BG24669A3 - Метод за получаване на амиди на n-/1-(w-фенилалкил)-пмперидил-4-/ n-(а-пиридил-карбонова киселина и на техните присъединителни с киселина соли - Google Patents

Метод за получаване на амиди на n-/1-(w-фенилалкил)-пмперидил-4-/ n-(а-пиридил-карбонова киселина и на техните присъединителни с киселина соли

Info

Publication number: BG24669A3
Authority: BG; Bulgaria
Prior art keywords: acid; pmperidyl; phenylalkyl; pyridyl; amides
Prior art date: 1973-08-20

Application number

BG027507A

Other languages

Bulgarian (bg)

English (en)

Inventor

Adolf Langbein

Herbert Merz

Gerhard Walther

Original Assignee

C.H.Boehringer Sohn

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1973-08-20

Filing date

1974-08-16

Publication date

1978-04-12

1974-08-16 Application filed by C.H.Boehringer Sohn filed Critical C.H.Boehringer Sohn

1978-04-12 Publication of BG24669A3 publication Critical patent/BG24669A3/xx

Links

150000001408 amides Chemical class 0.000 title 1
150000003839 salts Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C07D211/58—Nitrogen atoms attached in position 4

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Other In-Based Heterocyclic Compounds (AREA)
Hydrogenated Pyridines (AREA)

BG027507A 1973-08-20 1974-08-16 Метод за получаване на амиди на n-/1-(w-фенилалкил)-пмперидил-4-/ n-(а-пиридил-карбонова киселина и на техните присъединителни с киселина соли BG24669A3 (bg)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE2341965A DE2341965C3 (de)	1973-08-20	1973-08-20	4- [N- (o-PyridyD- N-acyl] -aminolphenäthylpiperidine, Verfahren zu deren Herstellung sowie deren Verwendung bei der Bekämpfung von Schmerzzuständen

Publications (1)

Publication Number	Publication Date
BG24669A3 true BG24669A3 (bg)	1978-04-12

Family

ID=5890196

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BG027507A BG24669A3 (bg)	1973-08-20	1974-08-16	Метод за получаване на амиди на n-/1-(w-фенилалкил)-пмперидил-4-/ n-(а-пиридил-карбонова киселина и на техните присъединителни с киселина соли

Country Status (26)

