BE2024C511I2 - - Google Patents

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Publication number
BE2024C511I2
BE2024C511I2 BE2024C511C BE2024C511C BE2024C511I2 BE 2024C511 I2 BE2024C511 I2 BE 2024C511I2 BE 2024C511 C BE2024C511 C BE 2024C511C BE 2024C511 C BE2024C511 C BE 2024C511C BE 2024C511 I2 BE2024C511 I2 BE 2024C511I2
Authority
BE
Belgium
Application number
BE2024C511C
Other languages
Dutch (nl)
Original Assignee
Japan Tobacco Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35079161&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BE2024C511(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Japan Tobacco Inc filed Critical Japan Tobacco Inc
Publication of BE2024C511I2 publication Critical patent/BE2024C511I2/nl

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Virology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
BE2024C511C 2004-05-20 2024-03-15 BE2024C511I2 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2004150979 2004-05-20

Publications (1)

Publication Number Publication Date
BE2024C511I2 true BE2024C511I2 (tr) 2024-10-08

Family

ID=35079161

Family Applications (1)

Application Number Title Priority Date Filing Date
BE2024C511C BE2024C511I2 (tr) 2004-05-20 2024-03-15

Country Status (33)

Country Link
US (7) US7635704B2 (tr)
EP (4) EP1636190B1 (tr)
JP (1) JP3754064B2 (tr)
KR (1) KR20080064909A (tr)
CN (1) CN1956961B (tr)
AR (2) AR049280A1 (tr)
AU (1) AU2005245296B2 (tr)
BE (1) BE2024C511I2 (tr)
BR (1) BRPI0510114B8 (tr)
CA (1) CA2566922C (tr)
CY (4) CY1113010T1 (tr)
DK (2) DK1636190T3 (tr)
ES (2) ES2388441T3 (tr)
FI (2) FI3281939T3 (tr)
FR (1) FR23C1040I1 (tr)
HR (2) HRP20231588T3 (tr)
HU (2) HUE064615T2 (tr)
IL (1) IL179250A0 (tr)
LT (2) LT3281939T (tr)
LU (1) LUC00334I2 (tr)
MX (1) MXPA06013405A (tr)
MY (1) MY134672A (tr)
NO (8) NO339223B1 (tr)
NZ (1) NZ551839A (tr)
PE (2) PE20120361A1 (tr)
PL (2) PL1636190T3 (tr)
PT (2) PT3281939T (tr)
RS (2) RS64845B1 (tr)
RU (1) RU2330845C1 (tr)
SI (2) SI1636190T1 (tr)
TW (1) TWI329015B (tr)
WO (1) WO2005113508A1 (tr)
ZA (1) ZA200610647B (tr)

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MY134672A (en) * 2004-05-20 2007-12-31 Japan Tobacco Inc Stable crystal of 4-oxoquinoline compound
WO2007063869A1 (ja) * 2005-11-30 2007-06-07 Japan Tobacco Inc. 高純度キノロン化合物の製造方法
EA201201496A1 (ru) 2005-12-30 2013-07-30 Джилид Сайэнс, Инк. Способ ингибирования интегразы вич, способ улучшения фармакокинетики 6-(3-хлор-2-фторбензил)-1-[(2s)-1-гидрокси-3-метилбутан-2-ил]-7-метокси-4-оксо-1,4-дигидрохинолин-3-карбоновой кислоты (варианты), набор, фармацевтическая композиция (варианты) и антиретровирусный агент (варианты)
US20090233964A1 (en) * 2005-12-30 2009-09-17 Gilead Sciences, Inc. Methods for improving the pharmacokinetics of hiv integrase inhibitors
AU2013203476C1 (en) * 2005-12-30 2016-11-17 Gilead Sciences, Inc. Methods for improving the pharmacokinetics of hiv integrase inhibitors
WO2007089030A1 (en) * 2006-02-01 2007-08-09 Japan Tobacco Inc. Use of 6-(3-chloro-2-fluorobenzyl)-1-[(2s)-1-hydroxy-3-methylbutan-2-yl]-7-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxylic acid or salt thereof for treating retrovirus infection
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WO2007102512A1 (ja) 2006-03-06 2007-09-13 Japan Tobacco Inc. ４－オキソキノリン化合物の製造方法
AU2007275860C1 (en) 2006-07-07 2014-06-12 Gilead Sciences, Inc. Modulators of pharmacokinetic properties of therapeutics
SG174787A1 (en) 2006-09-12 2011-10-28 Gilead Sciences Inc Process and intermediates for preparing integrase inhibitors
HUE029842T2 (en) 2007-02-23 2017-04-28 Gilead Sciences Inc Modulators of pharmacokinetic properties of therapeutics
TW200914011A (en) * 2007-06-29 2009-04-01 Gilead Sciences Inc Therapeutic compositions and methods
WO2009006203A1 (en) * 2007-06-29 2009-01-08 Gilead Sciences, Inc. Therapeutic compositions and the use thereof
AR068403A1 (es) 2007-09-11 2009-11-18 Gilead Sciences Inc Proceso e intermediarios para la preparacion de inhibidores de integrasa
PT2296633E (pt) 2008-05-02 2015-12-04 Gilead Sciences Inc A utilização de partículas de portador sólido para melhorar a processabilidade de um agente farmacêutico
JP5611242B2 (ja) 2009-02-06 2014-10-22 ギリアード サイエンシーズ， インコーポレイテッド 併用治療のための錠剤
WO2010137032A2 (en) * 2009-05-14 2010-12-02 Matrix Laboratories Ltd. Novel polymorphic forms of elvitegravir and its pharmaceutically acceptable salts
WO2011004389A2 (en) * 2009-06-18 2011-01-13 Matrix Laboratories Ltd An improved process for the preparation of elvitegravir
CN102212032B (zh) * 2011-04-20 2013-07-31 复旦大学 一种5-羟基喹诺酮类衍生物及其制备方法和用途
KR101663436B1 (ko) 2012-07-06 2016-10-06 제넨테크, 인크. N-치환된 벤즈아미드 및 이의 사용 방법
BR112015002275A2 (pt) 2012-08-03 2017-07-04 Gilead Sciences Inc processos e intermediários para a preparação de inibidores da integrase
CN103819402B (zh) * 2012-11-17 2016-03-30 上海迪赛诺化学制药有限公司 埃替拉韦中间体及其制备方法和应用
CN103864682B (zh) * 2012-12-18 2016-12-28 上海迪赛诺化学制药有限公司 一种制备iii型埃替拉韦晶体的方法
PL3608325T3 (pl) 2012-12-21 2022-11-07 Gilead Sciences, Inc. Policykliczne związki karbamoilopirydonu i ich zastosowanie farmaceutyczne
HUE037347T2 (hu) 2013-07-12 2018-08-28 Gilead Sciences Inc Policiklusos karmaboilpiridon vegyületek és alkalmazásuk HIV fertõzések kezelésére
NO2865735T3 (tr) 2013-07-12 2018-07-21
CN105315203A (zh) * 2014-06-06 2016-02-10 上海迪赛诺化学制药有限公司 一种v型埃替拉韦晶体及其制备方法
NO2717902T3 (tr) 2014-06-20 2018-06-23
TWI744723B (zh) 2014-06-20 2021-11-01 美商基利科學股份有限公司 多環型胺甲醯基吡啶酮化合物之合成
TW201613936A (en) 2014-06-20 2016-04-16 Gilead Sciences Inc Crystalline forms of(2R,5S,13aR)-8-hydroxy-7,9-dioxo-n-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide
TWI695003B (zh) 2014-12-23 2020-06-01 美商基利科學股份有限公司 多環胺甲醯基吡啶酮化合物及其醫藥用途
ES2837383T3 (es) 2015-04-02 2021-06-30 Gilead Sciences Inc Compuestos de carbamoilpiridonas policíclicos y su utilización farmacéutica
CN106008195B (zh) * 2016-05-19 2018-08-03 绍兴文理学院 一种2，4-二氟-5-碘苯甲酸的制备方法
EP3984536B1 (en) * 2020-10-19 2025-06-25 Centre national de la recherche scientifique Inhibition of the hiv-1 replication by compounds directed against a new target of the viral cycle

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Also Published As

Publication number Publication date
EP1636190B1 (en) 2012-06-27
TW200600097A (en) 2006-01-01
NO20161297A1 (no) 2007-02-07
US20060030710A1 (en) 2006-02-09
JP3754064B2 (ja) 2006-03-08
US7635704B2 (en) 2009-12-22
PT1636190E (pt) 2012-08-20
FI3281939T3 (fi) 2023-10-23
FR23C1040I1 (fr) 2023-12-29
EP3281939A1 (en) 2018-02-14
EP4299563A3 (en) 2024-02-28
CA2566922C (en) 2011-01-11
NO20190051A1 (no) 2007-02-07
MXPA06013405A (es) 2007-03-01
AR096100A2 (es) 2015-12-09
NO347902B1 (no) 2024-05-06
LTPA2024001I1 (tr) 2024-04-10
RS52375B (sr) 2012-12-31
DK3281939T3 (da) 2024-01-22
SI1636190T1 (sl) 2012-09-28
ES2388441T3 (es) 2012-10-15
NO20220690A1 (no) 2007-02-07
BRPI0510114B1 (pt) 2020-09-15
NO2024034I1 (no) 2024-07-15
CY2015009I1 (el) 2024-09-20
US20180029989A1 (en) 2018-02-01
CY1126560T1 (el) 2024-09-20
AR049280A1 (es) 2006-07-12
NO20240384A1 (no) 2007-02-07
FIC20240008I1 (fi) 2024-03-20
HRP20120681T1 (hr) 2012-09-30
US8981103B2 (en) 2015-03-17
EP2514746A1 (en) 2012-10-24
IL179250A0 (en) 2007-03-08
RU2330845C1 (ru) 2008-08-10
KR20080064909A (ko) 2008-07-09
PE20060358A1 (es) 2006-05-12
NO20230913A1 (no) 2007-02-07
NO20200873A1 (no) 2007-02-07
PL1636190T3 (pl) 2012-10-31
BRPI0510114B8 (pt) 2021-05-25
DK1636190T3 (da) 2012-09-24
JP2006001927A (ja) 2006-01-05
PL3281939T3 (pl) 2024-03-18
HK1083341A1 (en) 2006-06-30
HUE064615T2 (hu) 2024-04-28
ZA200610647B (en) 2008-06-25
CY2015009I2 (el) 2024-09-20
CY2024008I1 (el) 2024-09-20
US20250091995A1 (en) 2025-03-20
US20190185433A1 (en) 2019-06-20
CN1956961A (zh) 2007-05-02
HRP20231588T3 (hr) 2024-03-15
AU2005245296A1 (en) 2005-12-01
NO339223B1 (no) 2016-11-21
HUS2400006I1 (hu) 2024-04-28
US20220235009A1 (en) 2022-07-28
EP4299563A2 (en) 2024-01-03
LT3281939T (lt) 2023-11-27
US20150361044A1 (en) 2015-12-17
SI3281939T1 (sl) 2024-02-29
AU2005245296B2 (en) 2010-08-12
PT3281939T (pt) 2023-11-22
BRPI0510114A (pt) 2007-09-25
NO20065790L (no) 2007-02-07
CY1113010T1 (el) 2016-04-13
TWI329015B (en) 2010-08-21
LTC3281939I2 (tr) 2025-04-25
NZ551839A (en) 2009-11-27
LUC00334I2 (tr) 2024-07-01
WO2005113508A1 (en) 2005-12-01
EP3281939B1 (en) 2023-10-18
PE20120361A1 (es) 2012-05-03
MY134672A (en) 2007-12-31
ES2960824T3 (es) 2024-03-06
CY2024008I2 (el) 2024-09-20
US20100204271A1 (en) 2010-08-12
CN1956961B (zh) 2010-05-26
CA2566922A1 (en) 2005-12-01
RS64845B1 (sr) 2023-12-29
EP1636190A1 (en) 2006-03-22

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