BR0109770A - Uso de galantamina para o tratamento do comportamento neuropsiquiátrico associado com a doença de alzheimer - Google Patents
Uso de galantamina para o tratamento do comportamento neuropsiquiátrico associado com a doença de alzheimerInfo
- Publication number
- BR0109770A BR0109770A BR0109770-9A BR0109770A BR0109770A BR 0109770 A BR0109770 A BR 0109770A BR 0109770 A BR0109770 A BR 0109770A BR 0109770 A BR0109770 A BR 0109770A
- Authority
- BR
- Brazil
- Prior art keywords
- alzheimer
- galantamine
- disease
- behavior associated
- treat neuropsychiatric
- Prior art date
Links
- ASUTZQLVASHGKV-JDFRZJQESA-N galanthamine Chemical compound O1C(=C23)C(OC)=CC=C2CN(C)CC[C@]23[C@@H]1C[C@@H](O)C=C2 ASUTZQLVASHGKV-JDFRZJQESA-N 0.000 title abstract 9
- 229960003980 galantamine Drugs 0.000 title abstract 5
- 208000024827 Alzheimer disease Diseases 0.000 title abstract 4
- ASUTZQLVASHGKV-UHFFFAOYSA-N galanthamine hydrochloride Natural products O1C(=C23)C(OC)=CC=C2CN(C)CCC23C1CC(O)C=C2 ASUTZQLVASHGKV-UHFFFAOYSA-N 0.000 title abstract 4
- 208000017667 Chronic Disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 230000000087 stabilizing effect Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical & Material Sciences (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines Containing Plant Substances (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US19425900P | 2000-04-03 | 2000-04-03 | |
| PCT/EP2001/003553 WO2001074339A2 (fr) | 2000-04-03 | 2001-03-28 | Utilisation de la galantamine dans le traitement du comportement neuropsychiatrique associe a la maladie d'alzheimer |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR0109770A true BR0109770A (pt) | 2003-02-04 |
Family
ID=22716898
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0109770-9A BR0109770A (pt) | 2000-04-03 | 2001-03-28 | Uso de galantamina para o tratamento do comportamento neuropsiquiátrico associado com a doença de alzheimer |
Country Status (20)
| Country | Link |
|---|---|
| EP (1) | EP1272192A2 (fr) |
| JP (1) | JP2003528913A (fr) |
| KR (1) | KR20020086911A (fr) |
| CN (1) | CN1430514A (fr) |
| AU (2) | AU2001265844B2 (fr) |
| BG (1) | BG107093A (fr) |
| BR (1) | BR0109770A (fr) |
| CA (1) | CA2310926C (fr) |
| CZ (1) | CZ20023543A3 (fr) |
| EE (1) | EE200200554A (fr) |
| HR (1) | HRP20020778A2 (fr) |
| HU (1) | HUP0300566A3 (fr) |
| IL (1) | IL152061A0 (fr) |
| MX (1) | MXPA02009777A (fr) |
| NO (1) | NO20024746L (fr) |
| PL (1) | PL361272A1 (fr) |
| RU (1) | RU2002129298A (fr) |
| SK (1) | SK15422002A3 (fr) |
| WO (1) | WO2001074339A2 (fr) |
| ZA (1) | ZA200207935B (fr) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6617361B2 (en) * | 1999-11-05 | 2003-09-09 | Be Able, Llc | Behavior chemotherapy |
| ES2293287T3 (es) | 2003-07-25 | 2008-03-16 | F. Hoffmann-La Roche Ag | Combinacion de antagonista de mglur2 y de inhibidor de ache para el tratamiento de trastornos neurologicos agudos y/o cronicos. |
| DE10338544B4 (de) * | 2003-08-19 | 2017-08-31 | Janssen Pharmaceutica N.V. | Buccale Formulierungen des Galanthamins und deren Anwendungen |
| AU2009229372C1 (en) | 2008-03-27 | 2017-02-02 | Chase Pharmaceuticals Corporation | Use and composition for treating dementia |
| WO2013160728A1 (fr) | 2012-04-26 | 2013-10-31 | Alma Mater Studiorum - Universita' Di Bologna | Composés à double ciblage pour le traitement de la maladie d'alzheimer |
