ATE525110T1 - Inverse emulsionszusammensetzung mit ivermectin und verwendung davon in der kosmetik und in der dermatologie - Google Patents

Inverse emulsionszusammensetzung mit ivermectin und verwendung davon in der kosmetik und in der dermatologie

Info

Publication number: ATE525110T1
Authority: AT; Austria
Prior art keywords: ivermectin; dermatology; cosmetics; emulsion composition; inverse emulsion
Prior art date: 2005-12-20

Application number

AT06847168T

Other languages

English (en)

Inventor

Sandrine Segura-Orsoni

Fanny Diaz-Astruc

Original Assignee

Galderma Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2005-12-20

Filing date

2006-12-18

Publication date

2011-10-15

2006-12-18 Application filed by Galderma Sa filed Critical Galderma Sa

2011-10-15 Application granted granted Critical

2011-10-15 Publication of ATE525110T1 publication Critical patent/ATE525110T1/de

Links

AZSNMRSAGSSBNP-UHFFFAOYSA-N 22,23-dihydroavermectin B1a Natural products C1CC(C)C(C(C)CC)OC21OC(CC=C(C)C(OC1OC(C)C(OC3OC(C)C(O)C(OC)C3)C(OC)C1)C(C)C=CC=C1C3(C(C(=O)O4)C=C(C)C(O)C3OC1)O)CC4C2 AZSNMRSAGSSBNP-UHFFFAOYSA-N 0.000 title abstract 2
239000002537 cosmetic Substances 0.000 title abstract 2
239000000839 emulsion Substances 0.000 title abstract 2
229960002418 ivermectin Drugs 0.000 title abstract 2
AZSNMRSAGSSBNP-XPNPUAGNSA-N 22,23-dihydroavermectin B1a Chemical compound C1C[C@H](C)[C@@H]([C@@H](C)CC)O[C@@]21O[C@H](C\C=C(C)\[C@@H](O[C@@H]1O[C@@H](C)[C@H](O[C@@H]3O[C@@H](C)[C@H](O)[C@@H](OC)C3)[C@@H](OC)C1)[C@@H](C)\C=C\C=C/1[C@]3([C@H](C(=O)O4)C=C(C)[C@@H](O)[C@H]3OC\1)O)C[C@H]4C2 AZSNMRSAGSSBNP-XPNPUAGNSA-N 0.000 title 1
238000003874 inverse correlation nuclear magnetic resonance spectroscopy Methods 0.000 title 1
239000000203 mixture Substances 0.000 title 1
SPBDXSGPUHCETR-JFUDTMANSA-N 8883yp2r6d Chemical compound O1[C@@H](C)[C@H](O)[C@@H](OC)C[C@@H]1O[C@@H]1[C@@H](OC)C[C@H](O[C@@H]2C(=C/C[C@@H]3C[C@@H](C[C@@]4(O[C@@H]([C@@H](C)CC4)C(C)C)O3)OC(=O)[C@@H]3C=C(C)[C@@H](O)[C@H]4OC\C([C@@]34O)=C/C=C/[C@@H]2C)/C)O[C@H]1C.C1C[C@H](C)[C@@H]([C@@H](C)CC)O[C@@]21O[C@H](C\C=C(C)\[C@@H](O[C@@H]1O[C@@H](C)[C@H](O[C@@H]3O[C@@H](C)[C@H](O)[C@@H](OC)C3)[C@@H](OC)C1)[C@@H](C)\C=C\C=C/1[C@]3([C@H](C(=O)O4)C=C(C)[C@@H](O)[C@H]3OC\1)O)C[C@H]4C2 SPBDXSGPUHCETR-JFUDTMANSA-N 0.000 abstract 1
239000005660 Abamectin Substances 0.000 abstract 1
241001303601 Rosacea Species 0.000 abstract 1
-1 avermectin compound Chemical class 0.000 abstract 1
239000003995 emulsifying agent Substances 0.000 abstract 1
230000003647 oxidation Effects 0.000 abstract 1
238000007254 oxidation reaction Methods 0.000 abstract 1
201000004700 rosacea Diseases 0.000 abstract 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/24—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing atoms other than carbon, hydrogen, oxygen, halogen, nitrogen or sulfur, e.g. cyclomethicone or phospholipids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/32—Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0014—Skin, i.e. galenical aspects of topical compositions
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/10—Anti-acne agents

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Epidemiology (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Oil, Petroleum & Natural Gas (AREA)
Dermatology (AREA)
Molecular Biology (AREA)
Biophysics (AREA)
Dispersion Chemistry (AREA)
Inorganic Chemistry (AREA)
Bioinformatics & Cheminformatics (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Medicinal Preparation (AREA)
Cosmetics (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

