BE876042A - Nouvelles 4-(quinoleinylaminobenzoyl) piperidines et composition pharmaceutique les contenant - Google Patents
Nouvelles 4-(quinoleinylaminobenzoyl) piperidines et composition pharmaceutique les contenantInfo
- Publication number
- BE876042A BE876042A BE0/194994A BE194994A BE876042A BE 876042 A BE876042 A BE 876042A BE 0/194994 A BE0/194994 A BE 0/194994A BE 194994 A BE194994 A BE 194994A BE 876042 A BE876042 A BE 876042A
- Authority
- BE
- Belgium
- Prior art keywords
- quinoleinylaminobenzoyl
- piperidines
- news
- pharmaceutical composition
- composition containing
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 150000003053 piperidines Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US05/903,088 US4166853A (en) | 1978-05-05 | 1978-05-05 | Antihypertensive 7-trifluoromethyl-4-aminoquinolones |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BE876042A true BE876042A (fr) | 1979-11-05 |
Family
ID=25416923
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BE0/194994A BE876042A (fr) | 1978-05-05 | 1979-05-04 | Nouvelles 4-(quinoleinylaminobenzoyl) piperidines et composition pharmaceutique les contenant |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US4166853A (fr) |
| JP (1) | JPS54145676A (fr) |
| AU (1) | AU521628B2 (fr) |
| BE (1) | BE876042A (fr) |
| DE (1) | DE2914511A1 (fr) |
| FR (1) | FR2424917A1 (fr) |
| GB (1) | GB2021103B (fr) |
| IT (1) | IT1113370B (fr) |
| NL (1) | NL7903437A (fr) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4886795A (en) * | 1984-06-20 | 1989-12-12 | Schachar Ronald A | Treatment and prevention of retinal edema with dopaminergic antagonists |
| US4624957A (en) * | 1984-06-20 | 1986-11-25 | Schachar Ronald A | Treatment and prevention of retinal edema with dopaminergic antagonists |
| US4886815A (en) * | 1984-06-20 | 1989-12-12 | Schachar Ronald A | Treatment and prevention of retinal edema with dopaminergic antagonists |
| PH22302A (en) * | 1985-02-11 | 1988-07-22 | Fujisawa Pharmaceutical Co | Piperidine compounds |
| AU7195694A (en) * | 1993-07-19 | 1995-02-20 | Fujisawa Pharmaceutical Co., Ltd. | Benzimidazole derivatives useful as dopamine receptor antagonist, 5-ht receptor agonist or alpha1 receptor antagonist |
| KR20010113007A (ko) * | 2000-06-15 | 2001-12-24 | 주정호 | 항암제로서 유용한 n-치환된 피페리디닐우레아 유도체 및그의 제조방법 |
| GB0308333D0 (en) * | 2003-04-10 | 2003-05-14 | Glaxo Group Ltd | Novel compounds |
| US20060293298A1 (en) * | 2003-04-10 | 2006-12-28 | Bamford Mark J | Compounds |
| US7879880B2 (en) * | 2005-12-21 | 2011-02-01 | Schering Corporation | Substituted aniline derivatives useful as histamine H3 antagonists |
| EP1994022A2 (fr) * | 2006-03-15 | 2008-11-26 | Wyeth a Corporation of the State of Delaware | Azacyclylamines avec substitution n en tant qu'antagonistes de l'histamine-3 |
| CN101432261A (zh) * | 2006-05-19 | 2009-05-13 | 惠氏公司 | 作为组织胺-3拮抗剂的n-苯甲酰基-吡咯烷-3-基胺和n-苄基-吡咯烷-3-基胺 |
| PE20081152A1 (es) * | 2006-10-06 | 2008-08-10 | Wyeth Corp | Azaciclilaminas n-sustituidas como antagonistas de histamina-3 |
| CN101778838A (zh) * | 2007-05-24 | 2010-07-14 | 惠氏有限责任公司 | 作为组胺-3拮抗剂的氮杂环基苯甲酰胺衍生物 |
| CA2693138A1 (fr) | 2007-07-16 | 2009-01-22 | Wyeth Llc | Derives d'aminoalkylazole en tant qu'antagonistes d'histamine-3 |
| WO2009036144A1 (fr) * | 2007-09-12 | 2009-03-19 | Wyeth | Dérivés d'isoquinolinyle et d'isoindolinyle convenant comme antagonistes de l'histamine-3 |
| TW200918062A (en) * | 2007-09-12 | 2009-05-01 | Wyeth Corp | Azacyclylisoquinolinone and-isoindolinone derivatives as histamine-3 antagonists |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BE754586A (fr) * | 1969-08-08 | 1971-02-08 | Upjohn Co | Preparations pharmaceutiques a base de p-(4-quinolylamino) benzamide etleur utilisation |
| US3875165A (en) * | 1973-02-22 | 1975-04-01 | Wyeth John & Brother Ltd | (4-Quinolylamino)-(N-piperidyl)benzamides and N-{8 (quinolylamino)-benzoyl{9 piperidines |
| US3971787A (en) * | 1973-02-05 | 1976-07-27 | John Wyeth & Brother Limited | (4-Quinolylamino)benzamides |
| US4025629A (en) * | 1974-01-07 | 1977-05-24 | The Upjohn Company | P-(trifluoromethylquinolylamino)benzamides, pharmaceutical dosage forms and method of treatment |
-
1978
- 1978-05-05 US US05/903,088 patent/US4166853A/en not_active Expired - Lifetime
-
1979
- 1979-04-10 DE DE19792914511 patent/DE2914511A1/de not_active Ceased
- 1979-04-23 IT IT22088/79A patent/IT1113370B/it active
- 1979-04-24 AU AU46421/79A patent/AU521628B2/en not_active Ceased
- 1979-04-26 GB GB7914581A patent/GB2021103B/en not_active Expired
- 1979-05-02 NL NL7903437A patent/NL7903437A/xx not_active Application Discontinuation
- 1979-05-02 JP JP5356579A patent/JPS54145676A/ja active Pending
- 1979-05-04 BE BE0/194994A patent/BE876042A/fr not_active IP Right Cessation
- 1979-05-04 FR FR7911262A patent/FR2424917A1/fr active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| NL7903437A (nl) | 1979-11-07 |
| IT1113370B (it) | 1986-01-20 |
| JPS54145676A (en) | 1979-11-14 |
| GB2021103B (en) | 1982-08-11 |
| AU521628B2 (en) | 1982-04-22 |
| FR2424917A1 (fr) | 1979-11-30 |
| AU4642179A (en) | 1979-11-08 |
| US4166853A (en) | 1979-09-04 |
| DE2914511A1 (de) | 1979-11-08 |
| FR2424917B1 (fr) | 1983-01-14 |
| GB2021103A (en) | 1979-11-28 |
| IT7922088A0 (it) | 1979-04-23 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RE | Patent lapsed |
Owner name: THE UPJOHN CY Effective date: 19880531 |