Country	Link
US (1)	US3933832A (cs)
JP (1)	JPS5049285A (cs)
AT (2)	AT334900B (cs)
BE (1)	BE818989A (cs)
BG (1)	BG24669A3 (cs)
CA (1)	CA1041513A (cs)
CH (2)	CH603631A5 (cs)
CS (2)	CS181767B2 (cs)
DD (1)	DD114260A5 (cs)
DE (1)	DE2341965C3 (cs)
DK (1)	DK141097C (cs)
ES (2)	ES429221A1 (cs)
FI (1)	FI57749C (cs)
FR (1)	FR2241314B1 (cs)
GB (1)	GB1468283A (cs)
HU (1)	HU167563B (cs)
IE (1)	IE40511B1 (cs)
IL (1)	IL45494A (cs)
NL (1)	NL7410989A (cs)
NO (1)	NO140594C (cs)
PH (1)	PH11999A (cs)
PL (2)	PL91562B1 (cs)
RO (2)	RO63458A (cs)
SE (1)	SE402285B (cs)
SU (2)	SU504480A3 (cs)
ZA (1)	ZA745306B (cs)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4191683A (en) *	1975-05-28	1980-03-04	Ciba-Geigy Corporation	Derivatives of 4-aminopiperidine as stabilizers for polymers
US4225606A (en) *	1975-09-23	1980-09-30	Janssen Pharmaceutica N.V.	N-Aryl-N-(1-L-4-piperidinyl)arylacetamides
US4791112A (en) *	1987-02-02	1988-12-13	The Boc Group, Inc.	N-heterocyclic-N-(4-piperidyl)amides and pharmaceutical compositions and methods employing such compounds
USRE34201E (en) *	1989-04-20	1993-03-23	Anaquest, Inc.	N-aryl-N-[4-(1-heterocyclicalkyl)piperidinyl]amides and pharmaceutical compositions and methods employing such compounds
US7053089B2 (en)	2001-02-23	2006-05-30	Merck & Co., Inc.	N-substituted nonaryl-heterocyclic NMDA/NR2B antagonists
US20040142013A1 (en) *	2001-07-13	2004-07-22	Flow Focusing, Inc.	Implantable orthopedic surgical devices with controlled release antimicrobial component
US20030055075A1 (en) *	2001-07-13	2003-03-20	Rubsamen Reid M.	Programmable controlled release injectable opioid formulation
US20070254008A1 (en) *	2001-07-13	2007-11-01	Flow Focusing, Inc.	Antibiotic formulation and method of treatment
US20060263401A1 (en) *	2001-07-13	2006-11-23	Flow Focusing, Inc.	Formulation and Method for Preventing Infection
US20070254009A1 (en) *	2001-07-13	2007-11-01	Flow Focusing, Inc.	Antibiotic/bone morphogenic protein formulation and method of treatment
US7592360B2 (en) *	2003-06-04	2009-09-22	Merck & Co., Inc.	3-fluoro-piperidines as NMDA/NR2B antagonists
JO2769B1 (en) *	2005-10-26	2014-03-15	جانسين فارماسوتيكا ان. في	Rapid decomposition of physiologically antagonistic agents of the 2-dopamine receptor
JO2642B1 (en) *	2006-12-08	2012-06-17	جانسين فارماسوتيكا ان. في	Dopamine 2 receptor antagonists are rapidly hydrolyzed
JO2849B1 (en) *	2007-02-13	2015-03-15	جانسين فارماسوتيكا ان. في	Dopamine 2 receptor antagonists are rapidly hydrolyzed
RS52518B (sr) *	2007-04-23	2013-04-30	Janssen Pharmaceutica N.V.	Derivati 4-alkoksipiridazina kao brzo disocirajući dopamin 2 receptorski antagonisti
RU2489431C2 (ru) *	2007-04-23	2013-08-10	Янссен Фармацевтика Н.В.	Тиа(диа)золы как быстро диссоциирующие антагонисты рецептора допамина 2
CN101663291A (zh) *	2007-04-23	2010-03-03	詹森药业有限公司	作为快速离解的多巴胺2受体拮抗剂的吡啶衍生物
JP5417439B2 (ja) *	2008-07-03	2014-02-12	ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ	５−ｈｔ６受容体アンタゴニストとしての置換された６−（１−ピペラジニル）−ピリダジン類
LT2307374T (lt) *	2008-07-31	2017-04-25	Janssen Pharmaceutica Nv	Piperazin-1-il-trifluormetil-pakeistieji piridinai kaip greitai disocijuojantys dopamino 2 receptoriaus antagonistai

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE1232147B (de) *	1961-04-13	1967-01-12	Bayer Ag	Verfahren zur Herstellung von acylierten N-(Alkylaminoalkyl)-aminopyridinen
BE623427A (cs) *	1961-10-10
US3141823A (en) *	1962-09-04	1964-07-21	Res Lab Dr C Janssen N V	Method for producing analgesia
IL25840A (en) *	1965-07-24	1969-12-31	Bayer Ag	Optically active pyridine derivatives and their production