| BG66818B1 (bg) * | 2013-03-07 | 2019-01-31 | Berbee Beheer B. V. | Състав на екстракт от hippeastrum papilio за производство на лекарствени средства и хранителни добавки |
| AU2016264228B2 (en) * | 2015-05-18 | 2019-06-13 | Synaptec Development Llc | Galantamine clearance of amyloidß |
| WO2023036105A1 (fr) * | 2021-09-09 | 2023-03-16 | 上海日馨医药科技股份有限公司 | Méthode de traitement d'une maladie neurodégénérative |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4663318A (en) * | 1986-01-15 | 1987-05-05 | Bonnie Davis | Method of treating Alzheimer's disease |
| DE19509663A1 (de) * | 1995-03-17 | 1996-09-19 | Lohmann Therapie Syst Lts | Verfahren zur Isolierung von Galanthamin |
| GB9600080D0 (en) * | 1996-01-04 | 1996-03-06 | Chiroscience Ltd | Resolution process |
| AU1738800A (en) | 1998-11-23 | 2000-06-13 | Bonnie Davis | Dosage formulations for acetylcholinesterase inhibitors |
| AU775914B2 (en) * | 1998-12-24 | 2004-08-19 | Janssen Pharmaceutica N.V. | Controlled release galantamine composition |
| CA2310950C (fr) * | 2000-04-03 | 2005-11-08 | Janssen Pharmaceutica N.V. | Posologie de galantamine efficace qui reduit les effets secondaires |
| CA2310990A1 (fr) * | 2000-04-03 | 2000-10-09 | Michael Pontecorvo | Utilisation de la galantamine pour le traitement de la maladie d'alzheimer; ciblage de la cause sous-jacente de la maladie |
-
2000
- 2000-06-27 CA CA002310926A patent/CA2310926C/fr not_active Expired - Lifetime
-
2001
- 2001-03-28 EP EP01943200A patent/EP1272192A2/fr not_active Withdrawn
- 2001-03-28 RU RU2002129298/14A patent/RU2002129298A/ru not_active Application Discontinuation
- 2001-03-28 PL PL36127201A patent/PL361272A1/xx not_active Application Discontinuation
- 2001-03-28 KR KR1020027011063A patent/KR20020086911A/ko not_active Ceased
- 2001-03-28 SK SK1542-2002A patent/SK15422002A3/sk unknown
- 2001-03-28 AU AU2001265844A patent/AU2001265844B2/en not_active Ceased
- 2001-03-28 BR BR0109770-9A patent/BR0109770A/pt not_active IP Right Cessation
- 2001-03-28 HR HR20020778A patent/HRP20020778A2/xx not_active Application Discontinuation
- 2001-03-28 HU HU0300566A patent/HUP0300566A3/hu unknown
- 2001-03-28 CN CN01807334A patent/CN1430514A/zh active Pending
- 2001-03-28 WO PCT/EP2001/003553 patent/WO2001074339A2/fr not_active Ceased
- 2001-03-28 CZ CZ20023543A patent/CZ20023543A3/cs unknown
- 2001-03-28 EE EEP200200554A patent/EE200200554A/xx unknown
- 2001-03-28 IL IL15206101A patent/IL152061A0/xx unknown
- 2001-03-28 MX MXPA02009777A patent/MXPA02009777A/es unknown
- 2001-03-28 AU AU6584401A patent/AU6584401A/xx active Pending
- 2001-03-28 JP JP2001572084A patent/JP2003528913A/ja not_active Withdrawn
-
2002
- 2002-09-12 BG BG107093A patent/BG107093A/bg unknown
- 2002-10-02 NO NO20024746A patent/NO20024746L/no not_active Application Discontinuation
- 2002-10-02 ZA ZA200207935A patent/ZA200207935B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| RU2002129298A (ru) | 2004-03-27 |
| KR20020086911A (ko) | 2002-11-20 |
| HUP0300566A2 (hu) | 2003-06-28 |
| BG107093A (bg) | 2003-06-30 |
| PL361272A1 (en) | 2004-10-04 |
| AU6584401A (en) | 2001-10-15 |
| WO2001074339A3 (fr) | 2002-09-12 |
| HUP0300566A3 (en) | 2004-10-28 |
| WO2001074339A2 (fr) | 2001-10-11 |
| NO20024746D0 (no) | 2002-10-02 |
| NO20024746L (no) | 2002-11-28 |
| CA2310926A1 (fr) | 2000-10-04 |
| AU2001265844B2 (en) | 2005-04-14 |
| SK15422002A3 (sk) | 2003-04-01 |