AT06847168T 2005-12-20 2006-12-18 Inverse emulsionszusammensetzung mit ivermectin und verwendung davon in der kosmetik und in der dermatologie ATE525110T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR0512956A FR2894823B1 (fr)	2005-12-20	2005-12-20	Composition de type emulsion inverse comprenant de l'ivermectine, et ses utilisations en cosmetique et en dermatologie
PCT/FR2006/051378 WO2007071876A1 (fr)	2005-12-20	2006-12-18	Composition de type emulsion inverse comprenant de l'ivermectine, et ses utilisations en cosmetique et en dermatologie

Publications (1)

Publication Number	Publication Date
ATE525110T1 true ATE525110T1 (de)	2011-10-15

Family

ID=36215627

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT06847168T ATE525110T1 (de)	2005-12-20	2006-12-18	Inverse emulsionszusammensetzung mit ivermectin und verwendung davon in der kosmetik und in der dermatologie

Country Status (8)

Country	Link
US (1)	US8287891B2 (de)
EP (1)	EP1965864B1 (de)
AT (1)	ATE525110T1 (de)
BR (1)	BRPI0621115A2 (de)
CA (1)	CA2633040C (de)
ES (1)	ES2370912T3 (de)
FR (1)	FR2894823B1 (de)
WO (1)	WO2007071876A1 (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US9782425B2 (en)	2013-07-08	2017-10-10	Galderma S.A.	Treatment of papulopustular rosacea with ivermectin
US9233117B2 (en)	2013-07-08	2016-01-12	Galderma S. A.	Treatment of inflammatory lesions of rosacea with ivermectin
WO2017064205A1 (en) *	2015-10-13	2017-04-20	Galderma Sa	A process for preparing a stable emulsion comprising one or more avermectins
EP3362045B1 (de)	2015-10-13	2019-10-09	Galderma S.A.	Verfahren zur herstellung einer zusammensetzung mit einer hohen konzentration an einem oder mehreren avermectinen
EP3326609A1 (de) *	2016-11-24	2018-05-30	Nestlé Skin Health SA	Zusammensetzung mit avermectinverbindungen ohne geliermittel
EP3326614A1 (de)	2016-11-24	2018-05-30	Nestlé Skin Health SA	Zusammensetzung mit avermectinverbindungen ohne lösungsmittel und propenetrationsmittel aus avermectinverbindungen
EP3326608A1 (de) *	2016-11-24	2018-05-30	Nestlé Skin Health SA	Zusammensetzung mit avermectinverbindungen ohne feste fettsubstanzen
US11554086B2 (en)	2017-12-29	2023-01-17	L'oreal	Cosmetic composition comprising glycolic acid and methods of use

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4389397A (en) *	1980-08-04	1983-06-21	Merck & Co., Inc.	Solubilization of ivermectin in water
NZ197796A (en) *	1980-08-04	1984-11-09	Merck & Co Inc	Stabilised aqueous formulations containing ivermectin
US4675575A (en) *	1984-07-13	1987-06-23	E & G Enterprises	Light-emitting diode assemblies and systems therefore
US5952372A (en) *	1998-09-17	1999-09-14	Mcdaniel; William Robert	Method for treating rosacea using oral or topical ivermectin
US6133310A (en)	1999-08-26	2000-10-17	Parks; L. Dean	Method of treatment of rosacea
US6399652B1 (en) *	2000-06-29	2002-06-04	L. Dean Parks	Method of treating acne vulgaris using avermectin compound
US6319945B1 (en) *	2000-06-29	2001-11-20	L. Dean Parks	Method of treatment of seborrheic dermatitis
US7897559B2 (en) *	2000-06-29	2011-03-01	Parks L Dean	Dermatological composition and kit containing avermectin compound for treating dermatological conditions
US20030064940A1 (en) *	2001-10-02	2003-04-03	Parks L. Dean	Kit for treating acne vulgaris using avermectin compound
US6399651B1 (en) *	2000-06-29	2002-06-04	L. Dean Parks	Method of treating dermatoses using avermectin compound
AUPQ875700A0 (en) *	2000-07-13	2000-08-03	Reflex Research Limited	Combination compositions
FI118404B (fi) *	2001-11-27	2007-10-31	Pulse Finland Oy	Kaksoisantenni ja radiolaite
US7122961B1 (en) *	2002-05-21	2006-10-17	Imaging Systems Technology	Positive column tubular PDP
KR100436766B1 (ko) *	2002-07-19	2004-06-23	삼성광주전자 주식회사	왕복동식 압축기
CN1685090A (zh) *	2002-09-20	2005-10-19	三菱化学株式会社	Ⅲ－v化合物半导体晶体
WO2004093886A1 (en) *	2003-04-24	2004-11-04	Galderma S.A.	Topical formulation of ivermectin for the treatment of dermatological conditions
FR2867684B1 (fr) *	2004-03-18	2006-05-05	Galderma Sa	Gel creme contenant de l'ivermectine
DE602005020912D1 (de) *	2004-03-18	2010-06-10	Galderma Sa	Ivermectin enthaltende creme
US7144131B2 (en) *	2004-09-29	2006-12-05	Advanced Optical Technologies, Llc	Optical system using LED coupled with phosphor-doped reflective materials

2005
- 2005-12-20 FR FR0512956A patent/FR2894823B1/fr not_active Expired - Fee Related
2006
- 2006-12-18 BR BRPI0621115-1A patent/BRPI0621115A2/pt not_active IP Right Cessation
- 2006-12-18 ES ES06847168T patent/ES2370912T3/es active Active
- 2006-12-18 AT AT06847168T patent/ATE525110T1/de not_active IP Right Cessation
- 2006-12-18 WO PCT/FR2006/051378 patent/WO2007071876A1/fr not_active Ceased
- 2006-12-18 EP EP06847168A patent/EP1965864B1/de not_active Not-in-force
- 2006-12-18 CA CA2633040A patent/CA2633040C/fr not_active Expired - Fee Related
2008
- 2008-06-20 US US12/213,554 patent/US8287891B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
BRPI0621115A2 (pt)	2011-11-29
US20090035338A1 (en)	2009-02-05
US8287891B2 (en)	2012-10-16
FR2894823B1 (fr)	2008-02-29
CA2633040A1 (fr)	2007-06-28
EP1965864A1 (de)	2008-09-10
CA2633040C (fr)	2014-09-16
EP1965864B1 (de)	2011-09-21
FR2894823A1 (fr)	2007-06-22
ES2370912T3 (es)	2011-12-23
WO2007071876A1 (fr)	2007-06-28

Legal Events

Date	Code	Title	Description
2012-03-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties

Publication	Publication Date	Title
AR044050A1 (es)	2005-08-24	Utilizacion de ivermectina para el tratamiento de desordenes dermatologicos
BR0100335A (pt)	2001-10-09	Nanoemulsão óleo-em-água à base de lipìdios anfìfilos e de polìmeros catiÈnicos, composição cosmética de uso tópico, utilizações, processo de tratamento não-terapêutico e processo para espessar as nanoemulsões óleo-em-água
BRPI0409997A (pt)	2006-05-09	composições para tratamento de pele molhada compreendendo redes de gel
MXPA05011208A (es)	2005-12-14	Uso de ivermectina para el tratamiento de desordenes dermatologicos.
BRPI0407969A (pt)	2006-03-07	composição de microemulsão, e, métodos para o tratamento de plantas com um produto agroquìmico e para a produção de preparações pontas para uso contendo produtos agroquìmicos
BRPI0918878B8 (pt)	2017-06-13	composição cosmética ou dermatológica e processo de tratamento cosmético da pele, dos cabelos e/ou dos lábios
BRPI0411306A (pt)	2006-07-11	composições farmacêuticas compreendendo compostos ativos de vitamina d
AR046824A1 (es)	2005-12-28	Composicion y aparato para la administracion transdermica.
BRPI0409516A (pt)	2006-04-18	composição, uso de uma composição e processo de melhora da penetração de um ativo farmacêutico
WO2007106284A3 (en)	2008-06-26	Silicone based emulsions for topical drug delivery
FR2789076B1 (fr)	2001-03-02	Derives de alpha-azacyclomethyl quinoleine, leur preparation et leur application en therapeutique
ATE269047T1 (de)	2004-07-15	Emulgatorfreie und bornitrid enthaltende feindisperse systeme vom typ öl-in-wasser und wasser-in-öl
BRPI0510893A (pt)	2007-11-27	composição, composição cosmética ou dermatológica, processo de preparação de uma composição e uso de uma composição
ATE356606T1 (de)	2007-04-15	Juckreizstillende kosmetische und dermatologische zubereitungen
EP1544406A3 (de)	2007-09-05	Kolloid oder- kolloidartige-Systemen für wässerige tonenthaltende Spülungen
BRPI0416311A (pt)	2006-12-26	composição, uso de uma composição e processo para melhorar a penetração de um agente ativo farmacêutico
ATE525110T1 (de)	2011-10-15	Inverse emulsionszusammensetzung mit ivermectin und verwendung davon in der kosmetik und in der dermatologie
ATE253820T1 (de)	2003-11-15	Wirkstoffhaltige komposition sowie deren herstellung und verwendung
BRPI0909296A2 (pt)	2016-06-21	uso de pelo menos um princípio ativo, e, composições cosmética, farmacêutica e/ou dermatológica
BRPI0406490A (pt)	2005-12-06	Composições, composição cosmética ou dermatológica e uso de uma composição
WO2002024152A3 (en)	2002-07-25	Oil in glycerin emulsion
ATE328571T1 (de)	2006-06-15	Emulgatorfreie feindisperse systeme vom typ wasser-in-öl
NZ589971A (en)	2013-01-25	Emollient composition comprising glycerol, vaseline and liquid paraffin
ATE423186T1 (de)	2009-03-15	Emulsion
BR0211735A (pt)	2004-09-21	Composições, composição cosmética ou dermatológica, uso cosmético de uma composição e uso de uma composição