BR0010454A - Composição farmacêutica contendo ciclosporina - Google Patents
Composição farmacêutica contendo ciclosporinaInfo
- Publication number
- BR0010454A BR0010454A BR0010454-0A BR0010454A BR0010454A BR 0010454 A BR0010454 A BR 0010454A BR 0010454 A BR0010454 A BR 0010454A BR 0010454 A BR0010454 A BR 0010454A
- Authority
- BR
- Brazil
- Prior art keywords
- composition containing
- pharmaceutical composition
- pharmaceutical
- compositions
- cyclosporine
- Prior art date
Links
- PMATZTZNYRCHOR-CGLBZJNRSA-N Cyclosporin A Chemical compound CC[C@@H]1NC(=O)[C@H]([C@H](O)[C@H](C)C\C=C\C)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)N(C)C(=O)CN(C)C1=O PMATZTZNYRCHOR-CGLBZJNRSA-N 0.000 title abstract 3
- 108010036949 Cyclosporine Proteins 0.000 title abstract 3
- 229960001265 ciclosporin Drugs 0.000 title abstract 3
- 229930182912 cyclosporin Natural products 0.000 title abstract 3
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 3
- 239000000203 mixture Substances 0.000 abstract 4
- 229930105110 Cyclosporin A Natural products 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 150000001735 carboxylic acids Chemical class 0.000 abstract 1
- 239000003889 eye drop Substances 0.000 abstract 1
- 229940012356 eye drops Drugs 0.000 abstract 1
- 238000009472 formulation Methods 0.000 abstract 1
- 239000007924 injection Substances 0.000 abstract 1
- 238000002347 injection Methods 0.000 abstract 1
- 239000002674 ointment Substances 0.000 abstract 1
- 150000007524 organic acids Chemical class 0.000 abstract 1
- 235000005985 organic acids Nutrition 0.000 abstract 1
- 229920006395 saturated elastomer Polymers 0.000 abstract 1
- 235000003441 saturated fatty acids Nutrition 0.000 abstract 1
- 150000004671 saturated fatty acids Chemical class 0.000 abstract 1
- 239000007901 soft capsule Substances 0.000 abstract 1
- 239000000243 solution Substances 0.000 abstract 1
- 239000000758 substrate Substances 0.000 abstract 1
- 235000021122 unsaturated fatty acids Nutrition 0.000 abstract 1
- 150000004670 unsaturated fatty acids Chemical class 0.000 abstract 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
- A61K38/13—Cyclosporins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
Landscapes
- Health & Medical Sciences (AREA)
- Immunology (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Gastroenterology & Hepatology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Transplantation (AREA)
- Dispersion Chemistry (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
"COMPOSIçãO FARMACêUTICA CONTENDO CICLOSPORINA". A presente invenção tefere-se a composições farmacêuticas compreendendo ciclosporina como ingrediente ativo. é característico das composições que a escolha de um ou uma mistura de dois ou mais selecionados do grupo consistindo de ácidos orgânicos farmacêuticos, tais como ácidos graxos saturados ou insaturados de cadeia média/longa e ácidos carboxílicos substitutivos como componente lipofílico. Com a finalidade de satisfazer o requisito de diferentes formulações, um substrato hidrofílico pode ser feito adicionando adequadamente água ou não. A composição é adequada para cápsulas macias, pomadas, colírios, soluções orais, injeções e assim por diante.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CNB991028481A CN1167462C (zh) | 1999-03-09 | 1999-03-09 | 一种含环孢素的药物组合物 |
| PCT/CN2000/000041 WO2000053212A1 (fr) | 1999-03-09 | 2000-03-02 | Composition pharmaceutique contenant une cyclosporine |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR0010454A true BR0010454A (pt) | 2002-01-08 |
Family
ID=5271009
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0010454-0A BR0010454A (pt) | 1999-03-09 | 2000-03-02 | Composição farmacêutica contendo ciclosporina |
Country Status (7)
| Country | Link |
|---|---|
| KR (1) | KR20010112315A (pt) |
| CN (1) | CN1167462C (pt) |
| AU (1) | AU2792700A (pt) |
