BE847900A - Nouveaux derives d'aminoglycosides, leur procede de preparation et application a la formation de compositions antibacteriennes - Google Patents

Nouveaux derives d'aminoglycosides, leur procede de preparation et application a la formation de compositions antibacteriennes

Info

Publication number
BE847900A
BE847900A BE172004A BE172004A BE847900A BE 847900 A BE847900 A BE 847900A BE 172004 A BE172004 A BE 172004A BE 172004 A BE172004 A BE 172004A BE 847900 A BE847900 A BE 847900A
Authority
BE
Belgium
Prior art keywords
aminoglycosides
formation
application
preparation process
new derivatives
Prior art date
Application number
BE172004A
Other languages
English (en)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of BE847900A publication Critical patent/BE847900A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/22Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BE172004A 1975-11-04 1976-11-03 Nouveaux derives d'aminoglycosides, leur procede de preparation et application a la formation de compositions antibacteriennes BE847900A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US62863775A 1975-11-04 1975-11-04

Publications (1)

Publication Number Publication Date
BE847900A true BE847900A (fr) 1977-05-03

Family

ID=24519719

Family Applications (1)

Application Number Title Priority Date Filing Date
BE172004A BE847900A (fr) 1975-11-04 1976-11-03 Nouveaux derives d'aminoglycosides, leur procede de preparation et application a la formation de compositions antibacteriennes

Country Status (6)

Country Link
US (1) US4062947A (fr)
JP (1) JPS5259134A (fr)
BE (1) BE847900A (fr)
DE (1) DE2648973A1 (fr)
FR (1) FR2330407A1 (fr)
GB (1) GB1557687A (fr)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4217446A (en) * 1974-10-26 1980-08-12 Pfizer Inc. ωAmino-2-hydroxyalkyl derivatives of aminoglycoside antibiotics
NZ184213A (en) * 1976-06-16 1980-05-27 Pfizer 2-deoxystreptamine aminoglycosides and antibacterial pharmaceutical compositions
DE2712160A1 (de) * 1977-03-19 1978-09-28 Bayer Ag Pseudotrisaccharide, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
DE2753769A1 (de) * 1977-12-02 1979-06-13 Bayer Ag 1-n-4,6-di-o-(aminoglykosyl)-1,3- diamino-cyclitol-derivate, verfahren zu ihrer herstellung sowie ihre verwendung
US4180564A (en) * 1978-05-25 1979-12-25 Eli Lilly And Company A-38533 Antibiotics and process for production thereof
DE2832268A1 (de) * 1978-07-22 1980-01-31 Bayer Ag Pseudotrisaccharide
DE2840907A1 (de) * 1978-09-20 1980-04-03 Bayer Ag Selektiv geschuetzte 4,6-di-o-(aminoglykosyl)-1,3-diaminocyclitole
US4243801A (en) * 1979-07-12 1981-01-06 Schering Corporation 6"-Amino derivatives of 4-0-aminoglycosyl-6-0-garosaminyl-1,3-diaminocyclitols
JPS5950642B2 (ja) * 1981-04-08 1984-12-10 ウェルファイド株式会社 工業用殺菌剤
FI822671A7 (fi) * 1981-08-07 1983-02-08 Sandoz Ag Aminoglykosidijohdannaisia, menetelmiä niiden valmistamiseksi, niitä sisältäviä farmaseuttisia koostumuksia ssekä tällaisia johdannaisia kä ytettäviksi lääkeaineina.
US6481259B1 (en) * 2000-08-17 2002-11-19 Castle, Inc. Method for precision bending of a sheet of material and slit sheet therefor
US7829543B2 (en) * 2003-01-07 2010-11-09 Paratek Pharmaceuticals, Inc. Substituted polyamines as inhibitors of bacterial efflux pumps

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3920628A (en) * 1972-10-24 1975-11-18 Schering Corp 2{41 -Deoxyaminoglycosides and 2{41 -epi-amino-3{41 -desamino derivatives thereof, methods for their manufacture and novel intermediates useful therein
US4002742A (en) * 1974-03-19 1977-01-11 Schering Corporation 1-N-alkyl-4,6-di-(aminoglycosyl)-1,3-diaminocyclitols, methods for their manufacture, methods for their use as antibacterial agents, and compositions useful therefor

Also Published As

Publication number Publication date
JPS5259134A (en) 1977-05-16
FR2330407A1 (fr) 1977-06-03
GB1557687A (en) 1979-12-12
US4062947A (en) 1977-12-13
DE2648973A1 (de) 1977-05-12

Similar Documents

Publication Publication Date Title
FR2320295A1 (fr) Nouveaux derives de la 2,3-dioxopiperazine et leur procede de preparation
FR2281340A1 (fr) Derives de l'acide folique, leur procede de preparation et leur application
BE823027A (fr) Derives d'isoquinoleine et leur procede de preparation
FR2330407A1 (fr) Nouveaux derives d'aminoglycosides, leur procede de preparation et application a la formation de compositions antibacteriennes
BE844066A (fr) Nouveaux ethers de 2', 3,6'-trichloro-4-cyano-4'-benzoylureidodiphenyle, leur procede de preparation et leur application
BE783260A (fr) Nouveaux derives d'imidazolidinone-(2), leur procede de preparation et leur application comme herbicides
BE845317A (fr) Nouveaux procede de preparation d'azines
FR2331593A1 (fr) Compositions d'ether de polygalactomannane et leur procede de preparation
BE823692A (fr) Nouveaux derives d'acide prostanoique et leur procede de preparation
FR2337719A1 (fr) Nouveaux triazolyl-o,n-acetals acyles, leur procede de preparation et leur application comme fongicides
FR2317930A1 (fr) Nouveaux derives d'apovincaminol, leur procede de preparation et leur application
BE827870A (fr) Derives d'emidazole et leur procede de preparation
FR2290207A1 (fr) Nouveaux derives de 3,4-dihydrocarbostyril et leur procede de preparation
BE819321A (fr) Nouveaux 2,3-dihydrobenzofuranyl-7-n-methyl-carbamates n-sulfenyles, leur procede de preparation et leur application
BE792155A (fr) Nouveaux derives de l'adenosine et leur procede de production
BE815742A (fr) Nouveaux derives d'acide prostanoique et leur procede de preparation
BE819890A (fr) Nouveaux derives d'acide pyrazolyloxyacetique et leur procede de preparation
FR2308620A1 (fr) Procede de preparation de nouveaux derives d'azetidinone
BE831855A (fr) Nouveaux derives d'oxyphenylbutazone et leur procede de preparation
BE797563A (fr) Nouveaux derives de l'acetamidine et leur procede de preparation ainsi que les compositions therapeutiques les contenant
FR2299859A1 (fr) Derives d'acide glycyrrhetinique, leur procede de preparation et leur application
BE821893A (fr) Derives d'adenine et leur procede de preparation
FR2330675A1 (fr) Nouveaux derives d'isothiouree et leur procede de preparation
BE848627A (fr) Derives substitues d'aminobenzaldehydes et leur procede de preparation,
BE822766A (fr) Nouveaux derives d'amides alpha-aminoxycarboxyliques substitueset leur procede de preparation