BE618813A - Diazabicyclo-octanes - Google Patents

Diazabicyclo-octanes

Info

Publication number
BE618813A
BE618813A BE618813A BE618813A BE618813A BE 618813 A BE618813 A BE 618813A BE 618813 A BE618813 A BE 618813A BE 618813 A BE618813 A BE 618813A BE 618813 A BE618813 A BE 618813A
Authority
BE
Belgium
Prior art keywords
octanes
diazabicyclo
Prior art date
Application number
BE618813A
Other languages
English (en)
Original Assignee
Lepetit Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lepetit Spa filed Critical Lepetit Spa
Publication of BE618813A publication Critical patent/BE618813A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/5545Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having eight-membered rings not containing additional condensed or non-condensed nitrogen-containing 3-7 membered rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BE618813A 1961-06-26 1962-06-12 Diazabicyclo-octanes BE618813A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB23076/61A GB949088A (en) 1961-06-26 1961-06-26 Diazabicyclo-octane derivatives

Publications (1)

Publication Number Publication Date
BE618813A true BE618813A (fr) 1962-10-01

Family

ID=10189738

Family Applications (1)

Application Number Title Priority Date Filing Date
BE618813A BE618813A (fr) 1961-06-26 1962-06-12 Diazabicyclo-octanes

Country Status (6)

Country Link
BE (1) BE618813A (fr)
BR (1) BR6240334D0 (fr)
CH (1) CH423799A (fr)
DK (1) DK105414C (fr)
FI (1) FI40096C (fr)
GB (1) GB949088A (fr)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1995023152A1 (fr) * 1994-02-23 1995-08-31 Riace Establishment Derives de 3,8-diazabicyclo[3.2.1]octane possedant une activite analgesique
WO2006058879A1 (fr) * 2004-11-30 2006-06-08 Neurosearch A/S Nouveaux derives aryliques diazabicycliques utilises en tant que ligands cholinergiques

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0003795D0 (sv) 2000-10-20 2000-10-20 Astrazeneca Ab Pharmaceutically useful compounds
US8673920B2 (en) * 2009-05-06 2014-03-18 Merck Sharp & Dohme Corp. Inhibitors of the renal outer medullary potassium channel
WO2012058116A1 (fr) 2010-10-27 2012-05-03 Merck Sharp & Dohme Corp. Inhibiteurs du canal potassique de la médullaire externe rénale
EP2632464B1 (fr) 2010-10-29 2015-04-29 Merck Sharp & Dohme Corp. Inhibiteurs du canal à potassium de la medulla externe du rein
AU2012299227A1 (en) 2011-08-19 2014-02-20 Merck Sharp & Dohme Corp. Inhibitors of the renal outer medullary potassium channel
WO2013039802A1 (fr) 2011-09-16 2013-03-21 Merck Sharp & Dohme Corp. Inhibiteurs du canal à potassium de la medulla externe du rein
US8999990B2 (en) 2011-10-25 2015-04-07 Merck Sharp & Dohme Corp. Inhibitors of the renal outer medullary potassium channel
EP2771004B1 (fr) 2011-10-25 2016-05-18 Merck Sharp & Dohme Corp. Inhibiteurs du canal potassique médullaire externe rénal
WO2013066714A1 (fr) 2011-10-31 2013-05-10 Merck Sharp & Dohme Corp. Inhibiteurs du canal potassique médullaire externe rénal
EP2773351B1 (fr) 2011-10-31 2017-08-23 Merck Sharp & Dohme Corp. Inhibiteurs du canal potassique médullaire externe rénal
EP2773206B1 (fr) 2011-10-31 2018-02-21 Merck Sharp & Dohme Corp. Inhibiteurs du canal potassique médullaire externe rénal
EP2790511B1 (fr) 2011-12-16 2016-09-14 Merck Sharp & Dohme Corp. Inhibiteurs du canal à potassium de la medulla externe du rein
AR092031A1 (es) 2012-07-26 2015-03-18 Merck Sharp & Dohme Inhibidores del canal de potasio medular externo renal
EP2925322B1 (fr) 2012-11-29 2018-10-24 Merck Sharp & Dohme Corp. Inhibiteurs du canal potassique médullaire extérieur rénal
US9573961B2 (en) 2012-12-19 2017-02-21 Merck Sharp & Dohme Corp. Inhibitors of the renal outer medullary potassium channel
WO2014126944A2 (fr) 2013-02-18 2014-08-21 Merck Sharp & Dohme Corp. Inhibiteurs du canal potassique médullaire extérieur rénal
EP2968288B1 (fr) 2013-03-15 2018-07-04 Merck Sharp & Dohme Corp. Inhibiteurs du canal potassique médullaire extérieur rénal
EP3027625B1 (fr) 2013-07-31 2018-05-30 Merck Sharp & Dohme Corp. Derives spiro-fusionnes de piperidine utiles dans le traitement, entre autres, de l'hypertension et de l' insuffisance cardiaque aiguë ou chronique
WO2016127358A1 (fr) 2015-02-12 2016-08-18 Merck Sharp & Dohme Corp. Inhibiteurs du canal potassique médullaire externe rénal

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1995023152A1 (fr) * 1994-02-23 1995-08-31 Riace Establishment Derives de 3,8-diazabicyclo[3.2.1]octane possedant une activite analgesique
WO2006058879A1 (fr) * 2004-11-30 2006-06-08 Neurosearch A/S Nouveaux derives aryliques diazabicycliques utilises en tant que ligands cholinergiques
US7612074B2 (en) 2004-11-30 2009-11-03 Neurosearch A/S Diazabicyclic aryl derivatives as cholinergy ligands

Also Published As

Publication number Publication date
FI40096C (fi) 1968-10-10
FI40096B (fr) 1968-06-28
BR6240334D0 (pt) 1973-05-24
CH423799A (de) 1966-11-15
GB949088A (en) 1964-02-12
DK105414C (da) 1966-09-26

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