| BR (1) | BR0010454A (pt) |
| DE (1) | DE10084344T1 (pt) |
| GB (1) | GB2363572B (pt) |
| WO (1) | WO2000053212A1 (pt) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE60221287D1 (de) * | 2001-11-08 | 2007-08-30 | Atrium Medical Corp | Intraluminale vorrichtung mit einer ein therapeutisches-mittel enthaltenden beschichtung |
| AU2004264958B2 (en) | 2003-08-13 | 2010-04-15 | Biocon, Ltd | Micro-particle fatty acid salt solid dosage formulations for therapeutic agents |
| US9012506B2 (en) | 2004-09-28 | 2015-04-21 | Atrium Medical Corporation | Cross-linked fatty acid-based biomaterials |
| EP1811935B1 (en) | 2004-09-28 | 2016-03-30 | Atrium Medical Corporation | Heat cured gel and method of making |
| US9000040B2 (en) | 2004-09-28 | 2015-04-07 | Atrium Medical Corporation | Cross-linked fatty acid-based biomaterials |
| KR100678829B1 (ko) * | 2004-12-06 | 2007-02-05 | 한미약품 주식회사 | 타크로리무스의 경구용 마이크로에멀젼 조성물 |
| CN100478025C (zh) * | 2005-03-25 | 2009-04-15 | 中国科学院上海药物研究所 | 一种环孢菌素a眼用微乳制剂及其制备方法 |
| US9427423B2 (en) | 2009-03-10 | 2016-08-30 | Atrium Medical Corporation | Fatty-acid based particles |
| US9278161B2 (en) | 2005-09-28 | 2016-03-08 | Atrium Medical Corporation | Tissue-separating fatty acid adhesion barrier |
| CN101502641B (zh) * | 2009-02-23 | 2012-05-02 | 姚定全 | 一种注射给药的环孢素药物组合物 |
| US20110038910A1 (en) | 2009-08-11 | 2011-02-17 | Atrium Medical Corporation | Anti-infective antimicrobial-containing biomaterials |
| US10322213B2 (en) | 2010-07-16 | 2019-06-18 | Atrium Medical Corporation | Compositions and methods for altering the rate of hydrolysis of cured oil-based materials |
| US9867880B2 (en) | 2012-06-13 | 2018-01-16 | Atrium Medical Corporation | Cured oil-hydrogel biomaterial compositions for controlled drug delivery |
| KR101363776B1 (ko) * | 2012-12-21 | 2014-02-17 | 이상필 | 사이클로스포린을 포함하는 투명 점안액 조성물 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9113872D0 (en) * | 1991-06-27 | 1991-08-14 | Sandoz Ag | Improvements in or relating to organic compounds |
| IL102236A0 (en) * | 1991-06-27 | 1993-01-14 | Ltt Inst Co Ltd | Topical preparations containing cyclosporin |
| KR940002128Y1 (ko) * | 1992-04-21 | 1994-04-06 | 배순훈 | 비데오 테이프 레코더의 테이프 로딩장치 |
| US5603951A (en) * | 1994-11-09 | 1997-02-18 | Hanmi Pharm. Ind. Co., Ltd. | Cyclosporin-containing soft capsule compositions |
| KR0167613B1 (ko) * | 1994-12-28 | 1999-01-15 | 한스 루돌프 하우스, 니콜 케르커 | 사이클로스포린-함유 연질캅셀제 조성물 |
| DE19544507B4 (de) * | 1995-11-29 | 2007-11-15 | Novartis Ag | Cyclosporin enthaltende Präparate |
-
1999
- 1999-03-09 CN CNB991028481A patent/CN1167462C/zh not_active Expired - Lifetime
-
2000
- 2000-03-02 DE DE10084344T patent/DE10084344T1/de not_active Withdrawn
- 2000-03-02 WO PCT/CN2000/000041 patent/WO2000053212A1/zh not_active Ceased
- 2000-03-02 GB GB0121845A patent/GB2363572B/en not_active Expired - Lifetime
- 2000-03-02 BR BR0010454-0A patent/BR0010454A/pt not_active Application Discontinuation
- 2000-03-02 AU AU27927/00A patent/AU2792700A/en not_active Abandoned
- 2000-03-02 KR KR1020017011483A patent/KR20010112315A/ko not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| CN1167462C (zh) | 2004-09-22 |
| CN1265920A (zh) | 2000-09-13 |
| AU2792700A (en) | 2000-09-28 |
| GB2363572B (en) | 2004-02-18 |
| KR20010112315A (ko) | 2001-12-20 |
| GB2363572A (en) | 2002-01-02 |
| GB0121845D0 (en) | 2001-10-31 |
| DE10084344T1 (de) | 2002-07-11 |
| WO2000053212A1 (fr) | 2000-09-14 |
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Legal Events
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| B09B | Patent application refused [chapter 9.2 patent gazette] |
Free format text: INDEFIRO O PEDIDO DE ACORDO COM O(S) ARTIGO(S) 8O E 13 DA LPI. |
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| B09B | Patent application refused [chapter 9.2 patent gazette] |
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