BE876042A - Nouvelles 4-(quinoleinylaminobenzoyl) piperidines et composition pharmaceutique les contenant - Google Patents

Nouvelles 4-(quinoleinylaminobenzoyl) piperidines et composition pharmaceutique les contenant

Info

Publication number
BE876042A
BE876042A BE0/194994A BE194994A BE876042A BE 876042 A BE876042 A BE 876042A BE 0/194994 A BE0/194994 A BE 0/194994A BE 194994 A BE194994 A BE 194994A BE 876042 A BE876042 A BE 876042A
Authority
BE
Belgium
Prior art keywords
quinoleinylaminobenzoyl
piperidines
news
pharmaceutical composition
composition containing
Prior art date
Application number
BE0/194994A
Other languages
English (en)
Inventor
J Mccall
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of BE876042A publication Critical patent/BE876042A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BE0/194994A 1978-05-05 1979-05-04 Nouvelles 4-(quinoleinylaminobenzoyl) piperidines et composition pharmaceutique les contenant BE876042A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/903,088 US4166853A (en) 1978-05-05 1978-05-05 Antihypertensive 7-trifluoromethyl-4-aminoquinolones

Publications (1)

Publication Number Publication Date
BE876042A true BE876042A (fr) 1979-11-05

Family

ID=25416923

Family Applications (1)

Application Number Title Priority Date Filing Date
BE0/194994A BE876042A (fr) 1978-05-05 1979-05-04 Nouvelles 4-(quinoleinylaminobenzoyl) piperidines et composition pharmaceutique les contenant

Country Status (9)

Country Link
US (1) US4166853A (fr)
JP (1) JPS54145676A (fr)
AU (1) AU521628B2 (fr)
BE (1) BE876042A (fr)
DE (1) DE2914511A1 (fr)
FR (1) FR2424917A1 (fr)
GB (1) GB2021103B (fr)
IT (1) IT1113370B (fr)
NL (1) NL7903437A (fr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4624957A (en) * 1984-06-20 1986-11-25 Schachar Ronald A Treatment and prevention of retinal edema with dopaminergic antagonists
US4886815A (en) * 1984-06-20 1989-12-12 Schachar Ronald A Treatment and prevention of retinal edema with dopaminergic antagonists
US4886795A (en) * 1984-06-20 1989-12-12 Schachar Ronald A Treatment and prevention of retinal edema with dopaminergic antagonists
PH22302A (en) * 1985-02-11 1988-07-22 Fujisawa Pharmaceutical Co Piperidine compounds
WO1995003298A1 (fr) * 1993-07-19 1995-02-02 Fujisawa Pharmaceutical Co., Ltd. DERIVES BENZIMIDAZOLIQUES UTILISABLES COMME AGONISTE DU RECEPTEUR DOPAMINERGIQUE, ANTAGONISTE DU RECEPTEUR SEROTONINERGIQUE, OU ANTAGONISTE DU RECEPTEUR α¿1?
KR20010113007A (ko) * 2000-06-15 2001-12-24 주정호 항암제로서 유용한 n-치환된 피페리디닐우레아 유도체 및그의 제조방법
GB0308333D0 (en) * 2003-04-10 2003-05-14 Glaxo Group Ltd Novel compounds
US20060293298A1 (en) * 2003-04-10 2006-12-28 Bamford Mark J Compounds
EP1966143A2 (fr) * 2005-12-21 2008-09-10 Schering Corporation Derives substitues de l'aniline utilisables en tant qu'antagonistes de l'histamine h3
EP1994022A2 (fr) * 2006-03-15 2008-11-26 Wyeth a Corporation of the State of Delaware Azacyclylamines avec substitution n en tant qu'antagonistes de l'histamine-3
EP2027086B1 (fr) * 2006-05-19 2011-11-16 Wyeth LLC N-benzoyl-pyrrolidin-3-yl amines comme antagonistes de l'histamine-3
PE20081152A1 (es) * 2006-10-06 2008-08-10 Wyeth Corp Azaciclilaminas n-sustituidas como antagonistas de histamina-3
KR20100020487A (ko) * 2007-05-24 2010-02-22 와이어쓰 엘엘씨 히스타민-3 길항제로서 아자시클릴벤즈아미드 유도체
WO2009012252A1 (fr) 2007-07-16 2009-01-22 Wyeth Dérivés d'aminoalkylazole en tant qu'antagonistes d'histamine-3
TW200918062A (en) * 2007-09-12 2009-05-01 Wyeth Corp Azacyclylisoquinolinone and-isoindolinone derivatives as histamine-3 antagonists
WO2009036144A1 (fr) * 2007-09-12 2009-03-19 Wyeth Dérivés d'isoquinolinyle et d'isoindolinyle convenant comme antagonistes de l'histamine-3

