201200049A1 (ru) | 1,3-дизамещенные производные имидазолидин-2-она в качестве ингибиторов cyp 17 | |
| PH12017501192A1 (en) | Certain amino-pyridazines, compositions thereof, and methods of their use | |
| NO20090313L (no) | Derivater og analoger av N-etylkinoloner og N-etylazakinoloner | |
| NO20092710L (no) | Cyclopaminanaloger | |
| EA200970207A1 (ru) | Соединения пиридо[2,3-d]пиримидинона и их применение в качестве pi3 ингибиторов | |
| MX377581B (es) | Compuestos antihelmínticos y composiciones y método de uso de los mismos. | |
| CR20140294A (es) | Derivados de dihidro-benzo-oxazina y dihidro-pirido-oxazina | |
| CR20120348A (es) | Nuevos compuestos tricíclicos | |
| UY31545A1 (es) | Nuevos derivados de 2-carboxamida cianoaminourea, sus sales y profarmacos farmacéuticamente aceptables, procesos de preparacion y aplicaciones | |
| MX2013005826A (es) | Benzoxazepinas como inhibidores de fosfatidilinositol 3-cinasa/objetivo de rapamicina en mamiferos (p13k/mtor) y metodos de uso y fabricacion. | |
| EA201000113A1 (ru) | Пиразольные соединения | |
| EA201201378A1 (ru) | Определенные аминопиримидины, композиции на их основе и способы их использования | |
| MA35434B1 (fr) | Amino-quinazolines en tant qu'inhibiteurs de kinase | |
| EA200900924A1 (ru) | Циклизованные производные как ингибиторы eg-5 | |
| MA39866A (fr) | Amides 2-amino-6-méthyl-4,4a,5,6-tétrahydropyrano[3,4-d][1,3]thiazin-8a(8h)-yl-1,3-thiazol-4-yle | |
| MX375153B (es) | Compuestos antihelminticos. | |
| WO2011038234A3 (en) | Novel iodo pyrimidine derivatives useful for the treatment of macrophage migration inhibitory factor (mif)-implicated diseases and conditions | |
| ECSP109964A (es) | Pirimidinas bicíclicas fusionadas |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |