ATE528312T1 - METHOD FOR SYNTHESIS OF MACROLIDS - Google Patents

METHOD FOR SYNTHESIS OF MACROLIDS

Info

Publication number
ATE528312T1
ATE528312T1 AT07787934T AT07787934T ATE528312T1 AT E528312 T1 ATE528312 T1 AT E528312T1 AT 07787934 T AT07787934 T AT 07787934T AT 07787934 T AT07787934 T AT 07787934T AT E528312 T1 ATE528312 T1 AT E528312T1
Authority
AT
Austria
Prior art keywords
macrolides
making
macrolids
synthesis
methods
Prior art date
Application number
AT07787934T
Other languages
German (de)
Inventor
Fritz Blatter
Meinrad Brenner
Monika Brink
Kerstin Fleischhauer
Guixian Hu
Hans Peter Niedermann
Timo Rager
Tanja Schweisel
Stephan Veit
Ralf Warrass
Heinz-Joerg Wennesheimer
Original Assignee
Intervet Int Bv
Microbial Chem Res Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Intervet Int Bv, Microbial Chem Res Found filed Critical Intervet Int Bv
Priority claimed from PCT/EP2007/057710 external-priority patent/WO2008012343A2/en
Application granted granted Critical
Publication of ATE528312T1 publication Critical patent/ATE528312T1/en

Links

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

This invention relates to a method for making macrolides, and, in particular, to a method for making optionally substituted 20, 23-dipiperidinyl-5-O-mycaminosyl-tylonolide and derivatives thereof, as well as uses of macrolides to make medicaments, methods of treatment using macrolides, and methods for making intermediates that, inter alia, may be used to make macrolides.
AT07787934T 2006-07-28 2007-07-26 METHOD FOR SYNTHESIS OF MACROLIDS ATE528312T1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US83406706P 2006-07-28 2006-07-28
EP06118159 2006-07-31
PCT/EP2007/057710 WO2008012343A2 (en) 2006-07-28 2007-07-26 Macrolide synthesis process

Publications (1)

Publication Number Publication Date
ATE528312T1 true ATE528312T1 (en) 2011-10-15

Family

ID=37547702

Family Applications (1)

Application Number Title Priority Date Filing Date
AT07787934T ATE528312T1 (en) 2006-07-28 2007-07-26 METHOD FOR SYNTHESIS OF MACROLIDS

Country Status (8)

Country Link
CN (1) CN102875622B (en)
AT (1) ATE528312T1 (en)
BR (1) BRPI0715642C8 (en)
ES (1) ES2374950T3 (en)
NZ (1) NZ574193A (en)
RU (1) RU2450014C2 (en)
SI (1) SI2089408T1 (en)
TW (1) TWI397534B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN104497082B (en) * 2015-01-13 2017-12-12 中国兽医药品监察所 A kind of synthetic method of tylonolide
CN113121625B (en) * 2019-12-31 2023-05-23 湖北龙翔药业科技股份有限公司 A new preparation method of tedrol
CN116478217A (en) * 2023-04-24 2023-07-25 济南久隆医药科技有限公司 Continuous synthesis method of tylosin

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE667952A (en) * 1964-08-05
JPS5896096A (en) * 1981-11-30 1983-06-07 Microbial Chem Res Found 19-decarbonyl-4'-deoxy mycaminosyl tylonolide derivative
US4629786A (en) * 1983-02-28 1986-12-16 Eli Lilly And Company C-20- and C-23 modified macrolide derivatives
IL71032A0 (en) * 1983-02-28 1984-05-31 Lilly Co Eli C-20 and c-23-modified macrolide derivatives
US4921947A (en) * 1986-03-31 1990-05-01 Eli Lilly And Company Process for preparing macrolide derivatives
PT1216256E (en) * 1999-08-30 2004-07-30 Zaidan Hojin Biseibutsu MACROLID ANTIBIOTICS AND PASTEURELLOSIS TREATMENT
US6506885B1 (en) * 2001-09-27 2003-01-14 The United States Of America As Represented By The Secretary Of Agriculture Monoclonal antibodies to the drug tilmicosin and a method for detecting the same
CN101506220B (en) * 2006-07-28 2012-10-17 英特威国际有限公司 Synthetic method of macrolide

Also Published As

Publication number Publication date
SI2089408T1 (en) 2012-02-29
BRPI0715642A2 (en) 2013-07-09
BRPI0715642B8 (en) 2020-06-30
CN102875622A (en) 2013-01-16
CN102875622B (en) 2016-12-07
RU2450014C2 (en) 2012-05-10
BRPI0715642B1 (en) 2020-06-09
ES2374950T3 (en) 2012-02-23
TWI397534B (en) 2013-06-01
RU2009107167A (en) 2010-09-10
BRPI0715642C8 (en) 2020-07-28
TW200831524A (en) 2008-08-01
NZ574193A (en) 2011-09-30

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