AU2009232012A1 - Substituted piperidines as therapeutic compounds - Google Patents
Substituted piperidines as therapeutic compounds Download PDFInfo
- Publication number
- AU2009232012A1 AU2009232012A1 AU2009232012A AU2009232012A AU2009232012A1 AU 2009232012 A1 AU2009232012 A1 AU 2009232012A1 AU 2009232012 A AU2009232012 A AU 2009232012A AU 2009232012 A AU2009232012 A AU 2009232012A AU 2009232012 A1 AU2009232012 A1 AU 2009232012A1
- Authority
- AU
- Australia
- Prior art keywords
- methoxy
- straight
- chain
- acid
- methyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/06—Antimalarials
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Tropical Medicine & Parasitology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Virology (AREA)
- Neurology (AREA)
- Molecular Biology (AREA)
- Oncology (AREA)
- Hospice & Palliative Care (AREA)
- Communicable Diseases (AREA)
- AIDS & HIV (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP08153929 | 2008-04-02 | ||
| EP08153929.8 | 2008-04-02 | ||
| PCT/EP2009/053898 WO2009121914A1 (en) | 2008-04-02 | 2009-04-01 | Substituted piperidines as therapeutic compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2009232012A1 true AU2009232012A1 (en) | 2009-10-08 |
Family
ID=40627638
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2009232012A Abandoned AU2009232012A1 (en) | 2008-04-02 | 2009-04-01 | Substituted piperidines as therapeutic compounds |
Country Status (10)
| Country | Link |
|---|---|
| EP (1) | EP2271644A1 (pt) |
| JP (1) | JP2011516453A (pt) |
| KR (1) | KR20110002459A (pt) |
| CN (1) | CN101970431A (pt) |
| AU (1) | AU2009232012A1 (pt) |
| BR (1) | BRPI0910991A2 (pt) |
| CA (1) | CA2719070A1 (pt) |
| EA (1) | EA201001517A1 (pt) |
| MX (1) | MX2010010876A (pt) |
| WO (1) | WO2009121914A1 (pt) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2011057160A2 (en) * | 2009-11-06 | 2011-05-12 | The Regents Of The Uiversity Of California | Method to improve the immunogenicity of vaccine antigens by modification of cleavage sites in hiv-1 gp 120 |
| JP5099731B1 (ja) | 2009-10-14 | 2012-12-19 | メルク・シャープ・アンド・ドーム・コーポレーション | ｐ５３活性を増大する置換ピペリジン及びその使用 |
| GB201008209D0 (en) * | 2010-05-17 | 2010-06-30 | Senexis Ltd | Compounds |
| WO2013062923A1 (en) | 2011-10-28 | 2013-05-02 | Merck Sharp & Dohme Corp. | MACROCYCLES THAT INCREASE p53 ACTIVITY AND THE USES THEREOF |
| EP2935263B1 (en) | 2012-12-20 | 2018-12-05 | Merck Sharp & Dohme Corp. | Substituted imidazopyridines as hdm2 inhibitors |
| CN105001300A (zh) * | 2014-04-17 | 2015-10-28 | 复旦大学 | 组织蛋白酶d抑制剂及其制备方法、药物组合物和应用 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1816122A3 (en) * | 2006-01-19 | 2007-09-19 | Speedel Experimenta AG | 3,4,5-substituted piperidines as therapeutic compounds |
| EP1911758A1 (en) * | 2006-10-04 | 2008-04-16 | Speedel Experimenta AG | Phenyl piperidine derivatives for use as renin inhibitors |
| EP1908761A1 (en) * | 2006-10-04 | 2008-04-09 | Speedel Experimenta AG | Organic compounds |
-
2009
- 2009-04-01 EA EA201001517A patent/EA201001517A1/ru unknown
- 2009-04-01 CN CN2009801083136A patent/CN101970431A/zh active Pending
- 2009-04-01 MX MX2010010876A patent/MX2010010876A/es not_active Application Discontinuation
- 2009-04-01 EP EP09728288A patent/EP2271644A1/en not_active Withdrawn
- 2009-04-01 AU AU2009232012A patent/AU2009232012A1/en not_active Abandoned
- 2009-04-01 CA CA2719070A patent/CA2719070A1/en not_active Abandoned
- 2009-04-01 WO PCT/EP2009/053898 patent/WO2009121914A1/en not_active Ceased
- 2009-04-01 KR KR1020107022007A patent/KR20110002459A/ko not_active Withdrawn
- 2009-04-01 BR BRPI0910991A patent/BRPI0910991A2/pt not_active Application Discontinuation
- 2009-04-01 JP JP2011502382A patent/JP2011516453A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| EA201001517A1 (ru) | 2011-04-29 |
| EP2271644A1 (en) | 2011-01-12 |
| KR20110002459A (ko) | 2011-01-07 |
| MX2010010876A (es) | 2010-10-26 |
| JP2011516453A (ja) | 2011-05-26 |
| BRPI0910991A2 (pt) | 2016-01-19 |
| CN101970431A (zh) | 2011-02-09 |
| CA2719070A1 (en) | 2009-10-08 |
| WO2009121914A1 (en) | 2009-10-08 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK5 | Application lapsed section 142(2)(e) - patent request and compl. specification not accepted |