ATE540023T1 - Neuartige 3-aminoalkyl-1,3-dihydro-2h-indol-2-on- derivate, ihre herstellung und therapeutische verwendung - Google Patents

Neuartige 3-aminoalkyl-1,3-dihydro-2h-indol-2-on- derivate, ihre herstellung und therapeutische verwendung

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Publication number
ATE540023T1
ATE540023T1 AT09721627T AT09721627T ATE540023T1 AT E540023 T1 ATE540023 T1 AT E540023T1 AT 09721627 T AT09721627 T AT 09721627T AT 09721627 T AT09721627 T AT 09721627T AT E540023 T1 ATE540023 T1 AT E540023T1
Authority
AT
Austria
Prior art keywords
indol
aminoalkyl
dihydro
derivatives
novel
Prior art date
Application number
AT09721627T
Other languages
English (en)
Inventor
Loic Foulon
Laurent Goullieux
Brigitte Pouzet
Gal Claudine Serradeil-Le
Gerard Valette
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Sa filed Critical Sanofi Sa
Application granted granted Critical
Publication of ATE540023T1 publication Critical patent/ATE540023T1/de

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/32—Oxygen atoms
    • C07D209/34—Oxygen atoms in position 2
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AT09721627T 2008-02-19 2009-02-18 Neuartige 3-aminoalkyl-1,3-dihydro-2h-indol-2-on- derivate, ihre herstellung und therapeutische verwendung ATE540023T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0800866A FR2927625B1 (fr) 2008-02-19 2008-02-19 Nouveaux derives de 3-aminoalkyl-1,3-dihydro-2h-indol-2-one, leur preparation et leur application en therapeutique
PCT/FR2009/000179 WO2009115685A1 (fr) 2008-02-19 2009-02-18 Nouveaux derives de 3-aminoalkyl-1,3-dihydro-2h-indol-2-one, leur preparation et leur application en therapeutique.

Publications (1)

Publication Number Publication Date
ATE540023T1 true ATE540023T1 (de) 2012-01-15

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AT09721627T ATE540023T1 (de) 2008-02-19 2009-02-18 Neuartige 3-aminoalkyl-1,3-dihydro-2h-indol-2-on- derivate, ihre herstellung und therapeutische verwendung

Country Status (15)

Country Link
US (1) US8362067B2 (de)
EP (1) EP2265582B1 (de)
JP (1) JP5602639B2 (de)
KR (1) KR20100126401A (de)
CN (1) CN102015642A (de)
AR (1) AR070438A1 (de)
AT (1) ATE540023T1 (de)
AU (1) AU2009227111A1 (de)
BR (1) BRPI0907578A2 (de)
CA (1) CA2716035A1 (de)
FR (1) FR2927625B1 (de)
IL (1) IL207629A0 (de)
MX (1) MX2010009092A (de)
RU (1) RU2010138575A (de)
WO (1) WO2009115685A1 (de)

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Publication number Priority date Publication date Assignee Title
FR2927625B1 (fr) 2008-02-19 2010-03-12 Sanofi Aventis Nouveaux derives de 3-aminoalkyl-1,3-dihydro-2h-indol-2-one, leur preparation et leur application en therapeutique
AU2011272738B2 (en) 2010-07-01 2015-08-20 Azevan Pharmaceuticals, Inc. Methods for treating post traumatic stress disorder
BR112016022575A2 (pt) * 2014-03-28 2017-08-15 Azevan Pharmaceuticals Inc Composições e métodos para o tratamento de doenças neurodegenerativas
CN104592088B (zh) * 2015-01-05 2019-01-01 内蒙古工业大学 月桂酸催化制备3-胺烷基吲哚的方法
CN105061290B (zh) * 2015-08-28 2017-11-10 福建品派包装有限公司 一种吲哚酮类化合物的合成方法
CN105061291B (zh) * 2015-09-08 2017-08-04 江俞 一种杂稠环取代的吲哚酮类化合物的合成方法
KR102790657B1 (ko) 2017-09-15 2025-04-02 아제반 파마슈티칼스, 인코퍼레이티드 뇌 손상을 치료하기 위한 조성물 및 방법
CN108675945B (zh) * 2018-06-22 2020-09-22 湖南科技大学 ((2-羟基苄基)胺基)苯基脲类化合物及其制备方法和用途
CN118047699A (zh) * 2024-02-18 2024-05-17 武威广达科技有限公司 一种4-异丙氧基苯磺酰氯的制备方法

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AR070438A1 (es) 2010-04-07
FR2927625A1 (fr) 2009-08-21
CA2716035A1 (fr) 2009-09-24
JP2011512389A (ja) 2011-04-21
CN102015642A (zh) 2011-04-13
MX2010009092A (es) 2011-09-21
US20110059955A1 (en) 2011-03-10
JP5602639B2 (ja) 2014-10-08
RU2010138575A (ru) 2012-03-27
BRPI0907578A2 (pt) 2019-09-24
US8362067B2 (en) 2013-01-29
AU2009227111A1 (en) 2009-09-24
IL207629A0 (en) 2010-12-30
WO2009115685A1 (fr) 2009-09-24
FR2927625B1 (fr) 2010-03-12
KR20100126401A (ko) 2010-12-01
EP2265582B1 (de) 2012-01-04
EP2265582A1 (de) 2010-12-29

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