ATE516011T1 - Pharmazeutische zusammensetzungen eines a2a rezeptorantagonisten - Google Patents
Pharmazeutische zusammensetzungen eines a2a rezeptorantagonistenInfo
- Publication number
- ATE516011T1 ATE516011T1 AT04814759T AT04814759T ATE516011T1 AT E516011 T1 ATE516011 T1 AT E516011T1 AT 04814759 T AT04814759 T AT 04814759T AT 04814759 T AT04814759 T AT 04814759T AT E516011 T1 ATE516011 T1 AT E516011T1
- Authority
- AT
- Austria
- Prior art keywords
- pharmaceutical compositions
- receptor antagonist
- disclosed
- antagonist
- receptor
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 229940127600 A2A receptor antagonist Drugs 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
- A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4166—1,3-Diazoles having oxo groups directly attached to the heterocyclic ring, e.g. phenytoin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4858—Organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
- C07D487/14—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Psychiatry (AREA)
- Psychology (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US53156103P | 2003-12-19 | 2003-12-19 | |
| PCT/US2004/042616 WO2005060981A2 (en) | 2003-12-19 | 2004-12-17 | Pharmaceutical compositions |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE516011T1 true ATE516011T1 (de) | 2011-07-15 |
Family
ID=34710234
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT04814759T ATE516011T1 (de) | 2003-12-19 | 2004-12-17 | Pharmazeutische zusammensetzungen eines a2a rezeptorantagonisten |
Country Status (15)
| Country | Link |
|---|---|
| US (3) | US20060009504A1 (de) |
| EP (1) | EP1701699B1 (de) |
| JP (1) | JP2007514758A (de) |
| KR (1) | KR20060111581A (de) |
| CN (1) | CN100528162C (de) |
| AT (1) | ATE516011T1 (de) |
| AU (1) | AU2004303425C1 (de) |
| BR (1) | BRPI0417205A (de) |
| CA (1) | CA2550071A1 (de) |
| MX (1) | MXPA06007102A (de) |
| NO (1) | NO20063293L (de) |
| NZ (1) | NZ547557A (de) |
| PL (1) | PL380665A1 (de) |
| WO (1) | WO2005060981A2 (de) |
| ZA (1) | ZA200604874B (de) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL2368554T3 (pl) | 2003-04-08 | 2015-05-29 | Progenics Pharm Inc | Preparaty farmaceutyczne zawierające metylonaltrekson |
| TWI489984B (zh) | 2006-08-04 | 2015-07-01 | Wyeth Corp | 用於非經腸道傳輸化合物之配方及其用途 |
| US20090041839A1 (en) * | 2007-05-23 | 2009-02-12 | Beasley Martin W | Pharmaceutical compositions for the treatment of pain |
| SE531698C2 (sv) | 2007-07-12 | 2009-07-07 | Respiratorius Ab | Nya bronkdilaterande a,b-omättade amider |
| TWI605814B (zh) | 2010-03-11 | 2017-11-21 | 惠氏有限責任公司 | 甲基拿淬松（ｍｅｔｈｙｌｎａｌｔｒｅｘｏｎｅ）之口服製劑及親脂性鹽 |
| WO2012127472A1 (en) * | 2011-03-22 | 2012-09-27 | Mapi Pharma Ltd. | Process and intermediates for the preparation of preladenant and related compounds |
| CN106365221B (zh) * | 2016-11-09 | 2019-04-19 | 烟台史密得机电设备制造有限公司 | 一种金刚烷单季铵盐阳离子型三元复合驱采出水除油剂 |
| WO2018204872A2 (en) | 2017-05-05 | 2018-11-08 | Fusion Pharmaceuticals Inc. | Igf-1r monoclonal antibodies and uses thereof |
| US10093741B1 (en) | 2017-05-05 | 2018-10-09 | Fusion Pharmaceuticals Inc. | IGF-1R monoclonal antibodies and uses thereof |
| AU2018261888B2 (en) | 2017-05-05 | 2022-06-30 | Centre For Probe Development And Commercialization | Pharmacokinetic enhancements of bifunctional chelates and uses thereof |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4656028A (en) * | 1986-06-24 | 1987-04-07 | Norcliff Thayer Inc. | Encapsulated antacid |
| US5935584A (en) * | 1994-01-13 | 1999-08-10 | Elizabeth Arden Company | Vitamin C delivery system |
| PT901786E (pt) * | 1997-08-11 | 2007-08-07 | Pfizer Prod Inc | Disperções farmacêuticas sólidas com biodisponibilidade melhorada |