| CZ20023543A3 (cs) | 2003-03-12 |
| ZA200207935B (en) | 2004-01-30 |
| EE200200554A (et) | 2004-04-15 |
| MXPA02009777A (es) | 2003-03-27 |
| HRP20020778A2 (en) | 2004-04-30 |
| EP1272192A2 (fr) | 2003-01-08 |
| IL152061A0 (en) | 2003-05-29 |
| CN1430514A (zh) | 2003-07-16 |
| JP2003528913A (ja) | 2003-09-30 |
| CA2310926C (fr) | 2002-10-15 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| BR0012136A (pt) | Inibidores de reabsorção de norepinefrina altamente seletivos e métodos de uso dos mesmos | |
| BR9807673A (pt) | Processos para tratar asma alérgica e dermatite em um humano e composição farmacêutica. | |
| BR0115109A (pt) | Agentes terapêuticos e métodos de uso dos mesmos para a modulação da angiogênese | |
| DK0713701T3 (da) | 2-Brommelatonin til behandling af søvnforstyrrelser | |
| BR0008926A (pt) | Utilização de um extrato de uva, rico ouenriquecido em polifenóis e processo detratamento cosmético do corpo humano | |
| BR0013122A (pt) | Ciclobenzaprina para tratamento de distúrbio de ansiedade generalizado e composições de ciclobenzaprina | |
| WO2002002518A3 (fr) | Composes pour traiter la maladie d'alzheimer | |
| BR0114913A (pt) | Inibidores de metaloproteinase de espiro-pirimidina-2,4,6-triona | |
| BR0111913A (pt) | Análogos de gabapentina para distúrbios do sono | |
| KR970704429A (ko) | 심혈관 질환의 치료를 위한 드롤록시펜의 용도(use of droloxifene for the treatment of cardiovascular diseases) | |
| BR0114392A (pt) | Formulação de vacina, método para produzir uma formulação de vacina, uso de uma preparação de vacina contra rsv dividido, kit para liberação de uma formulação de vacina intranasal, dispositivo de liberação intranasal, e, método para proteger ou tratar um mamìfero susceptìvel a, ou sofrendo de doença causada por rsv | |
| BR0312845A (pt) | Tetratiomolibdato de tetrapropilamÈnio e compostos relacionados para terapias antiangiogênicas | |
| BR9509006A (pt) | Composiçao para aplicaçao tópica na pele composiçao farmacêutica uso de um inibidor de síntese de colesterol e processo para o tratamento mitigaçao ou prevençao de distúrbios de pele | |
| EP0401903A3 (fr) | Utilisation de vanilloides dans le traitement des maladies ou des troubles respiratoires | |
| BR0109770A (pt) | Uso de galantamina para o tratamento do comportamento neuropsiquiátrico associado com a doença de alzheimer | |
| BR0107628A (pt) | l,2-diarilbenzimidazóis para tratamento de doenças que estão associadas a uma ativação microglial | |
| KR890011589A (ko) | 벤즈아미드의 용도 | |
| BR0208405A (pt) | Compostos de diidropirimina substituìdos com ciano e seu uso para tratar doenças | |
| BR9812660A (pt) | Composições e métodos para tratar distúrbios respiratórios | |
| BR0112547A (pt) | Processo para encontrar compostos que sejam adequados para o tratamento e/ou profilaxia de obesidade | |
| BR9813549A (pt) | Processo para prevenção e tratamento de miocárdio afetado por lesão | |
| BR0107960A (pt) | Tratamento de condições alérgicas e inflamatórias | |
| BR9908885A (pt) | Medicamento para a profilaxia e/ou tratamento de mastocarcinoma, compreendendo um inibidor esteróide de aromatase | |
| DE3875349D1 (de) | Glykosaminoglykan zur behandlung von diabetischer mikroangiopathie. | |
| NO990450L (no) | Behandling av sinnslidelser |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE 8A. ANUIDADES. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 DA RPI 2016 DE 25/08/2009 |