BE876042A - Nouvelles 4-(quinoleinylaminobenzoyl) piperidines et composition pharmaceutique les contenant - Google Patents

Nouvelles 4-(quinoleinylaminobenzoyl) piperidines et composition pharmaceutique les contenant

Info

Publication number
BE876042A
BE876042A BE0/194994A BE194994A BE876042A BE 876042 A BE876042 A BE 876042A BE 0/194994 A BE0/194994 A BE 0/194994A BE 194994 A BE194994 A BE 194994A BE 876042 A BE876042 A BE 876042A
Authority
BE
Belgium
Prior art keywords
quinoleinylaminobenzoyl
piperidines
news
pharmaceutical composition
composition containing
Prior art date
Application number
BE0/194994A
Other languages
English (en)
Inventor
J Mccall
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of BE876042A publication Critical patent/BE876042A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BE0/194994A 1978-05-05 1979-05-04 Nouvelles 4-(quinoleinylaminobenzoyl) piperidines et composition pharmaceutique les contenant BE876042A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/903,088 US4166853A (en) 1978-05-05 1978-05-05 Antihypertensive 7-trifluoromethyl-4-aminoquinolones

Publications (1)

Publication Number Publication Date
BE876042A true BE876042A (fr) 1979-11-05

Family

ID=25416923

Family Applications (1)

Application Number Title Priority Date Filing Date
BE0/194994A BE876042A (fr) 1978-05-05 1979-05-04 Nouvelles 4-(quinoleinylaminobenzoyl) piperidines et composition pharmaceutique les contenant

Country Status (9)

Country Link
US (1) US4166853A (fr)
JP (1) JPS54145676A (fr)
AU (1) AU521628B2 (fr)
BE (1) BE876042A (fr)
DE (1) DE2914511A1 (fr)
FR (1) FR2424917A1 (fr)
GB (1) GB2021103B (fr)
IT (1) IT1113370B (fr)
NL (1) NL7903437A (fr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4886795A (en) * 1984-06-20 1989-12-12 Schachar Ronald A Treatment and prevention of retinal edema with dopaminergic antagonists
US4624957A (en) * 1984-06-20 1986-11-25 Schachar Ronald A Treatment and prevention of retinal edema with dopaminergic antagonists
US4886815A (en) * 1984-06-20 1989-12-12 Schachar Ronald A Treatment and prevention of retinal edema with dopaminergic antagonists
PH22302A (en) * 1985-02-11 1988-07-22 Fujisawa Pharmaceutical Co Piperidine compounds
AU7195694A (en) * 1993-07-19 1995-02-20 Fujisawa Pharmaceutical Co., Ltd. Benzimidazole derivatives useful as dopamine receptor antagonist, 5-ht receptor agonist or alpha1 receptor antagonist
KR20010113007A (ko) * 2000-06-15 2001-12-24 주정호 항암제로서 유용한 n-치환된 피페리디닐우레아 유도체 및그의 제조방법
GB0308333D0 (en) * 2003-04-10 2003-05-14 Glaxo Group Ltd Novel compounds
US20060293298A1 (en) * 2003-04-10 2006-12-28 Bamford Mark J Compounds
US7879880B2 (en) * 2005-12-21 2011-02-01 Schering Corporation Substituted aniline derivatives useful as histamine H3 antagonists
EP1994022A2 (fr) * 2006-03-15 2008-11-26 Wyeth a Corporation of the State of Delaware Azacyclylamines avec substitution n en tant qu'antagonistes de l'histamine-3
CN101432261A (zh) * 2006-05-19 2009-05-13 惠氏公司 作为组织胺-3拮抗剂的n-苯甲酰基-吡咯烷-3-基胺和n-苄基-吡咯烷-3-基胺
PE20081152A1 (es) * 2006-10-06 2008-08-10 Wyeth Corp Azaciclilaminas n-sustituidas como antagonistas de histamina-3
CN101778838A (zh) * 2007-05-24 2010-07-14 惠氏有限责任公司 作为组胺-3拮抗剂的氮杂环基苯甲酰胺衍生物
CA2693138A1 (fr) 2007-07-16 2009-01-22 Wyeth Llc Derives d'aminoalkylazole en tant qu'antagonistes d'histamine-3
WO2009036144A1 (fr) * 2007-09-12 2009-03-19 Wyeth Dérivés d'isoquinolinyle et d'isoindolinyle convenant comme antagonistes de l'histamine-3
TW200918062A (en) * 2007-09-12 2009-05-01 Wyeth Corp Azacyclylisoquinolinone and-isoindolinone derivatives as histamine-3 antagonists

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE754586A (fr) * 1969-08-08 1971-02-08 Upjohn Co Preparations pharmaceutiques a base de p-(4-quinolylamino) benzamide etleur utilisation
US3875165A (en) * 1973-02-22 1975-04-01 Wyeth John & Brother Ltd (4-Quinolylamino)-(N-piperidyl)benzamides and N-{8 (quinolylamino)-benzoyl{9 piperidines
US3971787A (en) * 1973-02-05 1976-07-27 John Wyeth & Brother Limited (4-Quinolylamino)benzamides
US4025629A (en) * 1974-01-07 1977-05-24 The Upjohn Company P-(trifluoromethylquinolylamino)benzamides, pharmaceutical dosage forms and method of treatment

Also Published As

Publication number Publication date
NL7903437A (nl) 1979-11-07
IT1113370B (it) 1986-01-20
JPS54145676A (en) 1979-11-14
GB2021103B (en) 1982-08-11
AU521628B2 (en) 1982-04-22
FR2424917A1 (fr) 1979-11-30
AU4642179A (en) 1979-11-08
US4166853A (en) 1979-09-04
DE2914511A1 (de) 1979-11-08
FR2424917B1 (fr) 1983-01-14
GB2021103A (en) 1979-11-28
IT7922088A0 (it) 1979-04-23

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: THE UPJOHN CY

Effective date: 19880531