1973
- 1973-08-20 DE DE2341965A patent/DE2341965C3/de not_active Expired
1974
- 1974-07-31 CS CS7400005454A patent/CS181767B2/cs unknown
- 1974-07-31 CS CS7400005455A patent/CS182263B2/cs unknown
- 1974-08-07 FI FI2349/74A patent/FI57749C/fi active
- 1974-08-08 AT AT651274A patent/AT334900B/de not_active IP Right Cessation
- 1974-08-08 AT AT651374A patent/AT334901B/de not_active IP Right Cessation
- 1974-08-13 ES ES429221A patent/ES429221A1/es not_active Expired
- 1974-08-13 ES ES429234A patent/ES429234A1/es not_active Expired
- 1974-08-14 US US05/497,455 patent/US3933832A/en not_active Expired - Lifetime
- 1974-08-15 PH PH16171A patent/PH11999A/en unknown
- 1974-08-16 CH CH1119074A patent/CH603631A5/xx not_active IP Right Cessation
- 1974-08-16 BG BG027507A patent/BG24669A3/xx unknown
- 1974-08-16 CH CH1118674A patent/CH603630A5/xx not_active IP Right Cessation
- 1974-08-16 RO RO7400079805A patent/RO63458A/ro unknown
- 1974-08-16 SU SU2055577A patent/SU504480A3/ru active
- 1974-08-16 NL NL7410989A patent/NL7410989A/xx not_active Application Discontinuation
- 1974-08-16 DK DK439974A patent/DK141097C/da active
- 1974-08-16 SU SU2056122A patent/SU507229A3/ru active
- 1974-08-16 RO RO7400079806A patent/RO63050A/ro unknown
- 1974-08-17 HU HUBO1516A patent/HU167563B/hu unknown
- 1974-08-19 GB GB3645574A patent/GB1468283A/en not_active Expired
- 1974-08-19 PL PL1974173565A patent/PL91562B1/pl unknown
- 1974-08-19 ZA ZA00745306A patent/ZA745306B/xx unknown
- 1974-08-19 IL IL45494A patent/IL45494A/en unknown
- 1974-08-19 JP JP49094904A patent/JPS5049285A/ja active Pending
- 1974-08-19 SE SE7410540A patent/SE402285B/xx unknown
- 1974-08-19 BE BE147736A patent/BE818989A/xx unknown
- 1974-08-19 PL PL1974173564A patent/PL91512B1/pl unknown
- 1974-08-19 CA CA207,296A patent/CA1041513A/en not_active Expired
- 1974-08-19 DD DD180589A patent/DD114260A5/xx unknown
- 1974-08-19 NO NO742970A patent/NO140594C/no unknown
- 1974-08-20 IE IE1734/74A patent/IE40511B1/xx unknown
- 1974-08-20 FR FR7428596A patent/FR2241314B1/fr not_active Expired

Also Published As

Publication number	Publication date
SU504480A3 (ru)	1976-02-25
AT334901B (de)	1977-02-10
SE402285B (sv)	1978-06-26
DK439974A (cs)	1975-04-28
CA1041513A (en)	1978-10-31
ZA745306B (en)	1976-04-28
PL91562B1 (cs)	1977-03-31
FI234974A7 (cs)	1975-02-21
NO742970L (cs)	1975-03-17
FR2241314A1 (cs)	1975-03-21
CH603630A5 (cs)	1978-08-31
US3933832A (en)	1976-01-20
IL45494A0 (en)	1974-11-29
FI57749C (fi)	1980-10-10
BE818989A (fr)	1975-02-19
RO63458A (fr)	1978-06-15
NO140594C (no)	1979-10-03
DK141097C (da)	1980-08-18
JPS5049285A (cs)	1975-05-01
HU167563B (cs)	1975-11-28
ES429234A1 (es)	1976-08-16
AU7248974A (en)	1976-02-19
SE7410540L (cs)	1975-02-21
CH603631A5 (cs)	1978-08-31
RO63050A (cs)	1978-05-15
SU507229A3 (ru)	1976-03-15
DE2341965A1 (de)	1975-03-06
CS181767B2 (en)	1978-03-31
DD114260A5 (cs)	1975-07-20
FI57749B (fi)	1980-06-30
GB1468283A (en)	1977-03-23
CS182263B2 (en)	1978-04-28
IE40511L (en)	1975-02-20
ATA651274A (de)	1976-06-15
NL7410989A (nl)	1975-02-24
DE2341965B2 (de)	1978-06-01
PH11999A (en)	1978-10-06
DK141097B (da)	1980-01-14
AT334900B (de)	1977-02-10
PL91512B1 (cs)	1977-02-28
IE40511B1 (en)	1979-06-20
DE2341965C3 (de)	1979-01-25
NO140594B (no)	1979-06-25
FR2241314B1 (cs)	1977-11-10
ES429221A1 (es)	1976-08-16
ATA651374A (de)	1976-06-15
IL45494A (en)	1977-07-31

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