BG20348A3 - Метод за получаване на 4-субституирани 1-(4,4-диарил-бутил) пиперидини - Google Patents

Метод за получаване на 4-субституирани 1-(4,4-диарил-бутил) пиперидини

Info

Publication number
BG20348A3
BG20348A3 BG021601A BG2160172A BG20348A3 BG 20348 A3 BG20348 A3 BG 20348A3 BG 021601 A BG021601 A BG 021601A BG 2160172 A BG2160172 A BG 2160172A BG 20348 A3 BG20348 A3 BG 20348A3
Authority
BG
Bulgaria
Prior art keywords
piperidines
diaryl
butyl
substituted
preparation
Prior art date
Application number
BG021601A
Other languages
Bulgarian (bg)
English (en)
Inventor
Marcel Janssen
Henri Dhaen
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of BG20348A3 publication Critical patent/BG20348A3/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/26—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D307/30—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D307/32—Oxygen atoms
    • C07D307/33—Oxygen atoms in position 2, the oxygen atom being in its keto or unsubstituted enol form
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C57/00—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
    • C07C57/52—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms containing halogen
    • C07C57/58—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms containing halogen containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C57/00—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
    • C07C57/64—Acyl halides
    • C07C57/72—Acyl halides containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40—Oxygen atoms
    • C07D211/44—Oxygen atoms attached in position 4
    • C07D211/52—Oxygen atoms attached in position 4 having an aryl radical as the second substituent in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
BG021601A 1971-11-25 1972-10-12 Метод за получаване на 4-субституирани 1-(4,4-диарил-бутил) пиперидини BG20348A3 (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP9485771A JPS5527915B2 (2) 1971-11-25 1971-11-25

Publications (1)

Publication Number Publication Date
BG20348A3 true BG20348A3 (bg) 1975-11-05

Family

ID=14121686

Family Applications (2)

Application Number Title Priority Date Filing Date
BG021601A BG20348A3 (bg) 1971-11-25 1972-10-12 Метод за получаване на 4-субституирани 1-(4,4-диарил-бутил) пиперидини
BG024007A BG20349A3 (bg) 1971-11-25 1972-10-12 Метод за получаване на 1(4,4-бис (р-флуор-фенил) бутил)-4-пиперидил) -2- бензимидазолинон

Family Applications After (1)

Application Number Title Priority Date Filing Date
BG024007A BG20349A3 (bg) 1971-11-25 1972-10-12 Метод за получаване на 1(4,4-бис (р-флуор-фенил) бутил)-4-пиперидил) -2- бензимидазолинон

Country Status (14)

Country Link
JP (1) JPS5527915B2 (2)
AR (2) AR198393A1 (2)
BG (2) BG20348A3 (2)
CA (1) CA983503A (2)
CH (1) CH579048A5 (2)
CS (1) CS168014B2 (2)
ES (1) ES408926A1 (2)
FR (1) FR2161007A1 (2)
HU (1) HU165208B (2)
IL (1) IL40917A (2)
NL (1) NL7214913A (2)
RO (2) RO63063A (2)
SU (1) SU462333A3 (2)
YU (1) YU35120B (2)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4082755A (en) * 1977-02-14 1978-04-04 Janssen Pharmaceutica N.V. 1-[(Diarylmethyl)aminoalkyl]piperidimes
CN106187863A (zh) * 2016-07-15 2016-12-07 湖南中南制药有限责任公司 五氟利多的制备方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE633495A (2) * 1962-06-13

Also Published As

Publication number Publication date
HU165208B (2) 1974-07-27
NL7214913A (2) 1973-05-29
RO63063A (fr) 1978-07-15
ES408926A1 (es) 1976-03-01
YU291672A (en) 1980-03-15
FR2161007A1 (en) 1973-07-06
SU462333A3 (ru) 1975-02-28
FR2161007B1 (2) 1976-03-05
RO62760A (fr) 1978-02-15
AR198393A1 (es) 1974-06-21
IL40917A0 (en) 1973-01-30
CA983503A (en) 1976-02-10
JPS5527915B2 (2) 1980-07-24
BG20349A3 (bg) 1975-11-05
JPS4860092A (2) 1973-08-23
AR199497A1 (es) 1974-09-09
IL40917A (en) 1976-10-31
CH579048A5 (2) 1976-08-31
CS168014B2 (2) 1976-05-28
YU35120B (en) 1980-09-25

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