ATE534635T1 - N-pyrazinyl-phenylsulfonamide und deren verwendung zur behandlung von durch chemokine vermittelten krankheiten - Google Patents

N-pyrazinyl-phenylsulfonamide und deren verwendung zur behandlung von durch chemokine vermittelten krankheiten

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Publication number
ATE534635T1
ATE534635T1 AT03700655T AT03700655T ATE534635T1 AT E534635 T1 ATE534635 T1 AT E534635T1 AT 03700655 T AT03700655 T AT 03700655T AT 03700655 T AT03700655 T AT 03700655T AT E534635 T1 ATE534635 T1 AT E534635T1
Authority
AT
Austria
Prior art keywords
phenylsulfonamides
pyrazinyl
mediated diseases
treating chemokine
chemokine
Prior art date
Application number
AT03700655T
Other languages
English (en)
Inventor
Andrew Baxter
Timothy Johnson
Nicholas Kindon
Bryan Roberts
Michael Stocks
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from SE0200119A external-priority patent/SE0200119D0/xx
Priority claimed from SE0201857A external-priority patent/SE0201857D0/xx
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Application granted granted Critical
Publication of ATE534635T1 publication Critical patent/ATE534635T1/de

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    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/14—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D241/22—Benzenesulfonamido pyrazines
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  • Health & Medical Sciences (AREA)
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  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
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  • Immunology (AREA)
  • Neurology (AREA)
  • Pulmonology (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Neurosurgery (AREA)
  • Dermatology (AREA)
  • Endocrinology (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
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AT03700655T 2002-01-16 2003-01-14 N-pyrazinyl-phenylsulfonamide und deren verwendung zur behandlung von durch chemokine vermittelten krankheiten ATE534635T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
SE0200119A SE0200119D0 (sv) 2002-01-16 2002-01-16 Novel compounds
SE0201857A SE0201857D0 (sv) 2002-06-17 2002-06-17 Novel compounds
PCT/SE2003/000041 WO2003059893A1 (en) 2002-01-16 2003-01-14 N-pyrazinyl-phenylsulphonamides and their use in the treatment of chemokine mediated diseases

Publications (1)

Publication Number Publication Date
ATE534635T1 true ATE534635T1 (de) 2011-12-15

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AT03700655T ATE534635T1 (de) 2002-01-16 2003-01-14 N-pyrazinyl-phenylsulfonamide und deren verwendung zur behandlung von durch chemokine vermittelten krankheiten

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US (2) US7662825B2 (de)
EP (1) EP1467976B1 (de)
JP (1) JP4504021B2 (de)
KR (1) KR20040073566A (de)
CN (1) CN100357275C (de)
AR (1) AR038179A1 (de)
AT (1) ATE534635T1 (de)
AU (1) AU2003201802A1 (de)
BR (1) BR0306922A (de)
CA (1) CA2472204A1 (de)
CO (1) CO5640137A2 (de)
ES (1) ES2375107T3 (de)
IL (1) IL162678A0 (de)
IS (1) IS7348A (de)
MX (1) MXPA04006806A (de)
NO (1) NO20043370L (de)
NZ (1) NZ533750A (de)
PL (1) PL371432A1 (de)
RU (1) RU2312105C9 (de)
TW (1) TWI328007B (de)
WO (1) WO2003059893A1 (de)

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AU2003252478A1 (en) * 2002-07-10 2004-02-02 Ono Pharmaceutical Co., Ltd. Ccr4 antagonist and medicinal use thereof
GB0217431D0 (en) 2002-07-27 2002-09-04 Astrazeneca Ab Novel compounds
WO2004018435A1 (en) 2002-08-24 2004-03-04 Astrazeneca Ab Pyrimidine derivatives as modulators of chemokine receptor activity
SE0301653D0 (sv) * 2003-06-05 2003-06-05 Astrazeneca Ab Novel compounds
SE0302304D0 (sv) * 2003-08-27 2003-08-27 Astrazeneca Ab Novel compounds
WO2005023771A1 (ja) * 2003-09-05 2005-03-17 Ono Pharmaceutical Co., Ltd. ケモカインレセプターアンタゴニストおよびその医薬用途
GB0401269D0 (en) * 2004-01-21 2004-02-25 Astrazeneca Ab Compounds
WO2006020830A2 (en) * 2004-08-12 2006-02-23 Amgen Inc. Bisaryl-sulfonamides
EP2311827A1 (de) 2004-08-28 2011-04-20 AstraZeneca AB Thiopyrimidin-Derivat zur Verwendung als Zwischenprodukt Chemokine-Rezeptor-Modulatoren
TW200800921A (en) * 2005-09-19 2008-01-01 Astrazeneca Ab Novel compounds
WO2007063935A1 (ja) * 2005-12-02 2007-06-07 Mitsubishi Tanabe Pharma Corporation 芳香族化合物
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HK1068885A1 (en) 2005-05-06
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