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE754586A (fr) * 1969-08-08 1971-02-08 Upjohn Co Preparations pharmaceutiques a base de p-(4-quinolylamino) benzamide etleur utilisation
US3875165A (en) * 1973-02-22 1975-04-01 Wyeth John & Brother Ltd (4-Quinolylamino)-(N-piperidyl)benzamides and N-{8 (quinolylamino)-benzoyl{9 piperidines
US3971787A (en) * 1973-02-05 1976-07-27 John Wyeth & Brother Limited (4-Quinolylamino)benzamides
US4025629A (en) * 1974-01-07 1977-05-24 The Upjohn Company P-(trifluoromethylquinolylamino)benzamides, pharmaceutical dosage forms and method of treatment

Also Published As

Publication number Publication date
IT7922088A0 (it) 1979-04-23
NL7903437A (nl) 1979-11-07
AU521628B2 (en) 1982-04-22
DE2914511A1 (de) 1979-11-08
IT1113370B (it) 1986-01-20
JPS54145676A (en) 1979-11-14
GB2021103A (en) 1979-11-28
US4166853A (en) 1979-09-04
GB2021103B (en) 1982-08-11
FR2424917B1 (fr) 1983-01-14
AU4642179A (en) 1979-11-08
FR2424917A1 (fr) 1979-11-30

Similar Documents

Publication Publication Date Title
LU81349A1 (fr) Nouveaux aminothiazoles et composition pharmaceutique les contenant
BE876042A (fr) Nouvelles 4-(quinoleinylaminobenzoyl) piperidines et composition pharmaceutique les contenant
BE877596A (fr) Nouvelles oxybenzylidene bornanones, procede pour leur preparation et compositions cosmetiques les contenant
LU80795A1 (fr) Nouveaux derives de thienohydantoine et composition pharmaceutique les contenant
BE867727A (fr) Nouveaux composes de phtalazine et composition pharmaceutique les contenant
FR2430410B1 (fr) Phenethanolamines et compositions pharmaceutiques en contenant
BE880065A (fr) Nouvelles spiro-polycyclo-imidazolidinediones et composition pharmaceutique les contenant
BE892805A (fr) Cycloalcanes substitues et compositions pharmaceutiques les contenant
BE870402A (fr) Nouveaux phenols a substituant hydroxyalkyle ou oxoalkyle et composition pharmaceutique les contenant
BE841048A (fr) Nouvelles matieres aromatiques, leur preparation et compositions de parfums en contenant
BE879472A (fr) Composition pharmaceutique contenant des 3,4-dihydro-3-oxo-2-quinoxalines
BE869166A (fr) Nouvelles 4-pyrones substituees en positions 2, 3 et 6 et medicament les contenant
FR2349585A1 (fr) Nouveau derive de xanthine et composition pharmaceutique le contenant
BE788280A (fr) Nouvelles 1-(3-trifluoro-methyl-phenyl)-4-((amido cyclique)- alkyl) piperazines et composition pharmaceutique les contenant
FR2450814B1 (fr) 24,24-difluoro-25-hydroxycholecalciferol et composition pharmaceutique renfermant ce produit
FR2528425B1 (fr) 1,4-dihydropyridines et composition pharmaceutique les contenant
FR2331339A1 (fr) Nouveaux composes heterocycliques et composition pharmaceutique les contenant
EP0018417A4 (fr) Nouveaux derives de piperidine et compositions pharmaceutiques les contenant.
FR2329281A1 (fr) Nouveaux 6,8-dioxamorphinanes n-substitues et composition pharmaceutique les contenant
BE884530A (fr) Nouveaux hexahydro-trans-pyrido-indoles et composition pharmaceutique les contenant
BE883859A (fr) Nouveaux pyridylaminotriazoles et composition pharmaceutique les contenant
BE888963A (fr) Compositions cardiotoniques contenant des aminophenylpyridines, nouvelles aminophenylpyridines et leur preparation
FR2343477A1 (fr) Nouvelles phenylpyridylhydantoines substituees et medicament les contenant
BE857535A (fr) Nouvelles organoprostaglandines et medicament les contenant
BE882443A (fr) Quinolones et compositions therapeutiques les contenant

Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: THE UPJOHN CY

Effective date: 19880531