| US6326390B1 (en) * | 1998-08-25 | 2001-12-04 | King Pharmaceuticals Reseach And Development, Inc. | Use of adenosine A3 receptor antagonists to inhibit tumor growth |
| US6921825B2 (en) * | 1998-09-16 | 2005-07-26 | King Pharmaceuticuals Research & Development, Inc. | Adenosine A3 receptor modulators |
| US6448253B1 (en) * | 1998-09-16 | 2002-09-10 | King Pharmaceuticals Research And Development, Inc. | Adenosine A3 receptor modulators |
| US6383471B1 (en) * | 1999-04-06 | 2002-05-07 | Lipocine, Inc. | Compositions and methods for improved delivery of ionizable hydrophobic therapeutic agents |
| KR20070058028A (ko) * | 1999-05-24 | 2007-06-07 | 소너스파머슈티칼즈인코포레이티드 | 난용성 약물용 에멀젼 부형제 |
| JP4100865B2 (ja) * | 1999-12-13 | 2008-06-11 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | 三環式縮合異項環化合物、その製造法およびその医薬 |
| PT1283839E (pt) * | 2000-05-26 | 2005-08-31 | Schering Corp | Antagonistas do receptor a2a da adenosina |
| JP4545437B2 (ja) * | 2001-10-15 | 2010-09-15 | シェーリング コーポレイション | アデノシンａ２ａ受容体アンタゴニストとしてのイミダゾ（４，３−ｅ）−１，２，４−トリアゾロ（１，５−ｃ）ピリミジン |
| AU2002346503A1 (en) * | 2001-11-30 | 2003-06-17 | Schering Corporation | Adenosine A2a receptor antagonists |
| MXPA04000908A (es) * | 2002-05-30 | 2004-03-26 | King Pharmaceuticals Res & Dev | Compuestos farmaceuticamente activos que tienen estructura de anillo de pirazolotriazolopirimidina triciclica y metodos de uso. |
| US6982253B2 (en) * | 2002-06-05 | 2006-01-03 | Supergen, Inc. | Liquid formulation of decitabine and use of the same |
-
2004
- 2004-12-17 CA CA002550071A patent/CA2550071A1/en not_active Abandoned
- 2004-12-17 AT AT04814759T patent/ATE516011T1/de not_active IP Right Cessation
- 2004-12-17 AU AU2004303425A patent/AU2004303425C1/en not_active Ceased
- 2004-12-17 KR KR1020067011952A patent/KR20060111581A/ko not_active Ceased
- 2004-12-17 NZ NZ547557A patent/NZ547557A/en not_active IP Right Cessation
- 2004-12-17 PL PL380665A patent/PL380665A1/pl not_active Application Discontinuation
- 2004-12-17 CN CNB2004800375628A patent/CN100528162C/zh not_active Expired - Fee Related
- 2004-12-17 MX MXPA06007102A patent/MXPA06007102A/es active IP Right Grant
- 2004-12-17 EP EP04814759A patent/EP1701699B1/de not_active Expired - Lifetime
- 2004-12-17 BR BRPI0417205-1A patent/BRPI0417205A/pt not_active IP Right Cessation
- 2004-12-17 US US11/015,946 patent/US20060009504A1/en not_active Abandoned
- 2004-12-17 WO PCT/US2004/042616 patent/WO2005060981A2/en not_active Ceased
- 2004-12-17 JP JP2006545514A patent/JP2007514758A/ja active Pending
-
2006
- 2006-06-13 ZA ZA200604874A patent/ZA200604874B/xx unknown
- 2006-07-14 NO NO20063293A patent/NO20063293L/no not_active Application Discontinuation
-
2008
- 2008-08-05 US US12/186,002 patent/US20080293734A1/en not_active Abandoned
-
2011
- 2011-04-04 US US13/079,378 patent/US20110207740A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO2005060981A3 (en) | 2005-12-29 |
| AU2004303425C1 (en) | 2010-02-18 |
| EP1701699B1 (de) | 2011-07-13 |
| KR20060111581A (ko) | 2006-10-27 |
| CN1893921A (zh) | 2007-01-10 |
| MXPA06007102A (es) | 2006-08-23 |
| EP1701699A2 (de) | 2006-09-20 |
| NZ547557A (en) | 2010-07-30 |
| US20080293734A1 (en) | 2008-11-27 |
| US20110207740A1 (en) | 2011-08-25 |
| PL380665A1 (pl) | 2007-03-05 |
| US20060009504A1 (en) | 2006-01-12 |
| WO2005060981A2 (en) | 2005-07-07 |
| CN100528162C (zh) | 2009-08-19 |
| AU2004303425B2 (en) | 2009-03-26 |
| NO20063293L (no) | 2006-07-14 |
| AU2004303425A1 (en) | 2005-07-07 |
| JP2007514758A (ja) | 2007-06-07 |
| ZA200604874B (en) | 2007-03-28 |
| BRPI0417205A (pt) | 2007-02-06 |
| CA2550071A1 (en) | 2005-07-07 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |