BE618813A - Diazabicyclo-octanes - Google Patents
Diazabicyclo-octanesInfo
- Publication number
- BE618813A BE618813A BE618813A BE618813A BE618813A BE 618813 A BE618813 A BE 618813A BE 618813 A BE618813 A BE 618813A BE 618813 A BE618813 A BE 618813A BE 618813 A BE618813 A BE 618813A
- Authority
- BE
- Belgium
- Prior art keywords
- octanes
- diazabicyclo
- Prior art date
Links
- NFDXQGNDWIPXQL-UHFFFAOYSA-N 1-cyclooctyldiazocane Chemical class C1CCCCCCC1N1NCCCCCC1 NFDXQGNDWIPXQL-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/5545—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having eight-membered rings not containing additional condensed or non-condensed nitrogen-containing 3-7 membered rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB23076/61A GB949088A (en) | 1961-06-26 | 1961-06-26 | Diazabicyclo-octane derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BE618813A true BE618813A (fr) | 1962-10-01 |
Family
ID=10189738
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BE618813A BE618813A (fr) | 1961-06-26 | 1962-06-12 | Diazabicyclo-octanes |
Country Status (6)
| Country | Link |
|---|---|
| BE (1) | BE618813A (fr) |
| BR (1) | BR6240334D0 (fr) |
| CH (1) | CH423799A (fr) |
| DK (1) | DK105414C (fr) |
| FI (1) | FI40096C (fr) |
| GB (1) | GB949088A (fr) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1995023152A1 (fr) * | 1994-02-23 | 1995-08-31 | Riace Establishment | Derives de 3,8-diazabicyclo[3.2.1]octane possedant une activite analgesique |
| WO2006058879A1 (fr) * | 2004-11-30 | 2006-06-08 | Neurosearch A/S | Nouveaux derives aryliques diazabicycliques utilises en tant que ligands cholinergiques |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE0003795D0 (sv) | 2000-10-20 | 2000-10-20 | Astrazeneca Ab | Pharmaceutically useful compounds |
| US8673920B2 (en) * | 2009-05-06 | 2014-03-18 | Merck Sharp & Dohme Corp. | Inhibitors of the renal outer medullary potassium channel |
| WO2012058116A1 (fr) | 2010-10-27 | 2012-05-03 | Merck Sharp & Dohme Corp. | Inhibiteurs du canal potassique de la médullaire externe rénale |
| EP2632464B1 (fr) | 2010-10-29 | 2015-04-29 | Merck Sharp & Dohme Corp. | Inhibiteurs du canal à potassium de la medulla externe du rein |
| AU2012299227A1 (en) | 2011-08-19 | 2014-02-20 | Merck Sharp & Dohme Corp. | Inhibitors of the renal outer medullary potassium channel |
| WO2013039802A1 (fr) | 2011-09-16 | 2013-03-21 | Merck Sharp & Dohme Corp. | Inhibiteurs du canal à potassium de la medulla externe du rein |
| US8999990B2 (en) | 2011-10-25 | 2015-04-07 | Merck Sharp & Dohme Corp. | Inhibitors of the renal outer medullary potassium channel |
| EP2771004B1 (fr) | 2011-10-25 | 2016-05-18 | Merck Sharp & Dohme Corp. | Inhibiteurs du canal potassique médullaire externe rénal |
| WO2013066714A1 (fr) | 2011-10-31 | 2013-05-10 | Merck Sharp & Dohme Corp. | Inhibiteurs du canal potassique médullaire externe rénal |
| EP2773351B1 (fr) | 2011-10-31 | 2017-08-23 | Merck Sharp & Dohme Corp. | Inhibiteurs du canal potassique médullaire externe rénal |
| EP2773206B1 (fr) | 2011-10-31 | 2018-02-21 | Merck Sharp & Dohme Corp. | Inhibiteurs du canal potassique médullaire externe rénal |
| EP2790511B1 (fr) | 2011-12-16 | 2016-09-14 | Merck Sharp & Dohme Corp. | Inhibiteurs du canal à potassium de la medulla externe du rein |
| AR092031A1 (es) | 2012-07-26 | 2015-03-18 | Merck Sharp & Dohme | Inhibidores del canal de potasio medular externo renal |
| EP2925322B1 (fr) | 2012-11-29 | 2018-10-24 | Merck Sharp & Dohme Corp. | Inhibiteurs du canal potassique médullaire extérieur rénal |
| US9573961B2 (en) | 2012-12-19 | 2017-02-21 | Merck Sharp & Dohme Corp. | Inhibitors of the renal outer medullary potassium channel |
| WO2014126944A2 (fr) | 2013-02-18 | 2014-08-21 | Merck Sharp & Dohme Corp. | Inhibiteurs du canal potassique médullaire extérieur rénal |
| EP2968288B1 (fr) | 2013-03-15 | 2018-07-04 | Merck Sharp & Dohme Corp. | Inhibiteurs du canal potassique médullaire extérieur rénal |
| EP3027625B1 (fr) | 2013-07-31 | 2018-05-30 | Merck Sharp & Dohme Corp. | Derives spiro-fusionnes de piperidine utiles dans le traitement, entre autres, de l'hypertension et de l' insuffisance cardiaque aiguë ou chronique |
| WO2016127358A1 (fr) | 2015-02-12 | 2016-08-18 | Merck Sharp & Dohme Corp. | Inhibiteurs du canal potassique médullaire externe rénal |
-
1961
- 1961-06-26 GB GB23076/61A patent/GB949088A/en not_active Expired
-
1962
- 1962-06-12 BE BE618813A patent/BE618813A/fr unknown
- 1962-06-18 CH CH727862A patent/CH423799A/de unknown
- 1962-06-25 DK DK282462AA patent/DK105414C/da active
- 1962-06-25 BR BR140334/62A patent/BR6240334D0/pt unknown
- 1962-06-25 FI FI122162A patent/FI40096C/fi active
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1995023152A1 (fr) * | 1994-02-23 | 1995-08-31 | Riace Establishment | Derives de 3,8-diazabicyclo[3.2.1]octane possedant une activite analgesique |
| WO2006058879A1 (fr) * | 2004-11-30 | 2006-06-08 | Neurosearch A/S | Nouveaux derives aryliques diazabicycliques utilises en tant que ligands cholinergiques |
| US7612074B2 (en) | 2004-11-30 | 2009-11-03 | Neurosearch A/S | Diazabicyclic aryl derivatives as cholinergy ligands |
Also Published As
| Publication number | Publication date |
|---|---|
| FI40096C (fi) | 1968-10-10 |
| FI40096B (fr) | 1968-06-28 |
| BR6240334D0 (pt) | 1973-05-24 |
| CH423799A (de) | 1966-11-15 |
| GB949088A (en) | 1964-02-12 |
| DK105414C (da) | 1966-09-26 |
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